FI57414C - Foerfarande foer framstaellning av i 6-,7-,8- och/eller 9-staellning substituerade 4-(substituerad amino)-1,3-dimetyl-1h-pyrazolo(3,4b)kinoliner med antiviral verkan - Google Patents

Foerfarande foer framstaellning av i 6-,7-,8- och/eller 9-staellning substituerade 4-(substituerad amino)-1,3-dimetyl-1h-pyrazolo(3,4b)kinoliner med antiviral verkan Download PDF

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Publication number
FI57414C
FI57414C FI2815/74A FI281574A FI57414C FI 57414 C FI57414 C FI 57414C FI 2815/74 A FI2815/74 A FI 2815/74A FI 281574 A FI281574 A FI 281574A FI 57414 C FI57414 C FI 57414C
Authority
FI
Finland
Prior art keywords
dimethyl
pyrazolo
substitutes
antiviral
formula
Prior art date
Application number
FI2815/74A
Other languages
English (en)
Finnish (fi)
Other versions
FI57414B (fi
FI281574A (no
Inventor
Ronnie Ray Crenshaw
George Michael Luke
Paul Siminoff
Original Assignee
Bristol Myers Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Co filed Critical Bristol Myers Co
Publication of FI281574A publication Critical patent/FI281574A/fi
Application granted granted Critical
Publication of FI57414B publication Critical patent/FI57414B/fi
Publication of FI57414C publication Critical patent/FI57414C/fi

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/38Nitrogen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D265/00Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D265/041,3-Oxazines; Hydrogenated 1,3-oxazines
    • C07D265/121,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems
    • C07D265/141,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • C07D265/201,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring with hetero atoms directly attached in position 4
    • C07D265/22Oxygen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Communicable Diseases (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Virology (AREA)
  • Oncology (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Fodder In General (AREA)
FI2815/74A 1973-10-01 1974-09-26 Foerfarande foer framstaellning av i 6-,7-,8- och/eller 9-staellning substituerade 4-(substituerad amino)-1,3-dimetyl-1h-pyrazolo(3,4b)kinoliner med antiviral verkan FI57414C (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US05/402,657 US4013665A (en) 1973-10-01 1973-10-01 Antiviral, substituted 1,3-dimethyl-1h-pyrazolo(3,4b)quinolines
US40265773 1973-10-01

Publications (3)

Publication Number Publication Date
FI281574A FI281574A (no) 1975-04-02
FI57414B FI57414B (fi) 1980-04-30
FI57414C true FI57414C (fi) 1980-08-11

Family

ID=23592812

Family Applications (1)

Application Number Title Priority Date Filing Date
FI2815/74A FI57414C (fi) 1973-10-01 1974-09-26 Foerfarande foer framstaellning av i 6-,7-,8- och/eller 9-staellning substituerade 4-(substituerad amino)-1,3-dimetyl-1h-pyrazolo(3,4b)kinoliner med antiviral verkan

Country Status (19)

