CH458372A - Verfahren zur Herstellung von Benzodiazepin-Derivaten - Google Patents

Verfahren zur Herstellung von Benzodiazepin-Derivaten

Info

Publication number
CH458372A
CH458372A CH118265A CH118265A CH458372A CH 458372 A CH458372 A CH 458372A CH 118265 A CH118265 A CH 118265A CH 118265 A CH118265 A CH 118265A CH 458372 A CH458372 A CH 458372A
Authority
CH
Switzerland
Prior art keywords
preparation
benzodiazepine derivatives
benzodiazepine
derivatives
Prior art date
Application number
CH118265A
Other languages
English (en)
Inventor
A Archer Giles
Ian Fryer Rodney
Reeder Earl
Henryk Sternbach Leo
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=23348328&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CH458372(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of CH458372A publication Critical patent/CH458372A/de

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients

Landscapes

  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Supply And Distribution Of Alternating Current (AREA)
  • Multicomponent Fibers (AREA)
CH118265A 1964-02-11 1965-01-28 Verfahren zur Herstellung von Benzodiazepin-Derivaten CH458372A (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US343941A US3299053A (en) 1964-02-11 1964-02-11 Novel 1-and/or 4-substituted alkyl 5-aromatic-3h-1, 4-benzodiazepines and benzodiazepine-2-ones

Publications (1)

Publication Number Publication Date
CH458372A true CH458372A (de) 1968-06-30

Family

ID=23348328

Family Applications (4)

Application Number Title Priority Date Filing Date
CH102465A CH460030A (de) 1964-02-11 1965-01-25 Verfahren zur Herstellung von Benzodiazepin-Derivaten
CH332768A CH460793A (de) 1964-02-11 1965-01-25 Verfahren zur Herstellung von Benzodiazepin-Derivaten
CH118165A CH467787A (de) 1964-02-11 1965-01-28 Verfahren zur Herstellung von Benzodiazepin-Derivaten
CH118265A CH458372A (de) 1964-02-11 1965-01-28 Verfahren zur Herstellung von Benzodiazepin-Derivaten

Family Applications Before (3)

Application Number Title Priority Date Filing Date
CH102465A CH460030A (de) 1964-02-11 1965-01-25 Verfahren zur Herstellung von Benzodiazepin-Derivaten
CH332768A CH460793A (de) 1964-02-11 1965-01-25 Verfahren zur Herstellung von Benzodiazepin-Derivaten
CH118165A CH467787A (de) 1964-02-11 1965-01-28 Verfahren zur Herstellung von Benzodiazepin-Derivaten

Country Status (13)

Country Link
US (1) US3299053A (de)
BE (4) BE659442A (de)
BR (4) BR6567051D0 (de)
CH (4) CH460030A (de)
DE (4) DE1545933A1 (de)
DK (3) DK118249B (de)
ES (4) ES309167A2 (de)
FR (6) FR4123M (de)
GB (4) GB1077358A (de)
IL (4) IL22869A (de)
NL (4) NL6501578A (de)
NO (3) NO117367B (de)
SE (4) SE307952B (de)

