ES2179798T3 - Procedimiento para la obtencion de compuestos heterociclicos. - Google Patents
Procedimiento para la obtencion de compuestos heterociclicos.Info
- Publication number
- ES2179798T3 ES2179798T3 ES00100235T ES00100235T ES2179798T3 ES 2179798 T3 ES2179798 T3 ES 2179798T3 ES 00100235 T ES00100235 T ES 00100235T ES 00100235 T ES00100235 T ES 00100235T ES 2179798 T3 ES2179798 T3 ES 2179798T3
- Authority
- ES
- Spain
- Prior art keywords
- group
- substituted
- compounds
- alkyl
- formula
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
- 150000001875 compounds Chemical class 0.000 title abstract 4
- 125000000217 alkyl group Chemical group 0.000 abstract 6
- LRHPLDYGYMQRHN-UHFFFAOYSA-N N-Butanol Chemical compound CCCCO LRHPLDYGYMQRHN-UHFFFAOYSA-N 0.000 abstract 2
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 2
- ZXEKIIBDNHEJCQ-UHFFFAOYSA-N isobutanol Chemical compound CC(C)CO ZXEKIIBDNHEJCQ-UHFFFAOYSA-N 0.000 abstract 2
- 229910052760 oxygen Inorganic materials 0.000 abstract 2
- 239000001301 oxygen Substances 0.000 abstract 2
- 229910052717 sulfur Inorganic materials 0.000 abstract 2
- XLYOFNOQVPJJNP-UHFFFAOYSA-N water Substances O XLYOFNOQVPJJNP-UHFFFAOYSA-N 0.000 abstract 2
- 125000003349 3-pyridyl group Chemical group N1=C([H])C([*])=C([H])C([H])=C1[H] 0.000 abstract 1
- 125000000339 4-pyridyl group Chemical group N1=C([H])C([H])=C([*])C([H])=C1[H] 0.000 abstract 1
- MYMOFIZGZYHOMD-UHFFFAOYSA-N Dioxygen Chemical compound O=O MYMOFIZGZYHOMD-UHFFFAOYSA-N 0.000 abstract 1
- LFQSCWFLJHTTHZ-UHFFFAOYSA-N Ethanol Chemical compound CCO LFQSCWFLJHTTHZ-UHFFFAOYSA-N 0.000 abstract 1
- AMQJEAYHLZJPGS-UHFFFAOYSA-N N-Pentanol Chemical compound CCCCCO AMQJEAYHLZJPGS-UHFFFAOYSA-N 0.000 abstract 1
- NINIDFKCEFEMDL-UHFFFAOYSA-N Sulfur Chemical compound [S] NINIDFKCEFEMDL-UHFFFAOYSA-N 0.000 abstract 1
- 229910052783 alkali metal Inorganic materials 0.000 abstract 1
- 150000001340 alkali metals Chemical class 0.000 abstract 1
- 125000003118 aryl group Chemical group 0.000 abstract 1
- QVGXLLKOCUKJST-UHFFFAOYSA-N atomic oxygen Chemical compound [O] QVGXLLKOCUKJST-UHFFFAOYSA-N 0.000 abstract 1
- 239000002585 base Substances 0.000 abstract 1
- 125000000816 ethylene group Chemical group [H]C([H])([*:1])C([H])([H])[*:2] 0.000 abstract 1
- 125000005843 halogen group Chemical group 0.000 abstract 1
- 125000005842 heteroatom Chemical group 0.000 abstract 1
- 125000000623 heterocyclic group Chemical group 0.000 abstract 1
- 125000004433 nitrogen atom Chemical group N* 0.000 abstract 1
- 239000011593 sulfur Substances 0.000 abstract 1
- 125000004434 sulfur atom Chemical group 0.000 abstract 1
- 125000003258 trimethylene group Chemical group [H]C([H])([*:2])C([H])([H])C([H])([H])[*:1] 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
- C07D207/34—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D207/36—Oxygen or sulfur atoms
- C07D207/40—2,5-Pyrrolidine-diones
- C07D207/416—2,5-Pyrrolidine-diones with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to other ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Pyridine Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Saccharide Compounds (AREA)
- Hydrogenated Pyridines (AREA)
Abstract
