FI62310C - Analogifoerfarande foer framstaellning av farmaceutiskt anvaendbara 2-oxo-2h-(1,2,4)-oxadiazolopyrimidin-7-karbamat - Google Patents

Analogifoerfarande foer framstaellning av farmaceutiskt anvaendbara 2-oxo-2h-(1,2,4)-oxadiazolopyrimidin-7-karbamat Download PDF

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Publication number
FI62310C
FI62310C FI780344A FI780344A FI62310C FI 62310 C FI62310 C FI 62310C FI 780344 A FI780344 A FI 780344A FI 780344 A FI780344 A FI 780344A FI 62310 C FI62310 C FI 62310C
Authority
FI
Finland
Prior art keywords
formula
alkyl
piperidine
oxo
benzyl
Prior art date
Application number
FI780344A
Other languages
English (en)
Finnish (fi)
Other versions
FI62310B (fi
FI780344A (fi
Inventor
Jean-Claude Muller
Henri Ramuz
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from AT74577A external-priority patent/AT351037B/de
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of FI780344A publication Critical patent/FI780344A/fi
Publication of FI62310B publication Critical patent/FI62310B/fi
Application granted granted Critical
Publication of FI62310C publication Critical patent/FI62310C/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/08—Vasodilators for multiple indications
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Cardiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
FI780344A 1977-02-04 1978-02-02 Analogifoerfarande foer framstaellning av farmaceutiskt anvaendbara 2-oxo-2h-(1,2,4)-oxadiazolopyrimidin-7-karbamat FI62310C (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
AT74577 1977-02-04
AT74577A AT351037B (de) 1977-02-04 1977-02-04 Verfahren zur herstellung von neuen oxadiazolo- pyrimidinderivaten und deren salzen
LU7778640A LU78640A1 (ja) 1977-02-04 1977-12-05
LU78640 1977-12-05

Publications (3)

Publication Number Publication Date
FI780344A FI780344A (fi) 1978-08-05
FI62310B FI62310B (fi) 1982-08-31
FI62310C true FI62310C (fi) 1982-12-10

Family

ID=25593802

Family Applications (1)

Application Number Title Priority Date Filing Date
FI780344A FI62310C (fi) 1977-02-04 1978-02-02 Analogifoerfarande foer framstaellning av farmaceutiskt anvaendbara 2-oxo-2h-(1,2,4)-oxadiazolopyrimidin-7-karbamat

Country Status (23)

Country Link
US (1) US4150131A (ja)
JP (1) JPS6026115B2 (ja)
AU (1) AU515104B2 (ja)
BE (1) BE863609A (ja)
CA (1) CA1096862A (ja)
CH (1) CH638216A5 (ja)
DE (1) DE2804519A1 (ja)
DK (1) DK50778A (ja)
ES (2) ES466590A1 (ja)
FI (1) FI62310C (ja)
FR (1) FR2383931A1 (ja)
GB (2) GB1566673A (ja)
GR (1) GR71603B (ja)
HU (1) HU178012B (ja)
IE (1) IE46320B1 (ja)
IL (2) IL53926A (ja)
IT (1) IT1092333B (ja)
MC (1) MC1184A1 (ja)
NL (1) NL7801289A (ja)
NO (1) NO780395L (ja)
NZ (1) NZ186335A (ja)
PT (1) PT67615B (ja)
SE (1) SE7801312L (ja)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1103245A (en) * 1978-07-21 1981-06-16 Jean-Claude Muller Process for the manufacture of novel oxadiazolopyrimidine derivatives
NZ190915A (en) * 1978-07-31 1984-07-31 Hoffmann La Roche Oxadiazolotriazine derivatives and pharmaceutical compositions
US4307093A (en) * 1980-06-23 1981-12-22 The Upjohn Company Animal feed and process
US4316901A (en) * 1980-06-23 1982-02-23 The Upjohn Company Animal feed and process
DK148826C (da) * 1980-12-19 1986-03-24 Hoffmann La Roche Analogifremgangsmaade til fremstilling af oxadiazolopyrimidinderivater eller salte deraf med baser og pyrimidinderivat til anvendelse som mellemprodukt ved denne fremgangsmaade
US4411690A (en) * 1981-01-26 1983-10-25 E. I. Du Pont De Nemours & Co. Fused [1,2,4]oxadiazolylidenebenzenesulfonamides and their use as herbicides and plant growth regulants
CH649291A5 (de) * 1982-03-16 1985-05-15 Hoffmann La Roche Dicarbamate.
EP0187854A4 (en) * 1984-07-13 1987-01-22 Gail S Bazzano SUBSTITUTED PYRIMIDINE OXIDES USEFUL FOR PROMOTING HAIR GROWTH.
HU196061B (en) * 1986-07-10 1988-09-28 Richter Gedeon Vegyeszet Process for production of pirimidine-derivatives
LU86547A1 (fr) * 1986-08-07 1988-03-02 Oreal Suspension pour induire et stimuler la croissance des cheveux et diminuer leur chute a base de derives de la pyrimidine

