ES8605165A1 - Procedimiento de preparar composiciones en emulsion de pros-taglandinas - Google Patents

Procedimiento de preparar composiciones en emulsion de pros-taglandinas

Info

Publication number
ES8605165A1
ES8605165A1 ES539828A ES539828A ES8605165A1 ES 8605165 A1 ES8605165 A1 ES 8605165A1 ES 539828 A ES539828 A ES 539828A ES 539828 A ES539828 A ES 539828A ES 8605165 A1 ES8605165 A1 ES 8605165A1
Authority
ES
Spain
Prior art keywords
phospholipid
prostaglandin
emulsified
compsn
compostion
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES539828A
Other languages
English (en)
Other versions
ES539828A0 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Mitsubishi Tanabe Pharma Corp
Original Assignee
Green Cross Corp Japan
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=11568883&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ES8605165(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Green Cross Corp Japan filed Critical Green Cross Corp Japan
Publication of ES8605165A1 publication Critical patent/ES8605165A1/es
Publication of ES539828A0 publication Critical patent/ES539828A0/es
Expired legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • A61K9/107Emulsions ; Emulsion preconcentrates; Micelles
    • A61K9/1075Microemulsions or submicron emulsions; Preconcentrates or solids thereof; Micelles, e.g. made of phospholipids or block copolymers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/557Eicosanoids, e.g. leukotrienes or prostaglandins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Dispersion Chemistry (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Colloid Chemistry (AREA)

Abstract

METODO PARA PREPARAR EMULSIONES DE PROSTAGLANDINAS. COMPRENDE SELECCIONAR UNA PROSTAGLANDINA DEL GRUPO: PGF2ALFA, PGE2, PGD2, PGF1ALFA, PGE1, PGA1, PGI2, PGB1 Y SUS DERIVADOS; AÑADIR ESTA A UN ACEITE VEGETAL DEL GRUPO: SOJA, SEMILLA ALGODON, SESAMO, CARTAMO Y MAIZ; MEZCLAR EL RESULTADO CON UN EMULSIONANTE FOSFOLIPIDO LIBRE DE FOSFATIDILETANOLAMINA, SIENDO PREDOMINANTEMENTE FOSFATIDILCOLINA. SE CALIENTE LA DISOLUCION A 40-75JC Y SE FORMA UNA EMULSION BRUTA AÑADIENDO AGUA Y CALENTANDO A 20-80JC. SE HOMOGEINIZA HACIENDO PASAR LA EMULSION VARIAS VECES POR DOS ETAPAS A PRESION. SE AÑADEN ESTABILIZANTE, AGENTE ISOTONIFICANTE Y UN COMPUESTO DE ALTO PESO MOLECULAR.-
ES539828A 1984-01-12 1985-01-11 Procedimiento de preparar composiciones en emulsion de pros-taglandinas Expired ES8605165A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP59003858A JPH0818989B2 (ja) 1984-01-12 1984-01-12 脂肪乳剤中のプロスタグランジンの安定化方法

Publications (2)

Publication Number Publication Date
ES8605165A1 true ES8605165A1 (es) 1986-04-01
ES539828A0 ES539828A0 (es) 1986-04-01

Family

ID=11568883

Family Applications (1)

Application Number Title Priority Date Filing Date
ES539828A Expired ES8605165A1 (es) 1984-01-12 1985-01-11 Procedimiento de preparar composiciones en emulsion de pros-taglandinas

Country Status (6)

Country Link
US (1) US4684633A (es)
EP (1) EP0150732B1 (es)
JP (1) JPH0818989B2 (es)
CA (1) CA1239873A (es)
DE (2) DE3570596D1 (es)
ES (1) ES8605165A1 (es)

