FI101344B1 - Menetelmä valmistaa valmiste, josta kontrolloidusti vapautuu farmaseuttisesti aktiivista ainetta - Google Patents

Menetelmä valmistaa valmiste, josta kontrolloidusti vapautuu farmaseuttisesti aktiivista ainetta

Info

Publication number
FI101344B1
FI101344B1 FI891163A FI891163A FI101344B1 FI 101344 B1 FI101344 B1 FI 101344B1 FI 891163 A FI891163 A FI 891163A FI 891163 A FI891163 A FI 891163A FI 101344 B1 FI101344 B1 FI 101344B1
Authority
FI
Finland
Prior art keywords
controlled release
pharmaceutically active
preparation
composition
active substance
Prior art date
Application number
FI891163A
Other languages
English (en)
Finnish (fi)
Swedish (sv)
Other versions
FI891163A0 (fi
FI891163A (fi
FI101344B (fi
Inventor
Masayoshi Samejima
Kazuo Noda
Yoshiyuki Hirakawa
Hiroyuki Yoshino
Original Assignee
Tanabe Seiyaku Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=13722933&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=FI101344(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Tanabe Seiyaku Co filed Critical Tanabe Seiyaku Co
Publication of FI891163A0 publication Critical patent/FI891163A0/fi
Publication of FI891163A publication Critical patent/FI891163A/fi
Application granted granted Critical
Publication of FI101344B1 publication Critical patent/FI101344B1/fi
Publication of FI101344B publication Critical patent/FI101344B/fi

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5073Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
    • A61K9/5078Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2833Organic macromolecular compounds
    • A61K9/286Polysaccharides, e.g. gums; Cyclodextrin
    • A61K9/2866Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose

Landscapes

  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
FI891163A 1988-03-31 1989-03-10 Menetelmä valmistaa valmiste, josta kontrolloidusti vapautuu farmaseut tisesti aktiivista ainetta FI101344B (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP8060488 1988-03-31
JP8060488 1988-03-31

Publications (4)

Publication Number Publication Date
FI891163A0 FI891163A0 (fi) 1989-03-10
FI891163A FI891163A (fi) 1989-10-01
FI101344B1 true FI101344B1 (fi) 1998-06-15
FI101344B FI101344B (fi) 1998-06-15

Family

ID=13722933

Family Applications (1)

Application Number Title Priority Date Filing Date
FI891163A FI101344B (fi) 1988-03-31 1989-03-10 Menetelmä valmistaa valmiste, josta kontrolloidusti vapautuu farmaseut tisesti aktiivista ainetta

Country Status (21)

Country Link
US (1) US5068112A (fr)
EP (1) EP0335560B2 (fr)
KR (1) KR950007202B1 (fr)
AT (1) ATE91888T1 (fr)
AU (1) AU610711B2 (fr)
BG (1) BG50712A3 (fr)
CA (1) CA1339078C (fr)
DE (1) DE68907762T3 (fr)
DK (1) DK156289A (fr)
ES (1) ES2059729T5 (fr)
FI (1) FI101344B (fr)
FR (1) FR2629344B1 (fr)
HK (1) HK76195A (fr)
HU (1) HU201882B (fr)
IE (1) IE64348B1 (fr)
IL (1) IL89695A0 (fr)
NO (1) NO178136C (fr)
PH (1) PH25791A (fr)
PT (1) PT90153B (fr)
RU (1) RU1836083C (fr)
ZA (1) ZA892131B (fr)

Families Citing this family (58)

