FI59253C - Foerfarande foer framstaellning av terapeutiskt anvaendbara 4-hydroxi-2h-tieno(2,3-e) och (3,4-e)-1,2-tiazin-3-karboxamid-1,1-dioxid-derivat - Google Patents
Foerfarande foer framstaellning av terapeutiskt anvaendbara 4-hydroxi-2h-tieno(2,3-e) och (3,4-e)-1,2-tiazin-3-karboxamid-1,1-dioxid-derivat Download PDFInfo
- Publication number
- FI59253C FI59253C FI752398A FI752398A FI59253C FI 59253 C FI59253 C FI 59253C FI 752398 A FI752398 A FI 752398A FI 752398 A FI752398 A FI 752398A FI 59253 C FI59253 C FI 59253C
- Authority
- FI
- Finland
- Prior art keywords
- methyl
- pyridyl
- formula
- hydroxy
- compound
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D333/30—Hetero atoms other than halogen
- C07D333/34—Sulfur atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D333/38—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pain & Pain Management (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Biomedical Technology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Rheumatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Manufacturing Of Printed Wiring (AREA)
- Electroplating Methods And Accessories (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CH1158274 | 1974-08-26 | ||
CH1158274A CH608500A5 (en) | 1974-08-26 | 1974-08-26 | Process for the preparation of thiazine derivatives |
CH1215774A CH608501A5 (en) | 1974-09-09 | 1974-09-09 | Process for the preparation of thiazine derivatives |
CH1215774 | 1974-09-09 |
Publications (3)
Publication Number | Publication Date |
---|---|
FI752398A FI752398A (zh) | 1976-02-27 |
FI59253B FI59253B (fi) | 1981-03-31 |
FI59253C true FI59253C (fi) | 1981-07-10 |
Family
ID=25708582
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FI752398A FI59253C (fi) | 1974-08-26 | 1975-08-26 | Foerfarande foer framstaellning av terapeutiskt anvaendbara 4-hydroxi-2h-tieno(2,3-e) och (3,4-e)-1,2-tiazin-3-karboxamid-1,1-dioxid-derivat |
Country Status (20)
Country | Link |
---|---|
JP (1) | JPS5826758B2 (zh) |
AR (1) | AR216288A1 (zh) |
AT (1) | AT350064B (zh) |
BR (1) | BR7505463A (zh) |
DD (1) | DD124119A5 (zh) |
DE (1) | DE2537070A1 (zh) |
DK (1) | DK137835B (zh) |
FI (1) | FI59253C (zh) |
FR (3) | FR2282893A1 (zh) |
GB (1) | GB1519811A (zh) |
HU (1) | HU173739B (zh) |
IE (1) | IE41457B1 (zh) |
IL (1) | IL47877A (zh) |
LU (2) | LU73257A1 (zh) |
NL (2) | NL183582C (zh) |
NO (1) | NO146096C (zh) |
PL (1) | PL106076B1 (zh) |
SE (1) | SE412066B (zh) |
SU (1) | SU603338A3 (zh) |
YU (1) | YU40266B (zh) |
Families Citing this family (17)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE2704485A1 (de) * | 1977-02-03 | 1978-08-10 | Thomae Gmbh Dr K | Neue 2,5-dihydro-1,2-thiazino eckige klammer auf 5,6-b eckige klammer zu indol-3-carboxamid-1,1-dioxide, verfahren zu ihrer herstellung und diese enthaltende arzneimittel |
LU78009A1 (de) | 1977-08-22 | 1979-05-23 | Hoffmann La Roche | Verfahren zur herstellung von thiazinderivaten |
ZA784958B (en) * | 1977-09-06 | 1979-08-29 | Hoffmann La Roche | Thiazine derivatives |
AU518216B2 (en) | 1977-09-06 | 1981-09-17 | Hafslund Nycomed Pharma Aktiengesellschaft | Thienothiazine derivatives |
DE2838377A1 (de) * | 1978-09-02 | 1980-03-20 | Thomae Gmbh Dr K | Neue 4-hydroxy-2h eckige klammer auf 1 eckige klammer zu benzothieno eckige klammer auf 2,3-e eckige klammer zu -1,2- thiazin-3-carboxamid-1,1-dioxide sowie deren salze, deren verwendung und verfahren zu ihrer herstellung |
