FI101538B1 - Menetelmä uusien, terapeuttisesti käyttökelpoisten 2-metyyli-4-(4-metyyli-1-piperatsinyyli)-10H-tieno[2,3-b][1,5]bentsodiatsepiinijohdannaisten valmistamiseksi - Google Patents
Menetelmä uusien, terapeuttisesti käyttökelpoisten 2-metyyli-4-(4-metyyli-1-piperatsinyyli)-10H-tieno[2,3-b][1,5]bentsodiatsepiinijohdannaisten valmistamiseksiInfo
- Publication number
- FI101538B1 FI101538B1 FI932445A FI932445A FI101538B1 FI 101538 B1 FI101538 B1 FI 101538B1 FI 932445 A FI932445 A FI 932445A FI 932445 A FI932445 A FI 932445A FI 101538 B1 FI101538 B1 FI 101538B1
- Authority
- FI
- Finland
- Prior art keywords
- methyl
- thieno
- piperazinyl
- preparation
- therapeutically useful
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Hospice & Palliative Care (AREA)
- Anesthesiology (AREA)
- Addiction (AREA)
- Otolaryngology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB929211379A GB9211379D0 (en) | 1992-05-29 | 1992-05-29 | Pharmaceutical compounds |
GB939309025A GB9309025D0 (en) | 1993-04-30 | 1993-04-30 | Pharmaceutical compounds |
Publications (4)
Publication Number | Publication Date |
---|---|
FI932445A0 FI932445A0 (fi) | 1993-05-28 |
FI932445A FI932445A (fi) | 1993-11-30 |
FI101538B1 true FI101538B1 (fi) | 1998-07-15 |
FI101538B FI101538B (fi) | 1998-07-15 |
Family
ID=26300951
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FI932445A FI101538B (fi) | 1992-05-29 | 1993-05-28 | Menetelmä uusien, terapeuttisesti käyttökelpoisten 2-metyyli-4-(4-mety yli-1-piperatsinyyli)-10H-tieno£2,3-b|£1,5|bentsodiatsepiinijohdannais ten valmistamiseksi |
Country Status (21)
Country | Link |
---|---|
EP (1) | EP0582368B1 (hr) |
JP (1) | JP3219541B2 (hr) |
CN (1) | CN1043994C (hr) |
AT (1) | ATE198891T1 (hr) |
AU (1) | AU668159B2 (hr) |
CA (1) | CA2097016A1 (hr) |
CZ (1) | CZ282783B6 (hr) |
DE (1) | DE69329887T2 (hr) |
DK (1) | DK0582368T3 (hr) |
ES (1) | ES2153373T3 (hr) |
FI (1) | FI101538B (hr) |
GR (1) | GR3035587T3 (hr) |
HU (1) | HU218278B (hr) |
IL (1) | IL105827A (hr) |
MX (1) | MX9303124A (hr) |
MY (1) | MY109943A (hr) |
NO (1) | NO305125B1 (hr) |
NZ (1) | NZ247703A (hr) |
PT (1) | PT582368E (hr) |
RU (1) | RU2125574C1 (hr) |
TW (1) | TW268005B (hr) |
Families Citing this family (29)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5457101A (en) * | 1994-06-03 | 1995-10-10 | Eli Lilly And Company | Thieno[1,5]benzoidiazepine use |
US5574028A (en) * | 1994-10-31 | 1996-11-12 | Eli Lilly And Company | Method for treating anxiety |
EG24221A (en) * | 1995-03-24 | 2008-11-10 | Lilly Co Eli | Process for preparing olanzapine |
CR5278A (es) | 1995-03-24 | 1996-07-04 | Lilly Co Eli | Formulacion oral de 2-metil-tieno-benzodiacepina |
EG23659A (en) * | 1995-03-24 | 2007-03-26 | Lilly Co Eli | Process and crystal forms of methyl-thieno-benzodiazepine |
US5891461A (en) * | 1995-09-14 | 1999-04-06 | Cygnus, Inc. | Transdermal administration of olanzapine |