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FI101344B (fi) 1988-03-31 1998-06-15 Tanabe Seiyaku Co Menetelmä valmistaa valmiste, josta kontrolloidusti vapautuu farmaseut tisesti aktiivista ainetta
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US6913767B1 (en) 1993-10-25 2005-07-05 Genentech, Inc. Compositions for microencapsulation of antigens for use as vaccines
US5536505A (en) * 1993-12-15 1996-07-16 Eastman Chemical Company Controlled release matrix system using cellulose acetate/poly-2-ethyl-2-oxazoline blends
US5523095A (en) * 1993-12-15 1996-06-04 Eastman Chemical Company Controlled release matrix system using cellulose acetate/polyvinylpyrrolidone blends
ES2120354B1 (es) * 1996-02-12 1999-07-01 Univ Sevilla Dispositivo terapeutico para direccionar farmacos hacia el tramo del tracto gastrointestinal deseado en funcion de las caracteristicas fisicoquimicas del mismo.
DE19628776A1 (de) * 1996-07-17 1998-01-22 Bayer Ag Oral applizierbare Granulate von Hexahydropyrazinderivaten
US20030100532A1 (en) * 1997-02-14 2003-05-29 Gary S. Jacob Use of n-substituted-1,5-dideoxy-1,5-imino-d-glucitol compounds in combination therapy for treating hepatitis virus infections
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EP1030839B1 (fr) 1997-11-10 2004-02-04 G.D. SEARLE & CO. Emploi d'iminosucres alkyles pour traiter la resistance multiple aux anticancereux
US6689759B1 (en) 1998-02-12 2004-02-10 G. D. Searle & Co. Methods of Treating hepatitis virus infections with N-substituted-1,5-dideoxy-1,5-imino-d-glucitol compounds in combination therapy
MY122185A (en) 1998-02-12 2006-03-31 Searle & Co Use of n-substituted-1, 5-dideoxy-1, 5-imino-d-glucitol compounds for treating hepatitis virus infections
DK1067910T3 (da) 1998-04-03 2004-10-04 Egalet As Komposition med styret afgivelse
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ATE402701T1 (de) 1999-02-12 2008-08-15 United Therapeutics Corp N-(8,8,8-trifluorooctyl)-1,5-dideoxy-1,5-imino- - glucitol zur behandlung von hepatitis-virus- infektionen
SE9903879D0 (sv) * 1999-10-28 1999-10-28 Ethical Pharmaceuticals Sweden Multipor food protection
CA2395231C (fr) 1999-12-23 2006-08-15 Pfizer Products Inc. Forme de dosage d'un medicament stratifie entraine par un hydrogel
WO2001054671A1 (fr) * 2000-01-27 2001-08-02 Tanabe Seiyaku Co., Ltd. Preparation a liberation prolongee et son procede de fabrication
CN1422156A (zh) * 2000-02-14 2003-06-04 法马西亚公司 N-取代的-1,5-二脱氧-1,5-亚氨基-d-葡萄糖醇化合物在治疗肝炎病毒感染中的用途
US6635277B2 (en) 2000-04-12 2003-10-21 Wockhardt Limited Composition for pulsatile delivery of diltiazem and process of manufacture
GB0106953D0 (en) * 2001-03-20 2001-05-09 Univ Aberdeen Neufofibrillary labels
US20040253310A1 (en) 2001-09-21 2004-12-16 Gina Fischer Morphine polymer release system
EP2957281A1 (fr) 2001-09-21 2015-12-23 Egalet Ltd. Systeme de liberation a base de polymere
US20040208936A1 (en) * 2002-07-22 2004-10-21 Roland Chorin Novel compositions
WO2004041252A1 (fr) 2002-11-08 2004-05-21 Egalet A/S Compositions de carvedilol a liberation commandee
US20060177506A1 (en) * 2003-03-17 2006-08-10 Shigeo Yanai Release control compositions
WO2004084868A1 (fr) 2003-03-26 2004-10-07 Egalet A/S Systeme de liberation regulee de morphine
ATE399538T1 (de) 2003-03-26 2008-07-15 Egalet As Matrixzubereitungen für die kontrollierte darreichung von arzneistoffen
US7115283B2 (en) * 2003-05-06 2006-10-03 Access Business Group International Llc Preparations for sustained release of nutraceuticals and methods of controllably releasing nutraceuticals
ES2272914T3 (es) * 2003-05-20 2007-05-01 Ethypharm Composicion farmaceutica oral de liberacion sostenida.
FR2855412B1 (fr) * 2003-05-27 2007-05-25 Menvielle Bourg Fabienn Joanny Composition a liberation prolongee de magnesium, et son application dans le domaine therapeutique, cosmetique et nutritionnel
JP2007520421A (ja) * 2003-06-26 2007-07-26 コリア リサーチ インスティテュート オブ ケミカル テクノロジー 経口投与用放出制御型薬物送達システム
US20060165793A1 (en) * 2003-08-04 2006-07-27 Koji Ukai Pharmaceutical preparation to be dispersed before administration
KR100615952B1 (ko) 2004-05-27 2006-08-28 한국화학연구원 서방형 약물 전달 시스템
CA2611081C (fr) * 2005-06-03 2016-05-31 Egalet A/S Systeme d'administration de medicaments permettant d'administrer des substances actives dispersees dans un milieu de dispersion
RU2309732C1 (ru) 2006-03-13 2007-11-10 Олег Ильич Эпштейн Спрессованная твердая оральная форма лекарственного препарата и способ получения твердой оральной формы лекарственного препарата
EP1880718B1 (fr) 2006-07-10 2011-09-21 Dr. R. Pfleger Chemische Fabrik GmbH Préparation pharmaceutique pour administration orale avec libération controlée d'actif dans l'intestin grêle et procédé de préparation
AU2008207200B2 (en) * 2007-01-16 2011-02-17 Egalet Ltd Use of i) a polyglycol and ii) an active drug substance for the preparation of a pharmaceutical composition for i) mitigating the risk of alcohol induced dose dumping and/or ii) reducing the risk of drug abuse
US20080181932A1 (en) * 2007-01-30 2008-07-31 Drugtech Corporation Compositions for oral delivery of pharmaceuticals
WO2008112388A1 (fr) 2007-03-14 2008-09-18 Drugtech Corporation Agencement spatial de particules dans un dispositif servant a boire, pour l'administration orale d'agents pharmaceutiques
CA2687192C (fr) 2007-06-04 2015-11-24 Egalet A/S Compositions pharmaceutiques a liberation controlee pour un effet prolonge
CA2696341C (fr) 2007-08-13 2016-05-17 Abuse Deterrent Pharmaceutical Llc Medicaments resistant aux abus, procedes d'utilisation et de fabrication
FR2931359B1 (fr) * 2008-05-20 2012-12-21 Menvielle Bourg Fabienne Joanny Utilisation d'une matrice pour administration orale de magnesium a liberation prolongee, et composition contenant cette matrice
FR2931361B1 (fr) * 2008-05-20 2012-08-31 Menvielle Bourg Fabienne Joanny Systeme a base de magnesium et son utilisation en cosmetique
CA2751667C (fr) 2009-02-06 2016-12-13 Egalet Ltd. Composition a liberation immediate resistant a une maltraitance par prise d'alcool
NZ597283A (en) 2009-06-24 2013-07-26 Egalet Ltd Controlled release formulations
EA030566B1 (ru) 2010-07-15 2018-08-31 Олег Ильич ЭПШТЕЙН Способ повышения терапевтической эффективности активированной-потенцированной формы антитела к эндогенной биомолекуле и фармацевтическая композиция
EA201590165A1 (ru) 2012-07-06 2015-08-31 Эгалет Лтд. Сдерживающие злоупотребление фармацевтические композиции для контролируемого высвобождения
US20140275038A1 (en) 2013-03-15 2014-09-18 Inspirion Delivery Technologies, Llc Abuse deterrent compositions and methods of use
US10729685B2 (en) 2014-09-15 2020-08-04 Ohemo Life Sciences Inc. Orally administrable compositions and methods of deterring abuse by intranasal administration