AU5811280A (en) * | 1979-06-13 | 1980-12-18 | F. Hoffmann-La Roche Ag | Thiazine derivatives |
JPS58109492A (ja) * | 1981-12-22 | 1983-06-29 | Mitsui Toatsu Chem Inc | チエノチアジン誘導体およびそれを含有する医薬組成物 |
EP0103142B1 (de) * | 1982-09-09 | 1987-04-22 | F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft | Thieno(2,3-e)-1,2-thiazin-Derivate |
JPS60163533U (ja) * | 1984-04-02 | 1985-10-30 | ホシデン株式会社 | リ−ル台の制動装置 |
JPH0318748Y2 (zh) * | 1985-12-18 | 1991-04-19 | ||
ATA39088A (de) | 1988-02-18 | 1990-06-15 | Binder Dieter Dr | Basisch substituierte thienoisothiazol-3(2h)-on-1,1-dioxide und ihre pharmazeutisch vertraeglichen salze, verfahren zu ihrer herstellung und ihre verwendung |
AT400568B (de) * | 1994-05-18 | 1996-01-25 | Chem Pharm Forsch Gmbh | Neue n-heterocyclische thienothiazincarboxamide, verfahren zu ihrer herstellung und ihre verwendung |
AT400437B (de) * | 1993-12-14 | 1995-12-27 | Chem Pharm Forsch Gmbh | Neue n-heterocyclische thienothiazincarboxamide, verfahren zu ihrer herstellung und ihre verwendung |
EP0658559A1 (de) * | 1993-12-14 | 1995-06-21 | Chemisch Pharmazeutische Forschungsgesellschaft m.b.H. | Thienothiazinderivate, Verfahren zu ihrer Herstellung und ihre Verwendung als 5-dipoxygenase und Cyclooxygenaseinhibitoren |
US5538966A (en) * | 1994-01-21 | 1996-07-23 | Alcon Laboratories, Inc. | Carbonic anhydrase inhibitors |
IT1308633B1 (it) | 1999-03-02 | 2002-01-09 | Nicox Sa | Nitrossiderivati. |
CN1171892C (zh) * | 2001-06-25 | 2004-10-20 | 李晶 | 具有抗炎镇痛活性的噻吩并噻嗪化合物及其制备方法和用途 |
-
1975
- 1975-08-05 IL IL47877A patent/IL47877A/xx unknown
- 1975-08-20 DE DE19752537070 patent/DE2537070A1/de active Granted
- 1975-08-22 FR FR7525999A patent/FR2282893A1/fr active Granted
- 1975-08-22 GB GB34943/75A patent/GB1519811A/en not_active Expired
- 1975-08-22 AR AR260104A patent/AR216288A1/es active
- 1975-08-25 SU SU752167373A patent/SU603338A3/ru active
- 1975-08-25 IE IE1856/75A patent/IE41457B1/en not_active IP Right Cessation
- 1975-08-25 HU HU75HO1829A patent/HU173739B/hu unknown
- 1975-08-25 AT AT655975A patent/AT350064B/de active Protection Beyond IP Right Term
- 1975-08-25 SE SE7509446A patent/SE412066B/xx not_active IP Right Cessation
- 1975-08-25 DK DK381175AA patent/DK137835B/da not_active IP Right Cessation
- 1975-08-25 DD DD188010A patent/DD124119A5/xx unknown
- 1975-08-26 YU YU2166/75A patent/YU40266B/xx unknown
- 1975-08-26 PL PL1975182921A patent/PL106076B1/pl unknown
- 1975-08-26 NO NO752932A patent/NO146096C/no unknown
- 1975-08-26 JP JP50102635A patent/JPS5826758B2/ja not_active Expired
- 1975-08-26 FI FI752398A patent/FI59253C/fi not_active IP Right Cessation
- 1975-08-26 BR BR7505463*A patent/BR7505463A/pt unknown
- 1975-08-26 NL NLAANVRAGE7510057,A patent/NL183582C/xx active Protection Beyond IP Right Term
- 1975-08-26 LU LU73257A patent/LU73257A1/xx active Protection Beyond IP Right Term
-
1976
- 1976-05-21 FR FR7615425A patent/FR2309558A1/fr active Granted
- 1976-05-21 FR FR7615424A patent/FR2303803A1/fr active Granted
-
1993
- 1993-06-16 LU LU88312C patent/LU88312I2/de unknown
- 1993-06-17 NL NL930080C patent/NL930080I2/nl unknown
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
MA | Patent expired | ||
MA | Patent expired |
Owner name: F. HOFFMANN-LA ROCHE AG |