CH457457A - Verfahren zur Herstellung von Benzodiazepin-Derivaten - Google Patents

Verfahren zur Herstellung von Benzodiazepin-Derivaten

Info

Publication number
CH457457A
CH457457A CH420065A CH420065A CH457457A CH 457457 A CH457457 A CH 457457A CH 420065 A CH420065 A CH 420065A CH 420065 A CH420065 A CH 420065A CH 457457 A CH457457 A CH 457457A
Authority
CH
Switzerland
Prior art keywords
preparation
benzodiazepine derivatives
benzodiazepine
derivatives
Prior art date
Application number
CH420065A
Other languages
English (en)
Inventor
Focella Antonio
Israel Rachlin Albert
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of CH457457A publication Critical patent/CH457457A/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D243/00Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/141,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/161,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/181,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/24Oxygen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C233/00Carboxylic acid amides
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D243/00Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/141,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/161,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/181,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/24Oxygen atoms
    • C07D243/28Preparation including building-up the benzodiazepine skeleton from compounds containing no hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
CH420065A 1964-04-17 1965-03-25 Verfahren zur Herstellung von Benzodiazepin-Derivaten CH457457A (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US360755A US3335181A (en) 1964-04-17 1964-04-17 Ammonolysis of 2-halo-2'-benzoyl-4'-nitroacetanilides

Publications (1)

Publication Number Publication Date
CH457457A true CH457457A (de) 1968-06-15

Family

ID=23419290

Family Applications (1)

Application Number Title Priority Date Filing Date
CH420065A CH457457A (de) 1964-04-17 1965-03-25 Verfahren zur Herstellung von Benzodiazepin-Derivaten

Country Status (7)

Country Link
US (1) US3335181A (de)
BR (1) BR6568465D0 (de)
CH (1) CH457457A (de)
DE (1) DE1545941C3 (de)
DK (1) DK120346B (de)
GB (1) GB1097951A (de)
IL (1) IL23206A (de)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5706829A (en) * 1996-06-06 1998-01-13 Creighton University Method for treating neurocardiogenic syncope

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE75915C (de) * Dr. A. voswinkel, Apothekenbesitzer, in Berlin W., Kurfürsten-trafse 154 Verfahren zur Darstellung von Glycocollderivaten der Amidoacetophenone
BE513053A (de) * 1951-07-26
US3136815A (en) * 1959-12-10 1964-06-09 Hoffmann La Roche Amino substituted benzophenone oximes and derivatives thereof

Also Published As

Publication number Publication date
IL23206A (en) 1968-07-25
DK120346B (da) 1971-05-17
GB1097951A (en) 1968-01-03
BR6568465D0 (pt) 1973-08-28
US3335181A (en) 1967-08-08
DE1545941A1 (de) 1969-12-18
DE1545941C3 (de) 1975-11-20
DE1545941B2 (de) 1975-04-03

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