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3382247A (en) * 1965-11-01 1968-05-07 Upjohn Co 6-amino-1, 2-dihydro-1-hydroxy-2-imino-4-phenoxypyrimidines
DE2118261A1 (de) * 1971-04-15 1972-11-02 C.H. Boehringer Sohn, 6507 Ingelheim Neue N-haltige Bicyclen, deren Säureadditionssalze sowie Verfahren zu deren Herstellung
BE786028A (fr) * 1971-07-08 1973-01-08 Boehringer Sohn Ingelheim 2,3-dihydro-oxo-imidazo(1,2-a)-pyrimidines, leurs sels d'addition avec des acides et procedes pour les fabriquer
BE790008A (fr) * 1971-10-15 1973-04-12 Fmc Corp Nouveaux composes herbicides
DE2210633C2 (de) * 1972-03-06 1983-09-22 Bayer Ag, 5090 Leverkusen Kondensierte Pyridinderivate, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende Arzneimittel
DE2252122A1 (de) * 1972-10-24 1974-04-25 Hoechst Ag Oxazolo-chinazoline und verfahren zu ihrer herstellung
DE2253555A1 (de) * 1972-11-02 1974-05-09 Hoechst Ag Oxazolo-pyrimidine und verfahren zu ihrer herstellung
US3910928A (en) * 1974-04-26 1975-10-07 Upjohn Co 3-(Cyanimino)-propionitriles

Also Published As

Publication number Publication date
DK50778A (da) 1978-08-05
JPS6026115B2 (ja) 1985-06-21
IL53926A0 (en) 1978-04-30
IL59713A0 (en) 1980-06-30
NZ186335A (en) 1980-04-28
IL53926A (en) 1980-12-31
IE780198L (en) 1978-08-04
MC1184A1 (fr) 1978-12-22
NL7801289A (nl) 1978-08-08
FR2383931B1 (ja) 1980-07-25
IT7819785A0 (it) 1978-01-30
AU3285878A (en) 1979-08-09
PT67615B (en) 1980-03-03
ES473787A1 (es) 1979-05-16
BE863609A (fr) 1978-08-03
CH638216A5 (de) 1983-09-15
FR2383931A1 (fr) 1978-10-13
HU178012B (en) 1982-02-28
GB1566673A (en) 1980-05-08
ES466590A1 (es) 1978-10-01
GB1566672A (en) 1980-05-08
DE2804519A1 (de) 1978-08-10
JPS5398993A (en) 1978-08-29
CA1096862A (en) 1981-03-03
IE46320B1 (en) 1983-05-04
FI62310B (fi) 1982-08-31
NO780395L (no) 1978-08-07
AU515104B2 (en) 1981-03-19
GR71603B (ja) 1983-06-17
US4150131A (en) 1979-04-17
FI780344A (fi) 1978-08-05
IT1092333B (it) 1985-07-06
SE7801312L (sv) 1978-08-05
DE2804519C2 (ja) 1990-06-13
PT67615A (en) 1978-03-01

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Legal Events

Date Code Title Description
MM Patent lapsed

Owner name: F. HOFFMANN-LA ROCHE & CO.