FI60207C - Foerfarande foer framstaellning av antibiotiskt aktiva 3-imidazo-rifamycinderivat - Google Patents

Foerfarande foer framstaellning av antibiotiskt aktiva 3-imidazo-rifamycinderivat Download PDF

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Publication number
FI60207C
FI60207C FI761392A FI761392A FI60207C FI 60207 C FI60207 C FI 60207C FI 761392 A FI761392 A FI 761392A FI 761392 A FI761392 A FI 761392A FI 60207 C FI60207 C FI 60207C
Authority
FI
Finland
Prior art keywords
formula
filtered
zinc
solution
substituted
Prior art date
Application number
FI761392A
Other languages
English (en)
Finnish (fi)
Other versions
FI761392A (de
FI60207B (fi
Inventor
Leonardo Marsili
Vittorio Rossetti
Carmine Pasqualucci
Original Assignee
Erba Farmitalia
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Erba Farmitalia filed Critical Erba Farmitalia
Publication of FI761392A publication Critical patent/FI761392A/fi
Publication of FI60207B publication Critical patent/FI60207B/fi
Application granted granted Critical
Publication of FI60207C publication Critical patent/FI60207C/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/08—Bridged systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A61P31/06—Antibacterial agents for tuberculosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D498/20—Spiro-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Communicable Diseases (AREA)
  • Veterinary Medicine (AREA)
  • Oncology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pulmonology (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
FI761392A 1975-05-20 1976-05-18 Foerfarande foer framstaellning av antibiotiskt aktiva 3-imidazo-rifamycinderivat FI60207C (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IT515775 1975-05-20
IT05157/75A IT1056271B (it) 1975-05-20 1975-05-20 Prodotti derivati dalle amine aromatiche

Publications (3)

Publication Number Publication Date
FI761392A FI761392A (de) 1976-11-21
FI60207B FI60207B (fi) 1981-08-31
FI60207C true FI60207C (fi) 1981-12-10

Family

ID=11118558

Family Applications (1)

Application Number Title Priority Date Filing Date
FI761392A FI60207C (fi) 1975-05-20 1976-05-18 Foerfarande foer framstaellning av antibiotiskt aktiva 3-imidazo-rifamycinderivat

Country Status (27)

Country Link
US (1) US4226765A (de)
JP (1) JPS5248698A (de)
AR (1) AR213175A1 (de)
AT (1) AT344897B (de)
AU (1) AU497327B2 (de)
BE (1) BE842036A (de)
CA (1) CA1053667A (de)
CH (1) CH625804A5 (de)
CS (1) CS194763B2 (de)
DE (1) DE2622638C2 (de)
DK (1) DK143852C (de)
FI (1) FI60207C (de)
FR (1) FR2311778A1 (de)
GB (1) GB1546954A (de)
HU (1) HU172924B (de)
IE (1) IE42997B1 (de)
IL (1) IL49606A (de)
IN (1) IN142992B (de)
IT (1) IT1056271B (de)
NL (1) NL180478C (de)
NO (1) NO761705L (de)
PL (1) PL101470B1 (de)
PT (1) PT65113B (de)
SE (1) SE443142B (de)
SU (1) SU686620A3 (de)
YU (1) YU39965B (de)
ZA (1) ZA762989B (de)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK345977A (da) * 1976-09-30 1978-03-31 Archifar Ind Chim Trentino G rifamycinforbindelser og fremgangsmaade til deres fremstillin
GB1576886A (en) * 1977-04-20 1980-10-15 Lepetit Spa Rifamycin derivatives
CH633014A5 (en) * 1978-06-09 1982-11-15 Erba Farmitalia Rifamycin compounds
BE886395A (fr) * 1980-02-13 1981-03-16 Erba Farmitalia Derives de rifamycine
IT1201963B (it) * 1983-03-24 1989-02-02 Prodotti Antibiotici Spa Derivati delle rifamicine e procedimento per la loro preparazione
JPS61197941U (de) * 1985-05-30 1986-12-10
WO2003045319A2 (en) * 2001-11-21 2003-06-05 Activbiotics, Inc. Targeted therapeutics and uses thereof
US7820652B2 (en) * 2003-09-24 2010-10-26 Activbiotics Pharma, Llc Regimen for the administration of rifamycin-class antibiotics

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL130099C (de) * 1963-10-11
FR208F (de) * 1964-07-31
CA930734A (en) * 1969-08-11 1973-07-24 Bickel Hans Antibiotically active rifamycin compounds and processes for their manufacture

Also Published As

Publication number Publication date
DE2622638C2 (de) 1986-11-13
CH625804A5 (de) 1981-10-15
FI761392A (de) 1976-11-21
CA1053667A (en) 1979-05-01
FR2311778B1 (de) 1979-06-15
NO761705L (de) 1976-11-23
CS194763B2 (en) 1979-12-31
US4226765A (en) 1980-10-07
NL7605355A (nl) 1976-11-23
DK220276A (da) 1976-11-21
YU121176A (en) 1982-08-31
AU497327B2 (en) 1978-12-07
BE842036A (fr) 1976-09-16
DE2622638A1 (de) 1976-12-09
SU686620A3 (ru) 1979-09-15
NL180478C (nl) 1987-03-02
IE42997L (en) 1976-11-20
AR213175A1 (es) 1978-12-29
PT65113A (en) 1976-06-01
FR2311778A1 (fr) 1976-12-17
DK143852B (da) 1981-10-19
JPS554756B2 (de) 1980-01-31
SE443142B (sv) 1986-02-17
GB1546954A (en) 1979-05-31
IL49606A0 (en) 1976-07-30
IN142992B (de) 1977-09-17
AU1404776A (en) 1977-11-24
PT65113B (en) 1977-10-10
PL101470B1 (pl) 1978-12-30
YU39965B (en) 1985-06-30
IT1056271B (it) 1982-01-30
HU172924B (hu) 1979-01-28
IL49606A (en) 1979-11-30
FI60207B (fi) 1981-08-31
AT344897B (de) 1978-08-10
ATA343076A (de) 1977-12-15
IE42997B1 (en) 1980-12-03
NL180478B (nl) 1986-10-01
SE7605341L (sv) 1976-11-21
ZA762989B (en) 1977-04-27
DK143852C (da) 1982-03-15
JPS5248698A (en) 1977-04-18

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Date Code Title Description
MM Patent lapsed

Owner name: FARMITALIA CARLO ERBA S.P.A.