BE838757A - Derives substitues de benzodiazepine et leurs procedes de preparation - Google Patents
Derives substitues de benzodiazepine et leurs procedes de preparationInfo
- Publication number
- BE838757A BE838757A BE164475A BE164475A BE838757A BE 838757 A BE838757 A BE 838757A BE 164475 A BE164475 A BE 164475A BE 164475 A BE164475 A BE 164475A BE 838757 A BE838757 A BE 838757A
- Authority
- BE
- Belgium
- Prior art keywords
- benzodiazepine
- preparation methods
- substitute derivatives
- substitute
- derivatives
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
- C07D495/14—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US05/552,023 US3953430A (en) | 1975-02-24 | 1975-02-24 | Substituted benzodiazepin-10-ones and method of use |
Publications (1)
Publication Number | Publication Date |
---|---|
BE838757A true BE838757A (fr) | 1976-08-20 |
Family
ID=24203630
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BE164475A BE838757A (fr) | 1975-02-24 | 1976-02-20 | Derives substitues de benzodiazepine et leurs procedes de preparation |
Country Status (2)
Country | Link |
---|---|
US (1) | US3953430A (fr) |
BE (1) | BE838757A (fr) |
Families Citing this family (15)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4172831A (en) * | 1974-11-26 | 1979-10-30 | Lilly Industries Limited | Thieno-benzodiazepines |
US4066647A (en) * | 1976-11-12 | 1978-01-03 | American Cyanamid Company | Substituted 6-(piperazinyl)-10H-pyrido[3,2-b]thieno[3,4-e][1,4]-diazepines |
US4168269A (en) * | 1978-04-12 | 1979-09-18 | American Cyanamid Company | Substituted thieno-benzodiazepines |
US4404137A (en) * | 1979-10-16 | 1983-09-13 | Lilly Industries Limited | Pyrazolo [3,4-b][1,5]benzodiazepine compounds |
IL62792A (en) * | 1980-05-07 | 1985-02-28 | Byk Gulden Lomberg Chem Fab | Acylated dihydrothienodiazepinone compounds,process for their preparation,and medicaments containing them |
US4381301A (en) * | 1980-05-07 | 1983-04-26 | Byk Gulden Lomberg Chemische Fabrik Gmbh | Substituted tricyclic thieno compounds, their synthesis, their use, their compositions and their medicaments |
US4431589A (en) * | 1980-12-11 | 1984-02-14 | Lilly House | Benzodiazepine compounds and their use as pharmaceuticals |
DE3204169A1 (de) * | 1982-02-06 | 1983-08-11 | Dr. Karl Thomae Gmbh, 7950 Biberach | Substituierte thienobenzodiazepinone, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel |
DE3529372A1 (de) * | 1985-08-16 | 1987-02-19 | Dompe Farmaceutici Spa | Aminoacyl-derivat von 4,9-dihydro-10h-pyrido(3,2-b)-thieno(3,2-e) (1,4)-diazepinon und von 4,9-dihydro-10h-pyrido(3,2-b)thieno(3,4-e) (1,4)diazepinon, verfahren zu deren herstellung und diese verbindungen enthaltende pharmazeutische zusammensetzungen |
GB9009229D0 (en) * | 1990-04-25 | 1990-06-20 | Lilly Industries Ltd | Pharmaceutical compounds |
US7893053B2 (en) * | 2006-06-16 | 2011-02-22 | Theracos, Inc. | Treating psychological conditions using muscarinic receptor M1 antagonists |
RU2477634C2 (ru) * | 2006-06-16 | 2013-03-20 | Теракос, Инк. | Лечение психологических состояний с применением антагонистов m1-мускариновых рецепторов |
CN101472476B (zh) * | 2006-06-16 | 2013-10-30 | 泰拉科斯有限公司 | 毒蕈碱型受体m1拮抗剂在制备治疗肥胖症的药物中的应用 |
US8748419B2 (en) | 2006-06-16 | 2014-06-10 | Theracos, Inc. | Treating obesity with muscarinic receptor M1 antagonists |
US8440655B2 (en) | 2010-06-21 | 2013-05-14 | Theracos, Inc. | Combination therapy for the treatment of diabetes |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE1470367A1 (de) * | 1964-04-21 | 1969-11-13 | Thomae Gmbh Dr K | Verfahren zur Herstellung von in 5-Stellung substituierten 5,6-Dihydro-6-oxopyrido[2,3-b][1,4]benzoxazepinen |
NL6600292A (fr) * | 1965-01-11 | 1966-07-12 | ||
GB1156781A (en) * | 1965-04-07 | 1969-07-02 | Lab U P S A | New Heterocyclic Compounds |
CH468400A (de) * | 1965-12-23 | 1969-02-15 | Sandoz Ag | Verfahren zur Herstellung neuer Thieno(2,3-b)(1,5)benzothiazepin-4-on-Verbindungen |
-
1975
- 1975-02-24 US US05/552,023 patent/US3953430A/en not_active Expired - Lifetime
-
1976
- 1976-02-20 BE BE164475A patent/BE838757A/fr unknown
Also Published As
Publication number | Publication date |
---|---|
US3953430A (en) | 1976-04-27 |
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