ES309169A1 - Un procedimiento para la preparacion de derivados benzodiazepinicos. - Google Patents

Un procedimiento para la preparacion de derivados benzodiazepinicos.

Info

Publication number
ES309169A1
ES309169A1 ES0309169A ES309169A ES309169A1 ES 309169 A1 ES309169 A1 ES 309169A1 ES 0309169 A ES0309169 A ES 0309169A ES 309169 A ES309169 A ES 309169A ES 309169 A1 ES309169 A1 ES 309169A1
Authority
ES
Spain
Prior art keywords
halogen
alkyl
see formula
represents hydrogen
hydrogen
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES0309169A
Other languages
English (en)
Spanish (es)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
F Hoffmann La Roche AG
Original Assignee
F Hoffmann La Roche AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=23348328&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ES309169(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by F Hoffmann La Roche AG filed Critical F Hoffmann La Roche AG
Publication of ES309169A1 publication Critical patent/ES309169A1/es
Expired legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients

Landscapes

  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Supply And Distribution Of Alternating Current (AREA)
  • Multicomponent Fibers (AREA)
ES0309169A 1964-02-11 1965-02-10 Un procedimiento para la preparacion de derivados benzodiazepinicos. Expired ES309169A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US343941A US3299053A (en) 1964-02-11 1964-02-11 Novel 1-and/or 4-substituted alkyl 5-aromatic-3h-1, 4-benzodiazepines and benzodiazepine-2-ones

Publications (1)

Publication Number Publication Date
ES309169A1 true ES309169A1 (es) 1965-10-16

Family

ID=23348328

Family Applications (4)

Application Number Title Priority Date Filing Date
ES0309169A Expired ES309169A1 (es) 1964-02-11 1965-02-10 Un procedimiento para la preparacion de derivados benzodiazepinicos.
ES0309170A Expired ES309170A1 (es) 1964-02-11 1965-02-10 Un procedimiento para preparar derivados benzodiazepinicos.
ES0309168A Expired ES309168A1 (es) 1964-02-11 1965-02-10 Un procedimiento para la preparacion de derivados benzodiazepinicos
ES0309167A Expired ES309167A2 (es) 1964-02-11 1965-02-10 Procedimiento para la fabricacion de derivados benzodiazepinicos

Family Applications After (3)

Application Number Title Priority Date Filing Date
ES0309170A Expired ES309170A1 (es) 1964-02-11 1965-02-10 Un procedimiento para preparar derivados benzodiazepinicos.
ES0309168A Expired ES309168A1 (es) 1964-02-11 1965-02-10 Un procedimiento para la preparacion de derivados benzodiazepinicos
ES0309167A Expired ES309167A2 (es) 1964-02-11 1965-02-10 Procedimiento para la fabricacion de derivados benzodiazepinicos

Country Status (13)

Country Link
US (1) US3299053A (index.php)
BE (4) BE659442A (index.php)
BR (4) BR6567051D0 (index.php)
CH (4) CH460030A (index.php)
DE (4) DE1545933A1 (index.php)
DK (3) DK118249B (index.php)
ES (4) ES309169A1 (index.php)
FR (6) FR4123M (index.php)
GB (4) GB1077358A (index.php)
IL (4) IL22869A (index.php)
NL (4) NL6501579A (index.php)
NO (3) NO117367B (index.php)
SE (4) SE309597B (index.php)

