FR2309558A1 - Derives de thienothiazine et leurs procedes de preparation - Google Patents

Derives de thienothiazine et leurs procedes de preparation

Info

Publication number
FR2309558A1
FR2309558A1 FR7615425A FR7615425A FR2309558A1 FR 2309558 A1 FR2309558 A1 FR 2309558A1 FR 7615425 A FR7615425 A FR 7615425A FR 7615425 A FR7615425 A FR 7615425A FR 2309558 A1 FR2309558 A1 FR 2309558A1
Authority
FR
France
Prior art keywords
preparation methods
thienothiazine derivatives
thienothiazine
derivatives
preparation
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR7615425A
Other languages
English (en)
Other versions
FR2309558B1 (fr
Inventor
Otto Hromatka
Dieter Binder
Rudolf Pfister
Paul Zeller
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
F Hoffmann La Roche AG
Original Assignee
F Hoffmann La Roche AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from CH1158274A external-priority patent/CH608500A5/de
Priority claimed from CH1215774A external-priority patent/CH608501A5/de
Application filed by F Hoffmann La Roche AG filed Critical F Hoffmann La Roche AG
Publication of FR2309558A1 publication Critical patent/FR2309558A1/fr
Application granted granted Critical
Publication of FR2309558B1 publication Critical patent/FR2309558B1/fr
Granted legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D333/00Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/30Hetero atoms other than halogen
    • C07D333/34Sulfur atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D333/00Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/38Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pain & Pain Management (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biomedical Technology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Manufacturing Of Printed Wiring (AREA)
  • Electroplating Methods And Accessories (AREA)
FR7615425A 1974-08-26 1976-05-21 Derives de thienothiazine et leurs procedes de preparation Granted FR2309558A1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH1158274A CH608500A5 (en) 1974-08-26 1974-08-26 Process for the preparation of thiazine derivatives
CH1215774A CH608501A5 (en) 1974-09-09 1974-09-09 Process for the preparation of thiazine derivatives

Publications (2)

Publication Number Publication Date
FR2309558A1 true FR2309558A1 (fr) 1976-11-26
FR2309558B1 FR2309558B1 (fr) 1979-05-04

Family

ID=25708582

Family Applications (3)

Application Number Title Priority Date Filing Date
FR7525999A Granted FR2282893A1 (fr) 1974-08-26 1975-08-22 Derives de thienothiazine utiles en tant que medicaments et leur procede de preparation
FR7615425A Granted FR2309558A1 (fr) 1974-08-26 1976-05-21 Derives de thienothiazine et leurs procedes de preparation
FR7615424A Granted FR2303803A1 (fr) 1974-08-26 1976-05-21 Acides sulfothiophene-carboxyliques et leur procede de preparation

Family Applications Before (1)

Application Number Title Priority Date Filing Date
FR7525999A Granted FR2282893A1 (fr) 1974-08-26 1975-08-22 Derives de thienothiazine utiles en tant que medicaments et leur procede de preparation

Family Applications After (1)

Application Number Title Priority Date Filing Date
FR7615424A Granted FR2303803A1 (fr) 1974-08-26 1976-05-21 Acides sulfothiophene-carboxyliques et leur procede de preparation

Country Status (20)