CN1146421C (zh) * | 1996-03-25 | 2004-04-21 | 伊莱利利公司 | 治疗疼痛的组合物以及药物在制备所述组合物中的应用 |
IL126063A (en) * | 1996-03-25 | 2002-04-21 | Lilly Co Eli | Medicinal products containing ulanzapine for the treatment of migraine pain |
CA2248873A1 (en) * | 1996-03-25 | 1997-10-02 | Daniel Edward Womer | Method for treating pain |
UA56184C2 (uk) | 1996-09-23 | 2003-05-15 | Елі Ліллі Енд Компані | Поліморфна модифікація оланзапіну дигідрату d, фармацевтична композиція та спосіб лікування психотичного стану |
ZA978515B (en) * | 1996-09-23 | 1999-03-23 | Lilly Co Eli | Intermediates and process for preparing olanzapine |
CZ98899A3 (cs) * | 1996-09-24 | 1999-12-15 | Eli Lilly And Company | Složení potahovaných částic |
WO2014031662A2 (en) | 2012-08-21 | 2014-02-27 | Ortho-Clinical Diagnostics, Inc | Antibodies to olanzapine and use thereof |
WO2014031645A1 (en) | 2012-08-21 | 2014-02-27 | Ortho-Clinical Diagnostics, Inc | Antibodies to risperidone haptens and use thereof |
PT3462173T (pt) | 2012-08-21 | 2021-04-28 | Janssen Pharmaceutica Nv | Anticorpos contra risperidona e utilização dos mesmos |
WO2014031630A2 (en) | 2012-08-21 | 2014-02-27 | Ortho-Clinical Diagnostics, Inc | Antibodies to paliperidone and use thereof |
PL3663317T3 (pl) | 2012-08-21 | 2023-06-05 | Janssen Pharmaceutica Nv | Przeciwciała skierowane przeciwko haptenom kwetiapinowym i ich zastosowanie |
PL3305784T3 (pl) | 2012-08-21 | 2021-03-08 | Janssen Pharmaceutica Nv | Hapteny kwetiapiny do zastosowania w testach immunologicznych |
EP2888287A4 (en) | 2012-08-21 | 2016-04-20 | Ortho Clinical Diagnostics Inc | ANTIBODIES AGAINST PALIPERIDONE HAPTENES AND THEIR USE |
WO2014031635A1 (en) | 2012-08-21 | 2014-02-27 | Ortho-Clinical Diagnostics, Inc | Antibodies to aripiprazole haptens and use thereof |
CA2882449C (en) | 2012-08-21 | 2018-09-04 | Ronghui Lin | Haptens of aripiprazole and their use in immunoassays |
CN109400708A (zh) | 2012-08-21 | 2019-03-01 | 詹森药业有限公司 | 奥氮平半抗原的抗体及其用途 |
PT3333195T (pt) | 2012-08-21 | 2020-10-12 | Janssen Pharmaceutica Nv | Anticorpos contra a quetiapina e sua utilização |
CN110003201A (zh) | 2012-08-21 | 2019-07-12 | 詹森药业有限公司 | 帕潘立酮半抗原 |
TR201816378T4 (tr) * | 2012-08-21 | 2018-11-21 | Janssen Pharmaceutica Nv | Olanzapin haptenleri. |
CA2882562C (en) | 2012-08-21 | 2019-08-27 | Eric Hryhorenko | Antibodies to aripiprazole and use thereof |
TR201809424T4 (tr) | 2012-08-21 | 2018-07-23 | Janssen Pharmaceutica Nv | Risperidon ve paliperidon haptenleri. |
AU2016370853A1 (en) | 2015-12-17 | 2018-06-07 | Saladax Biomedical Inc. | Antibodies to quetiapine and use thereof |
MA44056A (fr) | 2015-12-17 | 2018-10-24 | Janssen Pharmaceutica Nv | Anticorps anti-rispéridone et leur utilisation |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
SU629879A3 (ru) * | 1974-11-26 | 1978-10-25 | Лилли Индастриз Лимитед, (Фирма) | Способ получени тиено(1,5) бензодиазепинов или их солей |