Families Citing this family (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NO120269B (index.php) * 1965-11-02 1970-09-28 Hoffmann La Roche
US3464978A (en) * 1967-04-21 1969-09-02 Hoffmann La Roche 1-substituted urea alkyl 1,2-dihydro-1,4-benzodiazepines and benzodiazepin - 2-ones
US3523939A (en) * 1967-07-03 1970-08-11 Hoffmann La Roche 5-(2,6-disubstituted phenyl)-1,4-benzodiazepines and methods for their preparation
US3506403A (en) * 1967-12-19 1970-04-14 Hoffmann La Roche Colorimetric method for determining iron in fluids
US3506404A (en) * 1967-12-19 1970-04-14 Hoffmann La Roche Colorimetric method for determining iron in blood
US3609146A (en) * 1968-11-01 1971-09-28 Sandoz Ag Substituted benzodiazepinone derivatives
DE2008612A1 (de) * 1969-03-13 1970-10-01 F. Hoffmann-La Roche & Co Ag, Basel (Schweiz) Benzodiazepin-Derivate
US3691157A (en) * 1970-08-12 1972-09-12 Rodney Ian Fryer Preparation of 7-substituted-1-(2-diethylaminoethyl)-5-(2-halophenyl)-1,3-dihydro-2h-1,4-benzodiazepin-2-ones
AT314541B (de) * 1970-10-19 1974-04-10 Sumitomo Chemical Co Verfahren zur Herstellung von neuen Benzodiazepinen und ihren Salzen
US3678038A (en) * 1971-04-01 1972-07-18 Hoffmann La Roche 1,4-benzodiazepin-5-ones and methods for the preparation thereof
US3856802A (en) * 1971-05-10 1974-12-24 Upjohn Co 1,6-DISUBSTITUTED-4H-5-{8 4,3-a{9 BENZODIAZEPINES
US3872089A (en) * 1971-05-14 1975-03-18 Hoffmann La Roche Substituted thienodiazepines
US4008223A (en) * 1971-12-09 1977-02-15 Deutsche Gold- Und Silber-Scheideanstalt Vormals Roessler 6-Aza-3H-1,4-benzodiazepines
USRE31071E (en) * 1971-12-09 1982-11-02 Deutsche Gold- Und Silber-Scheideanstalt Vormals Roessler 6-Aza-3H-1,4-benzodiazepines
US3859276A (en) * 1972-12-13 1975-01-07 Merck & Co Inc 7-chloro-1,3-dihydro-5-2-polyfluoroalkoxyphenyl)-2h-1,4-benzodiazepin-2-ones
GB1414370A (en) * 1973-08-24 1975-11-19 Grindstedvaerket As Benzodiazepines and their production
US4232016A (en) * 1974-12-20 1980-11-04 Merck Patent Gesellschaft Mit Beschraenkter Haftung 3-Fluorobenzodiazepines
US4246270A (en) * 1976-05-26 1981-01-20 E. I. Du Pont De Nemours And Company 3-Fluorobenzodiazepines and compositions and uses thereof
DE2852606A1 (de) * 1977-12-14 1979-06-21 Gerot Pharmazeutika 3-di-n-propyl-acetoxy-benzodiazepin-2-one und verfahren zu deren herstellung
AT361492B (de) * 1978-12-18 1981-03-10 Gerot Pharmazeutika Verfahren zur herstellung von neuen 3-hydroxy- 1,4-benzodiazepin-2-onen
US8530463B2 (en) * 2007-05-07 2013-09-10 Hale Biopharma Ventures Llc Multimodal particulate formulations
CN101686983A (zh) 2007-05-10 2010-03-31 Amr科技公司 芳基和杂芳基取代的四氢苯并-1,4-二氮杂䓬及其阻断去甲肾上腺素、多巴胺和5-羟色胺重摄取的用途
ES2586032T3 (es) 2008-03-28 2016-10-11 Hale Biopharma Ventures, Llc Administración de composiciones de benzodiazepinas
JP6219272B2 (ja) 2011-06-14 2017-10-25 ヘイル バイオファーマ ベンチャーズ,エルエルシー ベンゾジアゼピン組成物の投与

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3121076A (en) * 1964-02-11 Benzodiazepinones and processes
US3109843A (en) * 1963-11-05 Process for preparing
US2461038A (en) * 1947-05-15 1949-02-08 Searle & Co Chemical compositions and the preparation thereof
US2532292A (en) * 1947-12-12 1950-12-05 Searle & Co Diarylmethyl ethers of amino alkanols
US2576106A (en) * 1948-07-13 1951-11-27 Searle & Co N-dicyclohexyl, dialkylaminoalkanamides
US2687414A (en) * 1948-11-26 1954-08-24 Searle & Co Method for producing aromatic aminoalkyl amines

Also Published As

Publication number Publication date
NO119798B (index.php) 1970-07-06
NL6501632A (index.php) 1965-08-12
ES309170A1 (es) 1965-07-16
IL22903A (en) 1969-03-27
US3299053A (en) 1967-01-17
SE321477B (index.php) 1970-03-09
GB1052144A (index.php)
BR6567054D0 (pt) 1973-08-14
FR4772M (index.php) 1967-01-23
BE659444A (index.php) 1965-08-09
DE1545935A1 (de) 1969-12-11
NL141781B (nl) 1974-04-16
BE659443A (index.php) 1965-08-09
SE307952B (index.php) 1969-01-27
SE307953B (index.php) 1969-01-27
FR4609M (index.php) 1966-11-21
NO118273B (index.php) 1969-12-08
CH460793A (de) 1968-08-15
BE659445A (index.php) 1965-08-09
DK118249B (da) 1970-07-27
IL22935A (en) 1969-11-30
BR6567051D0 (pt) 1973-08-14
GB1098242A (en) 1968-01-10
NL6501578A (index.php) 1965-08-12
GB1077358A (en) 1967-07-26
CH458372A (de) 1968-06-30
IL22869A (en) 1968-11-27
DE1545936B2 (de) 1975-09-18
NO117367B (index.php) 1969-08-04
ES309168A1 (es) 1965-10-01
BR6567055D0 (pt) 1973-08-02
FR4138M (index.php) 1966-05-02
CH467787A (de) 1969-01-31
NL6501631A (index.php) 1965-08-12
IL22902A (en) 1969-01-29
DK105984C (da) 1966-12-05
DE1545933A1 (de) 1969-12-18
FR1455059A (fr) 1966-10-07
CH460030A (de) 1968-07-31
NL6501579A (index.php) 1965-08-12
GB1051795A (index.php)
FR1443116A (fr) 1966-06-24
SE309597B (index.php) 1969-03-31
ES309167A2 (es) 1965-10-01
DE1545936A1 (de) 1969-12-18
DK107032C (da) 1967-04-17
BE659442A (index.php) 1965-08-09
BR6567053D0 (pt) 1973-12-26
FR4123M (index.php) 1966-04-25
DE1545934A1 (de) 1970-10-22

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