Families Citing this family (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NO120269B (de) * 1965-11-02 1970-09-28 Hoffmann La Roche
US3464978A (en) * 1967-04-21 1969-09-02 Hoffmann La Roche 1-substituted urea alkyl 1,2-dihydro-1,4-benzodiazepines and benzodiazepin - 2-ones
US3523939A (en) * 1967-07-03 1970-08-11 Hoffmann La Roche 5-(2,6-disubstituted phenyl)-1,4-benzodiazepines and methods for their preparation
US3506404A (en) * 1967-12-19 1970-04-14 Hoffmann La Roche Colorimetric method for determining iron in blood
US3506403A (en) * 1967-12-19 1970-04-14 Hoffmann La Roche Colorimetric method for determining iron in fluids
US3609146A (en) * 1968-11-01 1971-09-28 Sandoz Ag Substituted benzodiazepinone derivatives
IL33961A (en) * 1969-03-13 1973-03-30 Sparamedica Ag Benzodiazepine aminoalkyl carboxylates,their preparation and pharmaceutical compositions containing them
US3691157A (en) * 1970-08-12 1972-09-12 Rodney Ian Fryer Preparation of 7-substituted-1-(2-diethylaminoethyl)-5-(2-halophenyl)-1,3-dihydro-2h-1,4-benzodiazepin-2-ones
AT314541B (de) * 1970-10-19 1974-04-10 Sumitomo Chemical Co Verfahren zur Herstellung von neuen Benzodiazepinen und ihren Salzen
US3678038A (en) * 1971-04-01 1972-07-18 Hoffmann La Roche 1,4-benzodiazepin-5-ones and methods for the preparation thereof
US3856802A (en) * 1971-05-10 1974-12-24 Upjohn Co 1,6-DISUBSTITUTED-4H-5-{8 4,3-a{9 BENZODIAZEPINES
US3872089A (en) * 1971-05-14 1975-03-18 Hoffmann La Roche Substituted thienodiazepines
USRE31071E (en) * 1971-12-09 1982-11-02 Deutsche Gold- Und Silber-Scheideanstalt Vormals Roessler 6-Aza-3H-1,4-benzodiazepines
US4008223A (en) * 1971-12-09 1977-02-15 Deutsche Gold- Und Silber-Scheideanstalt Vormals Roessler 6-Aza-3H-1,4-benzodiazepines
US3859276A (en) * 1972-12-13 1975-01-07 Merck & Co Inc 7-chloro-1,3-dihydro-5-2-polyfluoroalkoxyphenyl)-2h-1,4-benzodiazepin-2-ones
GB1414370A (en) * 1973-08-24 1975-11-19 Grindstedvaerket As Benzodiazepines and their production
US4232016A (en) * 1974-12-20 1980-11-04 Merck Patent Gesellschaft Mit Beschraenkter Haftung 3-Fluorobenzodiazepines
US4246270A (en) * 1976-05-26 1981-01-20 E. I. Du Pont De Nemours And Company 3-Fluorobenzodiazepines and compositions and uses thereof
FI783743A (fi) * 1977-12-14 1979-06-15 Gerot Pharmazeutika Foerfarande foer framstaellning av 3-di-n-propyl-acetoxi-benzodiazepin-2-oner
AT361492B (de) * 1978-12-18 1981-03-10 Gerot Pharmazeutika Verfahren zur herstellung von neuen 3-hydroxy- 1,4-benzodiazepin-2-onen
US8530463B2 (en) * 2007-05-07 2013-09-10 Hale Biopharma Ventures Llc Multimodal particulate formulations
JP2010526825A (ja) 2007-05-10 2010-08-05 エーエムアール テクノロジー インコーポレイテッド アリール置換およびヘテロアリール置換テトラヒドロベンゾ−1,4−ジアゼピンならびにノルエピネフリン、ドーパミンおよびセロトニンの再取り込みを遮断するためのその使用
JP5613657B2 (ja) 2008-03-28 2014-10-29 ヘイル バイオファーマ ベンチャーズ,エルエルシー ベンゾジアゼピン組成物の投与
CN107737100A (zh) 2011-06-14 2018-02-27 哈尔生物药投资有限责任公司 苯二氮卓组合物的投与

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3109843A (en) * 1963-11-05 Process for preparing
US3121076A (en) * 1964-02-11 Benzodiazepinones and processes
US2461038A (en) * 1947-05-15 1949-02-08 Searle & Co Chemical compositions and the preparation thereof
US2532292A (en) * 1947-12-12 1950-12-05 Searle & Co Diarylmethyl ethers of amino alkanols
US2576106A (en) * 1948-07-13 1951-11-27 Searle & Co N-dicyclohexyl, dialkylaminoalkanamides
US2687414A (en) * 1948-11-26 1954-08-24 Searle & Co Method for producing aromatic aminoalkyl amines

Also Published As

Publication number Publication date
DK107032C (da) 1967-04-17
IL22902A (en) 1969-01-29
SE309597B (de) 1969-03-31
BE659445A (de) 1965-08-09
IL22935A (en) 1969-11-30
ES309167A2 (es) 1965-10-01
CH467787A (de) 1969-01-31
BE659443A (de) 1965-08-09
FR1455059A (fr) 1966-10-07
NL141781B (nl) 1974-04-16
SE307952B (de) 1969-01-27
BR6567054D0 (pt) 1973-08-14
NO118273B (de) 1969-12-08
NL6501632A (de) 1965-08-12
GB1052144A (de)
GB1051795A (de)
NO117367B (de) 1969-08-04
DE1545933A1 (de) 1969-12-18
BR6567053D0 (pt) 1973-12-26
GB1098242A (en) 1968-01-10
ES309169A1 (es) 1965-10-16
BE659442A (de) 1965-08-09
NL6501631A (de) 1965-08-12
DK118249B (da) 1970-07-27
BR6567055D0 (pt) 1973-08-02
BR6567051D0 (pt) 1973-08-14
FR4772M (de) 1967-01-23
ES309170A1 (es) 1965-07-16
FR4123M (de) 1966-04-25
NO119798B (de) 1970-07-06
SE307953B (de) 1969-01-27
FR4609M (de) 1966-11-21
NL6501579A (de) 1965-08-12
DE1545935A1 (de) 1969-12-11
CH460793A (de) 1968-08-15
DE1545934A1 (de) 1970-10-22
DE1545936A1 (de) 1969-12-18
NL6501578A (de) 1965-08-12
CH460030A (de) 1968-07-31
GB1077358A (en) 1967-07-26
ES309168A1 (es) 1965-10-01
US3299053A (en) 1967-01-17
IL22903A (en) 1969-03-27
FR1443116A (fr) 1966-06-24
SE321477B (de) 1970-03-09
DK105984C (da) 1966-12-05
FR4138M (de) 1966-05-02
DE1545936B2 (de) 1975-09-18
IL22869A (en) 1968-11-27
BE659444A (de) 1965-08-09

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