ES479446A1 - Un metodo de producir derivados de bencimidazol. - Google Patents
Un metodo de producir derivados de bencimidazol.Info
- Publication number
- ES479446A1 ES479446A1 ES479446A ES479446A ES479446A1 ES 479446 A1 ES479446 A1 ES 479446A1 ES 479446 A ES479446 A ES 479446A ES 479446 A ES479446 A ES 479446A ES 479446 A1 ES479446 A1 ES 479446A1
- Authority
- ES
- Spain
- Prior art keywords
- substituted
- aryl
- heterocyclic group
- benzyl
- alkyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- BASPJMOEXODOEJ-UHFFFAOYSA-N 3h-benzimidazole-5-sulfonamide Chemical class NS(=O)(=O)C1=CC=C2NC=NC2=C1 BASPJMOEXODOEJ-UHFFFAOYSA-N 0.000 title 1
- MXMZCLLIUQEKSN-UHFFFAOYSA-N benzimidazoline Chemical class C1=CC=C2NCNC2=C1 MXMZCLLIUQEKSN-UHFFFAOYSA-N 0.000 title 1
- 125000000623 heterocyclic group Chemical group 0.000 abstract 6
- 125000003118 aryl group Chemical group 0.000 abstract 4
- 125000001797 benzyl group Chemical group [H]C1=C([H])C([H])=C(C([H])=C1[H])C([H])([H])* 0.000 abstract 4
- 125000003107 substituted aryl group Chemical group 0.000 abstract 4
- 125000000217 alkyl group Chemical group 0.000 abstract 3
- 150000002431 hydrogen Chemical class 0.000 abstract 3
- 229910052739 hydrogen Inorganic materials 0.000 abstract 3
- 239000001257 hydrogen Substances 0.000 abstract 3
- 125000002252 acyl group Chemical group 0.000 abstract 2
- 125000003710 aryl alkyl group Chemical group 0.000 abstract 2
- 229910052736 halogen Inorganic materials 0.000 abstract 2
- 150000002367 halogens Chemical group 0.000 abstract 2
- 150000003839 salts Chemical class 0.000 abstract 2
- QUVNDNJVCZLXNI-UHFFFAOYSA-N N=1C=2C=C(Cl)C(S(=O)(=O)N)=CC=2NC=1N1C(=O)C1=O Chemical compound N=1C=2C=C(Cl)C(S(=O)(=O)N)=CC=2NC=1N1C(=O)C1=O QUVNDNJVCZLXNI-UHFFFAOYSA-N 0.000 abstract 1
- -1 amino, substituted amino, guanidino, substituted guanidino Chemical group 0.000 abstract 1
- 230000003276 anti-hypertensive effect Effects 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 239000002934 diuretic Substances 0.000 abstract 1
- 230000001882 diuretic effect Effects 0.000 abstract 1
- FDDDEECHVMSUSB-UHFFFAOYSA-N sulfanilamide Chemical compound NC1=CC=C(S(N)(=O)=O)C=C1 FDDDEECHVMSUSB-UHFFFAOYSA-N 0.000 abstract 1
- 229940124530 sulfonamide Drugs 0.000 abstract 1
- 125000002023 trifluoromethyl group Chemical group FC(F)(F)* 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/06—Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/10—Antioedematous agents; Diuretics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/06—Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
- C07D235/08—Radicals containing only hydrogen and carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/18—Benzimidazoles; Hydrogenated benzimidazoles with aryl radicals directly attached in position 2
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/24—Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D235/30—Nitrogen atoms not forming part of a nitro radical
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Public Health (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Hematology (AREA)
- Diabetes (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US89504878A | 1978-04-10 | 1978-04-10 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES479446A1 true ES479446A1 (es) | 1979-08-01 |
Family
ID=25403870
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES479446A Expired ES479446A1 (es) | 1978-04-10 | 1979-04-09 | Un metodo de producir derivados de bencimidazol. |
Country Status (19)
| Country | Link |
|---|---|
| JP (1) | JPS54138561A (enExample) |
| AT (1) | AT372951B (enExample) |
| AU (1) | AU531086B2 (enExample) |
| BE (1) | BE875425A (enExample) |
| CA (1) | CA1126280A (enExample) |
