CH478812A - Verfahren zur Herstellung von Benzodiazepin-Derivaten - Google Patents

Verfahren zur Herstellung von Benzodiazepin-Derivaten

Info

Publication number
CH478812A
CH478812A CH1667266A CH1667266A CH478812A CH 478812 A CH478812 A CH 478812A CH 1667266 A CH1667266 A CH 1667266A CH 1667266 A CH1667266 A CH 1667266A CH 478812 A CH478812 A CH 478812A
Authority
CH
Switzerland
Prior art keywords
preparation
benzodiazepine derivatives
benzodiazepine
derivatives
Prior art date
Application number
CH1667266A
Other languages
English (en)
Inventor
Ian Fryer Rodney
Ernest Garcia Edward
Henryk Sternbach Leo
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of CH478812A publication Critical patent/CH478812A/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D243/00Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/141,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/161,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/181,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/24Oxygen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
CH1667266A 1965-12-09 1966-11-21 Verfahren zur Herstellung von Benzodiazepin-Derivaten CH478812A (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US512775A US3371083A (en) 1965-12-09 1965-12-09 Process for preparing therapeutically useful 3-substituted benzodiazepines

Publications (1)

Publication Number Publication Date
CH478812A true CH478812A (de) 1969-09-30

Family

ID=24040509

Family Applications (1)

Application Number Title Priority Date Filing Date
CH1667266A CH478812A (de) 1965-12-09 1966-11-21 Verfahren zur Herstellung von Benzodiazepin-Derivaten

Country Status (11)

Country Link
US (1) US3371083A (de)
BE (1) BE690313A (de)
BR (1) BR6685049D0 (de)
CH (1) CH478812A (de)
DE (1) DE1695169A1 (de)
DK (1) DK124823B (de)
ES (1) ES334299A1 (de)
FR (1) FR1503278A (de)
GB (1) GB1138888A (de)
NL (1) NL6617254A (de)
SE (1) SE338049B (de)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3427304A (en) * 1959-12-10 1969-02-11 Hoffmann La Roche Process for preparing 5-phenyl-3h-1,4-benzodiazepin-2(1h)-ones
US3414562A (en) * 1964-06-15 1968-12-03 Hoffmann La Roche Process for preparing 1, 3, 4, 5-tetrahydro-5-phenyl-2h-1, 4-benzodiazepin-2-ones
US3678043A (en) * 1966-03-14 1972-07-18 American Home Prod 2,3-dihydro-2-oxo-1h-1,4-benzodiazepine-3-carboxylic acid esters and related compounds
US3446800A (en) * 1968-02-09 1969-05-27 American Home Prod Process for the preparation of 1,3-dihydro-2h-1,4-benzodiazepin-2-ones
DE19639567C2 (de) * 1996-09-26 1998-11-26 Daimler Benz Ag Dachkonstruktion für einen offenen Personenkraftwagen

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3340253A (en) * 1962-11-28 1967-09-05 Hoffmann La Roche Preparation of certain benzodiazepine compounds

Also Published As

Publication number Publication date
DK124823B (da) 1972-11-27
SE338049B (de) 1971-08-30
US3371083A (en) 1968-02-27
FR1503278A (fr) 1967-11-24
BR6685049D0 (pt) 1973-12-26
BE690313A (de) 1967-05-29
NL6617254A (de) 1967-06-12
GB1138888A (en) 1969-01-01
DE1695169A1 (de) 1971-03-18
ES334299A1 (es) 1968-02-01

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Legal Events

Date Code Title Description
PL Patent ceased