Country Link
JP (1) JPS5826758B2 (fr)
AR (1) AR216288A1 (fr)
AT (1) AT350064B (fr)
BR (1) BR7505463A (fr)
DD (1) DD124119A5 (fr)
DE (1) DE2537070A1 (fr)
DK (1) DK137835B (fr)
FI (1) FI59253C (fr)
FR (3) FR2282893A1 (fr)
GB (1) GB1519811A (fr)
HU (1) HU173739B (fr)
IE (1) IE41457B1 (fr)
IL (1) IL47877A (fr)
LU (2) LU73257A1 (fr)
NL (2) NL183582C (fr)
NO (1) NO146096C (fr)
PL (1) PL106076B1 (fr)
SE (1) SE412066B (fr)
SU (1) SU603338A3 (fr)
YU (1) YU40266B (fr)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2704485A1 (de) * 1977-02-03 1978-08-10 Thomae Gmbh Dr K Neue 2,5-dihydro-1,2-thiazino eckige klammer auf 5,6-b eckige klammer zu indol-3-carboxamid-1,1-dioxide, verfahren zu ihrer herstellung und diese enthaltende arzneimittel
LU78009A1 (de) 1977-08-22 1979-05-23 Hoffmann La Roche Verfahren zur herstellung von thiazinderivaten
AU518216B2 (en) * 1977-09-06 1981-09-17 Hafslund Nycomed Pharma Aktiengesellschaft Thienothiazine derivatives
ZA784958B (en) * 1977-09-06 1979-08-29 Hoffmann La Roche Thiazine derivatives
DE2838377A1 (de) * 1978-09-02 1980-03-20 Thomae Gmbh Dr K Neue 4-hydroxy-2h eckige klammer auf 1 eckige klammer zu benzothieno eckige klammer auf 2,3-e eckige klammer zu -1,2- thiazin-3-carboxamid-1,1-dioxide sowie deren salze, deren verwendung und verfahren zu ihrer herstellung
AU5811280A (en) * 1979-06-13 1980-12-18 F. Hoffmann-La Roche Ag Thiazine derivatives
JPS58109492A (ja) * 1981-12-22 1983-06-29 Mitsui Toatsu Chem Inc チエノチアジン誘導体およびそれを含有する医薬組成物
DE3371082D1 (de) * 1982-09-09 1987-05-27 Hoffmann La Roche Thieno(2,3-e)-1,2-thiazine derivatives
JPS60163533U (ja) * 1984-04-02 1985-10-30 ホシデン株式会社 リ−ル台の制動装置
JPH0318748Y2 (fr) * 1985-12-18 1991-04-19
ATA39088A (de) 1988-02-18 1990-06-15 Binder Dieter Dr Basisch substituierte thienoisothiazol-3(2h)-on-1,1-dioxide und ihre pharmazeutisch vertraeglichen salze, verfahren zu ihrer herstellung und ihre verwendung
AT400568B (de) * 1994-05-18 1996-01-25 Chem Pharm Forsch Gmbh Neue n-heterocyclische thienothiazincarboxamide, verfahren zu ihrer herstellung und ihre verwendung
AT400437B (de) * 1993-12-14 1995-12-27 Chem Pharm Forsch Gmbh Neue n-heterocyclische thienothiazincarboxamide, verfahren zu ihrer herstellung und ihre verwendung
EP0658559A1 (fr) * 1993-12-14 1995-06-21 Chemisch Pharmazeutische Forschungsgesellschaft m.b.H. Dérivés thiénothianine, procédé pour leur préparation et leur application comme inhibiteurs de 5-dipoxygenase et cyclooxygenase
US5538966A (en) * 1994-01-21 1996-07-23 Alcon Laboratories, Inc. Carbonic anhydrase inhibitors
IT1308633B1 (it) 1999-03-02 2002-01-09 Nicox Sa Nitrossiderivati.
CN1171892C (zh) * 2001-06-25 2004-10-20 李晶 具有抗炎镇痛活性的噻吩并噻嗪化合物及其制备方法和用途

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
NEANT *

Also Published As

Publication number Publication date
FR2303803B1 (fr) 1979-07-13
JPS5826758B2 (ja) 1983-06-04
AR216288A1 (es) 1979-12-14
NL183582C (nl) 1988-12-01
AT350064B (de) 1979-05-10
NL930080I1 (nl) 1993-09-16
SU603338A3 (ru) 1978-04-15
FI59253C (fi) 1981-07-10
NL7510057A (nl) 1976-03-01
GB1519811A (en) 1978-08-02
AU8418675A (en) 1977-02-24
IL47877A0 (en) 1975-11-25
DK137835C (fr) 1978-10-16
FI59253B (fi) 1981-03-31
DD124119A5 (fr) 1977-02-02
DE2537070C2 (fr) 1987-06-25
DE2537070A1 (de) 1976-03-18
HU173739B (hu) 1979-08-28
NO146096C (no) 1982-07-28
NO752932L (fr) 1976-02-27
FR2282893A1 (fr) 1976-03-26
IE41457B1 (en) 1980-01-02
PL106076B1 (pl) 1979-11-30
JPS5148694A (fr) 1976-04-26
SE7509446L (sv) 1976-02-27
IE41457L (en) 1976-02-26
NL930080I2 (nl) 1994-01-03
LU88312I2 (de) 1994-09-09
FR2309558B1 (fr) 1979-05-04
FI752398A (fr) 1976-02-27
YU216675A (en) 1982-08-31
NL183582B (nl) 1988-07-01
LU73257A1 (fr) 1977-04-15
FR2303803A1 (fr) 1976-10-08
SE412066B (sv) 1980-02-18
FR2282893B1 (fr) 1980-05-16
NO146096B (no) 1982-04-19
YU40266B (en) 1985-12-31
DK381175A (fr) 1976-02-27
BR7505463A (pt) 1976-08-03
DK137835B (da) 1978-05-16
ATA655975A (de) 1978-10-15
IL47877A (en) 1978-10-31

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Legal Events

Date Code Title Description
TP Transmission of property
CC Supplementary protection certificate (spc) laid open to the public (law of 25 june 1990)

Free format text: 92C0155, 920504

CB Supplementary protection certificate (spc) granted (law of 25 june 1990)

Free format text: 92C0155, 760521

CL Concession to grant licences