FI106458B - Terapeuttisesti käyttökelpoisten tienosyklopentanonioksiimien eetterien valmistusmenetelmä - Google Patents

Terapeuttisesti käyttökelpoisten tienosyklopentanonioksiimien eetterien valmistusmenetelmä Download PDF

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Publication number
FI106458B
FI106458B FI924281A FI924281A FI106458B FI 106458 B FI106458 B FI 106458B FI 924281 A FI924281 A FI 924281A FI 924281 A FI924281 A FI 924281A FI 106458 B FI106458 B FI 106458B
Authority
FI
Finland
Prior art keywords
formula
alkyl
acid
oxime
give
Prior art date
Application number
FI924281A
Other languages
English (en)
Finnish (fi)
Swedish (sv)
Other versions
FI924281A (fi
FI924281A0 (fi
Inventor
Daniel Frehel
Claudine Serradeil-Legal
Alain Badorc
Jean Courregelongue
Daniel Ducros
Antonina Giudice
Original Assignee
Sanofi Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Synthelabo filed Critical Sanofi Synthelabo
Publication of FI924281A0 publication Critical patent/FI924281A0/fi
Publication of FI924281A publication Critical patent/FI924281A/fi
Application granted granted Critical
Publication of FI106458B publication Critical patent/FI106458B/fi

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
    • C07D333/08—Hydrogen atoms or radicals containing only hydrogen and carbon atoms
    • C07D333/10—Thiophene
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D333/78—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems condensed with rings other than six-membered or with ring systems containing such rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Psychiatry (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pain & Pain Management (AREA)
  • Cardiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
FI924281A 1991-09-25 1992-09-24 Terapeuttisesti käyttökelpoisten tienosyklopentanonioksiimien eetterien valmistusmenetelmä FI106458B (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9111822 1991-09-25
FR9111822 1991-09-25

Publications (3)

Publication Number Publication Date
FI924281A0 FI924281A0 (fi) 1992-09-24
FI924281A FI924281A (fi) 1993-03-26
FI106458B true FI106458B (fi) 2001-02-15

Family

ID=9417295

Family Applications (1)

Application Number Title Priority Date Filing Date
FI924281A FI106458B (fi) 1991-09-25 1992-09-24 Terapeuttisesti käyttökelpoisten tienosyklopentanonioksiimien eetterien valmistusmenetelmä

Country Status (23)

Country Link
US (1) US5252749A (de)
EP (1) EP0534856B1 (de)
JP (1) JP3162822B2 (de)
KR (1) KR100199848B1 (de)
AR (1) AR248275A1 (de)
AT (1) ATE157360T1 (de)
AU (1) AU652072B2 (de)
BR (1) BR9203744A (de)
CA (1) CA2079016A1 (de)
CZ (1) CZ281936B6 (de)
DE (1) DE69221802T2 (de)
DK (1) DK0534856T3 (de)
ES (1) ES2108098T3 (de)
FI (1) FI106458B (de)
GR (1) GR3025335T3 (de)
HU (1) HU218204B (de)
IL (1) IL103106A (de)
MX (1) MX9205390A (de)
NO (1) NO301327B1 (de)
NZ (1) NZ244452A (de)
PH (1) PH30225A (de)
RU (1) RU2060253C1 (de)
ZA (1) ZA927318B (de)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1997044062A1 (en) * 1996-05-23 1997-11-27 Alcon Laboratories, Inc. The use of 5-ht1b/1d agonists to treat ocular pain
WO2003014107A1 (en) * 2001-08-01 2003-02-20 Basell Polyolefine Gmbh Process for the preparation of heterocyclic pentalene derivatives
US7432328B2 (en) * 2005-06-14 2008-10-07 Univation Technologies, Llc Enhanced ESCR bimodal HDPE for blow molding applications

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE371190B (de) * 1972-03-24 1974-11-11 Kabi Ab
US3301874A (en) * 1963-12-26 1967-01-31 Sam Joseph Thienocyclopentanone antibacterial agents
SE371193B (de) * 1972-03-24 1974-11-11 Kabi Ab
US4154740A (en) * 1976-03-23 1979-05-15 American Cyanamid Company Substituted tetrahydrobenzothiophenes and method of preparation thereof
FR2471980A1 (fr) * 1979-12-21 1981-06-26 Sanofi Sa Nouveaux derives de l'amino-1 propanol-2, leur procede de preparation et leur application therapeutique
FR2567125B1 (fr) * 1984-07-09 1986-12-05 Lipha Acides dihydro-5,6-4h-cyclopenta (b) thiophenecarboxylique-6, procedes de preparation et medicaments les contenant
FR2639942B1 (fr) * 1988-12-02 1991-03-29 Sanofi Sa Ethers oximes de propenone, procede pour leur preparation et compositions pharmaceutiques les contenant

Also Published As

Publication number Publication date
CZ291892A3 (en) 1993-04-14
JP3162822B2 (ja) 2001-05-08
MX9205390A (es) 1993-05-01
RU2060253C1 (ru) 1996-05-20
BR9203744A (pt) 1994-03-29
PH30225A (en) 1997-02-05
ZA927318B (en) 1994-03-24
FI924281A (fi) 1993-03-26
CZ281936B6 (cs) 1997-04-16
EP0534856B1 (de) 1997-08-27
JPH05213932A (ja) 1993-08-24
GR3025335T3 (en) 1998-02-27
HU9203050D0 (en) 1992-12-28
EP0534856A1 (de) 1993-03-31
US5252749A (en) 1993-10-12
NO923720L (no) 1993-03-26
IL103106A0 (en) 1993-02-21
IL103106A (en) 1998-06-15
NO923720D0 (no) 1992-09-24
DE69221802T2 (de) 1998-04-02
KR100199848B1 (ko) 1999-06-15
DE69221802D1 (de) 1997-10-02
DK0534856T3 (da) 1998-04-20
AU2454892A (en) 1993-04-01
ES2108098T3 (es) 1997-12-16
NO301327B1 (no) 1997-10-13
HUT62876A (en) 1993-06-28
KR930006001A (ko) 1993-04-20
HU218204B (hu) 2000-06-28
AU652072B2 (en) 1994-08-11
FI924281A0 (fi) 1992-09-24
NZ244452A (en) 1994-08-26
ATE157360T1 (de) 1997-09-15
CA2079016A1 (en) 1993-03-26
AR248275A1 (es) 1995-07-12

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Owner name: SANOFI