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DD146547A5 (de) 1978-07-15 1981-02-18 Boehringer Sohn Ingelheim Arzneimittel-retardform mit unloeslichen poroesen diffusionshuellen
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US5254347A (en) 1988-03-31 1993-10-19 Tanabe Seiyaku Co., Ltd. Controlled release pharmaceutical preparation and method for producing the same

Also Published As

Publication number Publication date
BG50712A3 (en) 1992-10-15
HUT50050A (en) 1989-12-28
NO891052L (no) 1989-10-02
NO891052D0 (no) 1989-03-13
CA1339078C (fr) 1997-07-29
KR890014095A (ko) 1989-10-21
PT90153B (pt) 1994-07-29
FI891163A0 (fi) 1989-03-10
DK156289A (da) 1989-10-01
EP0335560B2 (fr) 2002-01-23
IE64348B1 (en) 1995-07-26
FI891163A (fi) 1989-10-01
HU201882B (en) 1991-01-28
ES2059729T3 (es) 1994-11-16
NO178136B (no) 1995-10-23
IL89695A0 (en) 1989-09-28
DE68907762T2 (de) 1993-11-11
ZA892131B (en) 1989-11-29
PT90153A (pt) 1989-11-10
RU1836083C (ru) 1993-08-23
ATE91888T1 (de) 1993-08-15
NO178136C (no) 1996-01-31
DK156289D0 (da) 1989-03-30
HK76195A (en) 1995-05-26
PH25791A (fr) 1991-11-05
FI101344B (fi) 1998-06-15
IE891006L (en) 1989-09-30
DE68907762T3 (de) 2003-11-20
EP0335560B1 (fr) 1993-07-28
DE68907762D1 (de) 1993-09-02
EP0335560A3 (en) 1990-12-27
KR950007202B1 (ko) 1995-07-04
AU3227389A (en) 1989-10-05
US5068112A (en) 1991-11-26
EP0335560A2 (fr) 1989-10-04
ES2059729T5 (es) 2002-09-16
FR2629344A1 (fr) 1989-10-06
FR2629344B1 (fr) 1994-09-16
AU610711B2 (en) 1991-05-23

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Legal Events

Date Code Title Description
FG Patent granted

Owner name: TANABE SEIYAKU CO., . LTD.

MA Patent expired