Country Link
US (1) US4013665A (no)
JP (1) JPS582948B2 (no)
BE (1) BE820400A (no)
CA (1) CA1032538A (no)
CH (3) CH621552A5 (no)
CY (1) CY1087A (no)
DE (1) DE2446821A1 (no)
DK (1) DK516274A (no)
ES (1) ES430554A1 (no)
FI (1) FI57414C (no)
FR (1) FR2245369B1 (no)
GB (1) GB1488692A (no)
HK (1) HK59380A (no)
KE (1) KE3086A (no)
MY (1) MY8100219A (no)
NL (1) NL7412959A (no)
NO (1) NO143223C (no)
SE (1) SE419760B (no)
ZA (1) ZA746138B (no)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA848968B (en) * 1983-11-18 1986-06-25 Riker Laboratories Inc 1h-imidazo(4,5-c)quinolines and 1h-imidazo(4,5-c)quinolin-4-amines
IL73534A (en) * 1983-11-18 1990-12-23 Riker Laboratories Inc 1h-imidazo(4,5-c)quinoline-4-amines,their preparation and pharmaceutical compositions containing certain such compounds
US5332734A (en) * 1991-04-10 1994-07-26 Japan Tobacco, Incorporated Oxazinone derivative
US5608067A (en) * 1993-12-09 1997-03-04 Afonso; Adriano 4-substituted pyrazoloquinoline derivatives
US5506236A (en) * 1994-04-28 1996-04-09 Schering Corporation 4-substituted pyrazoloquinoline derivatives
US5786480A (en) * 1994-04-28 1998-07-28 Schering Corporation 4-substituted pyrazoloquinoline derivatives
US5614530A (en) * 1995-03-10 1997-03-25 Sterling Winthrop Inc. Substituted N-arylmethyl and heterocyclmethyl-1H-pyrazolo[3,4-b]quinolin-4-amines and compositions and methods of use thereof
US6008226A (en) * 1995-03-10 1999-12-28 Sanofi-Synthelabo Substituted N-arylmethyl and heterocylylmethyl-1H-pyrazolo[3,4-b]quinolin-4-amines and compositions and methods of use thereof
US5488055A (en) * 1995-03-10 1996-01-30 Sanofi Winthrop Inc. Substituted N-cycloalkylmethyl-1H-pyrazolo(3,4-b)quinolin-4 amines and compositions and methods of use thereof
US7084156B2 (en) * 2001-11-27 2006-08-01 Merck & Co., Inc. 2-Aminoquinoline compounds
WO2003045920A1 (en) * 2001-11-27 2003-06-05 Merck & Co., Inc. 4-aminoquinoline compounds
US8080560B2 (en) * 2004-12-17 2011-12-20 3M Innovative Properties Company Immune response modifier formulations containing oleic acid and methods
US8889154B2 (en) 2005-09-15 2014-11-18 Medicis Pharmaceutical Corporation Packaging for 1-(2-methylpropyl)-1H-imidazo[4,5-c] quinolin-4-amine-containing formulation
WO2008010963A2 (en) * 2006-07-18 2008-01-24 3M Innovative Properties Company Immune response modifier formulations
WO2008016475A2 (en) * 2006-07-31 2008-02-07 3M Innovative Properties Company Immune response modifier compositions and methods
WO2010062559A1 (en) * 2008-10-28 2010-06-03 Schering Corporation Substituted pyrazoloquinolines and derivatives thereof

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1152421B (de) * 1961-03-21 1963-08-08 Bayer Ag Verfahren zur Herstellung von 4-Hydroxy-pyrazolo[3, 4-b]chinolinen
DE1445719A1 (de) * 1961-03-21 1969-01-09 Bayer Ag Verfahren zur Herstellung von 4-Chlor- oder 4-Brom-pyrazolo[3,4-]chinolinen
DE1186867B (de) * 1961-05-03 1965-02-11 Bayer Ag Verfahren zur Herstellung von heterocyclischen Verbindungen
DE1222885B (de) * 1962-05-25 1966-08-18 Bayer Ag Optische Aufhellungsmittel
US3600393A (en) * 1969-03-03 1971-08-17 Aldrich Chem Co Inc Dialkylamino alkylamino pyrazolo (3,4b) quinolines
JPS4826797A (no) * 1971-08-07 1973-04-09
US3790576A (en) * 1972-03-20 1974-02-05 Parke Davis & Co 9 substituted 4,9-dihydro-1,3,4,4-tetraalkyl-1h-pyrazolo(3,4-b)quinolines

Also Published As

Publication number Publication date
FR2245369A1 (no) 1975-04-25
NL7412959A (nl) 1975-04-03
FR2245369B1 (no) 1978-07-28
CY1087A (en) 1980-12-27
CH621552A5 (no) 1981-02-13
GB1488692A (en) 1977-10-12
JPS5059396A (no) 1975-05-22
NO143223B (no) 1980-09-22
US4013665A (en) 1977-03-22
KE3086A (en) 1980-11-07
NO143223C (no) 1981-01-02
ES430554A1 (es) 1977-07-01
ZA746138B (en) 1975-10-29
NO743528L (no) 1975-04-28
CH622793A5 (no) 1981-04-30
DE2446821A1 (de) 1975-04-10
BE820400A (fr) 1975-03-26
AU7379874A (en) 1976-04-01
JPS582948B2 (ja) 1983-01-19
SE419760B (sv) 1981-08-24
CA1032538A (en) 1978-06-06
CH619712A5 (no) 1980-10-15
HK59380A (en) 1980-10-31
SE7412275L (no) 1975-04-02
MY8100219A (en) 1981-12-31
FI57414B (fi) 1980-04-30
DK516274A (no) 1975-06-30
USB402657I5 (no) 1976-04-06
FI281574A (no) 1975-04-02

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