| DE (1) | DE2914084A1 (enExample) |
| DK (1) | DK139079A (enExample) |
| ES (1) | ES479446A1 (enExample) |
| FI (1) | FI74461C (enExample) |
| FR (1) | FR2422644A1 (enExample) |
| GB (1) | GB2018766B (enExample) |
| GR (1) | GR68483B (enExample) |
| IL (1) | IL57105A (enExample) |
| IT (1) | IT1193755B (enExample) |
| NL (1) | NL7902802A (enExample) |
| NZ (1) | NZ190136A (enExample) |
| PT (1) | PT69458A (enExample) |
| SE (1) | SE446532B (enExample) |
| ZA (1) | ZA791726B (enExample) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN102070466A (zh) * | 2010-12-28 | 2011-05-25 | 天津市筠凯化工科技有限公司 | 5-氯-2-硝基苯胺制备方法 |
| CN108558712A (zh) * | 2018-06-20 | 2018-09-21 | 新乡市锦源化工有限公司 | 一种以乙酰苯胺为原料合成高纯度对氨基苯磺酰胺的方法及对氨基苯磺酰胺 |
| CN110305018B (zh) * | 2019-06-06 | 2022-07-15 | 浙江普洛家园药业有限公司 | 一种3-溴-2-氟硝基苯的制备方法 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CH404675A (de) * | 1961-06-29 | 1965-12-31 | Siegfried Ag | Verfahren zur Herstellung neuer heterocyclischer Sulfonamidoverbindungen |
| FR1469504A (fr) * | 1964-10-22 | 1967-02-17 | Fisons Pest Control Ltd | Composés insecticides |
| FR1477792A (fr) * | 1965-03-24 | 1967-04-21 | Fisons Pest Control Ltd | Nouveaux benzimidazoles |
| GB1163711A (en) * | 1966-01-13 | 1969-09-10 | Fisons Pest Control Ltd | Substituted Benzimidazoles and Biocidally-Active Compositions |
| GB1356244A (en) * | 1970-07-29 | 1974-06-12 | Fisons Ltd | Substituted benzimidazole parasiticides |
-
1979
- 1979-03-26 CA CA324,146A patent/CA1126280A/en not_active Expired
- 1979-04-02 FI FI791083A patent/FI74461C/fi not_active IP Right Cessation
- 1979-04-02 SE SE7902911A patent/SE446532B/sv not_active IP Right Cessation
- 1979-04-02 AU AU45675/79A patent/AU531086B2/en not_active Ceased
- 1979-04-03 GR GR58771A patent/GR68483B/el unknown
- 1979-04-04 DK DK139079A patent/DK139079A/da not_active IP Right Cessation
- 1979-04-06 GB GB7912255A patent/GB2018766B/en not_active Expired
- 1979-04-07 DE DE19792914084 patent/DE2914084A1/de not_active Withdrawn
- 1979-04-09 AT AT0263379A patent/AT372951B/de not_active IP Right Cessation
- 1979-04-09 ES ES479446A patent/ES479446A1/es not_active Expired
- 1979-04-09 FR FR7908945A patent/FR2422644A1/fr active Granted
- 1979-04-09 PT PT69458A patent/PT69458A/pt unknown
- 1979-04-09 JP JP4211979A patent/JPS54138561A/ja active Granted
- 1979-04-09 NZ NZ190136A patent/NZ190136A/xx unknown
- 1979-04-09 BE BE0/194480A patent/BE875425A/xx not_active IP Right Cessation
- 1979-04-10 NL NL7902802A patent/NL7902802A/xx not_active Application Discontinuation
- 1979-04-10 ZA ZA791726A patent/ZA791726B/xx unknown
- 1979-04-10 IT IT48686/79A patent/IT1193755B/it active
- 1979-04-22 IL IL57105A patent/IL57105A/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| JPH0250904B2 (enExample) | 1990-11-05 |
| IL57105A0 (en) | 1979-07-25 |
| FR2422644A1 (fr) | 1979-11-09 |
| CA1126280A (en) | 1982-06-22 |
| ATA263379A (de) | 1983-04-15 |
| ZA791726B (en) | 1980-05-28 |
| GB2018766B (en) | 1982-09-22 |
| DK139079A (da) | 1979-10-11 |
| IT7948686A0 (it) | 1979-04-10 |
| FI74461C (fi) | 1988-02-08 |
| JPS54138561A (en) | 1979-10-27 |
| AU4567579A (en) | 1979-10-18 |
| FI74461B (fi) | 1987-10-30 |
| FI791083A7 (fi) | 1979-10-11 |
| DE2914084A1 (de) | 1979-10-25 |
| AU531086B2 (en) | 1983-08-11 |
| AT372951B (de) | 1983-12-12 |
| NL7902802A (nl) | 1979-10-12 |
| SE7902911L (sv) | 1979-10-11 |
| SE446532B (sv) | 1986-09-22 |
| IT1193755B (it) | 1988-08-24 |
| IL57105A (en) | 1983-10-31 |
| FR2422644B1 (enExample) | 1982-12-17 |
| BE875425A (fr) | 1979-07-31 |
| GR68483B (enExample) | 1982-01-04 |
| NZ190136A (en) | 1982-11-23 |
| GB2018766A (en) | 1979-10-24 |
| PT69458A (en) | 1979-05-01 |
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