Families Citing this family (38)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR920007569B1 (ko) * 1984-11-30 1992-09-07 쥬우가이 세이야꾸 가부시끼가이샤 프로스타글란딘 e 유도체의 안정한 제제의 제조방법
JPS61289034A (ja) * 1985-06-17 1986-12-19 Teijin Ltd イソカルバサイクリン類脂肪乳剤
US4997823A (en) * 1986-02-18 1991-03-05 Syntex (U.S.A.) Inc. Anti-infective injectable formulations
US6759057B1 (en) 1986-06-12 2004-07-06 The Liposome Company, Inc. Methods and compositions using liposome-encapsulated non-steroidal anti-inflammatory drugs
US5811118A (en) * 1987-05-22 1998-09-22 The Liposome Company, Inc. Methods of treatment using unilamellar liposomal arachidonic acid metabolite formulations
US5082664A (en) * 1987-05-22 1992-01-21 The Liposome Company, Inc. Prostaglandin-lipid formulations
US5262168A (en) * 1987-05-22 1993-11-16 The Liposome Company, Inc. Prostaglandin-lipid formulations
US5925375A (en) * 1987-05-22 1999-07-20 The Liposome Company, Inc. Therapeutic use of multilamellar liposomal prostaglandin formulations
US4840968A (en) * 1987-10-02 1989-06-20 Tsuyoshi Ohnishi Preparation and uses of new prostaglandin derivatives which protect cell membranes against ischemic, physical, chemical, and biological injuries
JPH0669966B2 (ja) * 1989-07-05 1994-09-07 株式会社ミドリ十字 血管造影補助剤
GB8919172D0 (en) * 1989-08-23 1989-10-04 Univ Nottingham Useful composition
JPH03101622A (ja) * 1989-09-11 1991-04-26 Green Cross Corp:The 肝炎予防治療剤
US5194670A (en) * 1989-10-16 1993-03-16 Yutaka Mizushima, Asahi Glass Company Ltd. Emulsion of lipid containing a prostaglandin analogue
JP2602964B2 (ja) * 1989-10-16 1997-04-23 裕 水島 プロスタグランジン類縁体およびその脂肪乳剤
US5882678A (en) * 1990-01-12 1999-03-16 The Liposome Co, Inc. Interdigitation-fusion liposomes containing arachidonic acid metabolites
US5817646A (en) * 1991-11-15 1998-10-06 Laboratoires Inocosm Polar lipid composition of plant origin
DE4309579C3 (de) * 1993-03-24 2000-01-27 Sanol Arznei Schwarz Gmbh Pharmazeutische Zusammensetzung in Form einer Packung
SE9303281D0 (sv) * 1993-10-07 1993-10-07 Astra Ab New formulation
US5840328A (en) * 1994-01-11 1998-11-24 The Liposome Company, Inc. Treatment using arachidonic acid metabolite and particulate formulations
CA2231682A1 (en) * 1995-09-13 1997-03-20 Junzo Seki Pge1-containing freeze-dried preparation and the production thereof
DE19645657A1 (de) * 1996-11-06 1998-05-28 Rhone Poulenc Rorer Gmbh Phospholipidische Zusammensetzung, Verfahren zur Herstellung einer derartigen Zusammensetzung und Verwendung derselben
US6103765A (en) 1997-07-09 2000-08-15 Androsolutions, Inc. Methods for treating male erectile dysfunction
CA2295595A1 (en) 1997-07-09 1999-01-21 Androsolutions, Inc. Improved methods and compositions for treating male erectile dysfunction
KR20010023360A (ko) 1997-08-27 2001-03-26 미즈시마 유타카 혈관신생 촉진제
KR100446960B1 (ko) * 2001-12-04 2004-09-01 김종국 프로스타글란딘 e1을 포함하는 온도감응성 에멀젼 외용제조성물
EP1562557B2 (en) 2002-11-01 2016-11-16 University of Medicine and Dentistry of New Jersey Geodate delivery vehicles
TWI495471B (zh) * 2003-08-12 2015-08-11 R Tech Ueno Ltd 促進毛髮生長之組成物及方法
ES2314354T3 (es) * 2004-11-09 2009-03-16 Novagali Pharma S.A. Emulsion de tipo aceite en agua con baja concentracion de agente cationico y potencial zeta positivo.
AU2005304034B2 (en) * 2004-11-09 2012-02-16 Santen Sas Ophthalmic emulsions containing an immunosuppressive agent
ES2351358T3 (es) * 2005-10-10 2011-02-03 Novagali Pharma S.A. Emulsiones oftálmicas que contienen prostaglandinas.
JP5193870B2 (ja) * 2006-09-05 2013-05-08 キユーピー株式会社 プロスタグランジン脂肪乳剤およびその製造方法、ならびにその安定化方法および乳化剤
GB0701609D0 (en) 2007-01-29 2007-03-07 Boc Group Plc Vacuum pump
US20080234376A1 (en) * 2007-03-21 2008-09-25 Taiwan Liposome Company (A Taiwan Corporation) Emulsion composition comprising prostaglandin e1
WO2009093650A1 (ja) * 2008-01-24 2009-07-30 Techno Guard Co. Ltd. プロスタグランジン含有脂肪乳剤およびその製造方法
EP2228058A1 (en) 2009-03-04 2010-09-15 Novagali Pharma S.A. Anionic oil-in-water emulsion containing prostaglandins and uses thereof
EP2389939A1 (en) 2010-05-28 2011-11-30 Novagali Pharma S.A. Use of prostaglandins F2alpha and analogues for the healing of corneal and conjunctival lesions
WO2012133554A1 (ja) 2011-03-31 2012-10-04 富士フイルム株式会社 プロスタグランジン含有脂肪乳剤
TWI754659B (zh) 2016-08-08 2022-02-11 台灣微脂體股份有限公司 用於製備含有弱酸性劑之微脂體組合物的傳輸載體、方法及套組

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3069322A (en) * 1958-05-28 1962-12-18 Bergstrom Sune Pge and pgf
US4190669A (en) * 1976-03-08 1980-02-26 The Regents Of The University Of Michigan Method for treating psoriasis
IT1202370B (it) * 1976-07-12 1989-02-09 Hoffmann La Roche Soluzioni inietabili in cui l'atti vita' emolitica degli agenti di formazione di micelle naturali e' evitata mediante l'aggiunta di lipoidi e relativi prodotti
JPS5562010A (en) * 1978-10-31 1980-05-10 Ajinomoto Co Inc Fat emulsion for intravenous injection
JPS6030652B2 (ja) * 1979-05-07 1985-07-17 株式会社ミドリ十字 静脈注射用脂肪乳剤
JPS58104624A (ja) * 1981-12-16 1983-06-22 Kao Corp 乳化組成物
JPS58222014A (ja) * 1982-06-18 1983-12-23 Taisho Pharmaceut Co Ltd プロスタグランジンe↓1脂肪乳剤
JPS59912A (ja) * 1982-06-26 1984-01-06 Tokyo Electric Co Ltd 放電灯安定器
US4563354A (en) * 1983-10-26 1986-01-07 Kabivitrum Ab Oil-in-water emulsion for parenteral administration

Also Published As

Publication number Publication date
DE3570596D1 (en) 1989-07-06
CA1239873A (en) 1988-08-02
DE150732T1 (de) 1986-07-24
JPH0818989B2 (ja) 1996-02-28
ES539828A0 (es) 1986-04-01
JPS60149524A (ja) 1985-08-07
EP0150732A3 (en) 1985-08-21
EP0150732B1 (en) 1989-05-31
EP0150732A2 (en) 1985-08-07
US4684633A (en) 1987-08-04

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Legal Events

Date Code Title Description
PC1A Transfer granted
PC1A Transfer granted
FD1A Patent lapsed

Effective date: 20050706