DE2641378A1 (de) * | 1975-09-24 | 1977-04-07 | Sandoz Ag | Neue organische verbindungen, ihre verwendung und herstellung |
GB9009229D0 (en) * | 1990-04-25 | 1990-06-20 | Lilly Industries Ltd | Pharmaceutical compounds |
-
1993
- 1993-05-26 DE DE69329887T patent/DE69329887T2/de not_active Expired - Fee Related
- 1993-05-26 NZ NZ247703A patent/NZ247703A/en unknown
- 1993-05-26 TW TW082104161A patent/TW268005B/zh active
- 1993-05-26 ES ES93304102T patent/ES2153373T3/es not_active Expired - Lifetime
- 1993-05-26 NO NO931917A patent/NO305125B1/no not_active IP Right Cessation
- 1993-05-26 CA CA002097016A patent/CA2097016A1/en not_active Abandoned
- 1993-05-26 DK DK93304102T patent/DK0582368T3/da active
- 1993-05-26 PT PT93304102T patent/PT582368E/pt unknown
- 1993-05-26 AT AT93304102T patent/ATE198891T1/de not_active IP Right Cessation
- 1993-05-26 AU AU39807/93A patent/AU668159B2/en not_active Ceased
- 1993-05-26 EP EP93304102A patent/EP0582368B1/en not_active Expired - Lifetime
- 1993-05-27 MX MX9303124A patent/MX9303124A/es not_active IP Right Cessation
- 1993-05-28 MY MYPI93001036A patent/MY109943A/en unknown
- 1993-05-28 JP JP12642993A patent/JP3219541B2/ja not_active Expired - Fee Related
- 1993-05-28 CZ CZ931024A patent/CZ282783B6/cs not_active IP Right Cessation
- 1993-05-28 CN CN93108212A patent/CN1043994C/zh not_active Expired - Fee Related
- 1993-05-28 RU RU93005057A patent/RU2125574C1/ru active
- 1993-05-28 IL IL10582793A patent/IL105827A/xx not_active IP Right Cessation
- 1993-05-28 FI FI932445A patent/FI101538B/fi active
- 1993-05-28 HU HU9301579A patent/HU218278B/hu not_active IP Right Cessation
-
2001
- 2001-03-15 GR GR20010400431T patent/GR3035587T3/el not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
CA2097016A1 (en) | 1993-11-30 |
RU2125574C1 (ru) | 1999-01-27 |
GR3035587T3 (en) | 2001-06-29 |
TW268005B (hr) | 1996-01-11 |
DE69329887D1 (de) | 2001-03-01 |
IL105827A0 (en) | 1993-09-22 |
JP3219541B2 (ja) | 2001-10-15 |
DE69329887T2 (de) | 2001-05-23 |
HU218278B (en) | 2000-07-28 |
NO931917L (no) | 1993-11-30 |
FI932445A (fi) | 1993-11-30 |
EP0582368A1 (en) | 1994-02-09 |
IL105827A (en) | 1997-02-18 |
AU668159B2 (en) | 1996-04-26 |
PT582368E (pt) | 2001-05-31 |
EP0582368B1 (en) | 2001-01-24 |
CZ102493A3 (en) | 1993-12-15 |
ATE198891T1 (de) | 2001-02-15 |
FI932445A0 (fi) | 1993-05-28 |
AU3980793A (en) | 1993-12-02 |
NO305125B1 (no) | 1999-04-06 |
CZ282783B6 (cs) | 1997-10-15 |
NO931917D0 (no) | 1993-05-26 |
HU9301579D0 (en) | 1993-09-28 |
CN1043994C (zh) | 1999-07-07 |
JPH0687862A (ja) | 1994-03-29 |
ES2153373T3 (es) | 2001-03-01 |
CN1085903A (zh) | 1994-04-27 |
HUT66180A (en) | 1994-09-28 |
MY109943A (en) | 1997-10-31 |
MX9303124A (es) | 1993-11-01 |
FI101538B (fi) | 1998-07-15 |
NZ247703A (en) | 1995-07-26 |
DK0582368T3 (da) | 2001-02-05 |
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