Procedimiento para la obtención de los compuestos de la fórmula (I) en la que R1 significa un átomo de hidrógeno o un grupo alquilo, A significa un grupo etileno, que puede estar substituido por alquilo, o significa un grupo trimetileno, que puede estar substituido por alquilo, X significa un átomo de oxígeno o de azufre o el grupo - CH-R3, donde R3 significa un átomo de hidrógeno o un grupo alquilo, y Z significa un grupo heterocíclico con 5 o 6 miembros, substituido en caso dado, que contiene al menos dos heteroátomos elegidos entre los átomos de oxígeno, de azufre y de nitrógeno, o significa un grupo 3- o 4-piridilo, substituido en caso dado, caracterizado porque se hacen reaccionar compuestos de la fórmula (II) en la que A y X tienen los significados anteriormente indicados, con compuestos de la fórmula (III) en la que R1 y Z tienen los significados anteriormente indicados y M1 significa un átomo de halógeno o el agrupamiento =OSO2-M2, donde M2 significa un grupo alquilo inferior, un grupo arilo o OM3, donde M3 significa un grupo alquilo inferior o un metal alcalino, en presencia de un alcohol no miscible con agua o solo parcialmente miscible con agua, elegido del grupo formado por iso-butanol, n-butanol o alcohol amílico y, en caso dado, en presencia de una base.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE19904310A DE19904310A1 (de) | 1999-01-28 | 1999-01-28 | Verfahren zur Herstellung heterocyclischer Verbindungen |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES2179798T3 true ES2179798T3 (es) | 2003-02-01 |
Family
ID=7896280
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES00100235T Expired - Lifetime ES2179798T3 (es) | 1999-01-28 | 2000-01-17 | Procedimiento para la obtencion de compuestos heterociclicos. |
Country Status (15)
| Country | Link |
|---|---|
| US (1) | US6211379B1 (es) |
| EP (1) | EP1024140B1 (es) |
| JP (1) | JP2000219688A (es) |
| KR (1) | KR100632521B1 (es) |
| CN (1) | CN1161354C (es) |
| AT (1) | ATE221530T1 (es) |
| BR (1) | BR0000184B1 (es) |
| CZ (1) | CZ297921B6 (es) |
| DE (2) | DE19904310A1 (es) |
| DK (1) | DK1024140T3 (es) |
| ES (1) | ES2179798T3 (es) |
| HK (1) | HK1031871A1 (es) |
| HU (1) | HU225245B1 (es) |
| IL (1) | IL134228A (es) |
| ZA (1) | ZA200000357B (es) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ATE364042T1 (de) * | 1999-06-23 | 2007-06-15 | Syngenta Participations Ag | Verfahren zur herstellung von thiamethoxam |
| SK285671B6 (sk) * | 2000-01-19 | 2007-06-07 | Bayer Aktiengesellschaft | Spôsob výroby heterocyklických zlúčenín |
| ES2556470T3 (es) * | 2011-09-02 | 2016-01-18 | Bayer Intellectual Property Gmbh | Procedimiento para preparar [3-[(6-cloro-3-piridinil)metil]-2-tiazolidiniliden]cianamida |
| WO2017211594A1 (de) | 2016-06-06 | 2017-12-14 | Bayer Cropscience Aktiengesellschaft | Verfahren zur herstellung heterocyclischer verbindungen |
| CN107629045A (zh) * | 2017-11-10 | 2018-01-26 | 上海生农生化制品股份有限公司 | 一种噻虫啉的水相合成方法 |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS5933283A (ja) * | 1982-08-19 | 1984-02-23 | Fujimoto Seiyaku Kk | イソチオウレア誘導体およびその製造法 |
| HU188852B (en) * | 1983-03-16 | 1986-05-28 | Richter Gedeon Vegyeszeti Gyar Rt,Hu | Process for producing thiazolidine derivatives active against gastric ulcer and intestinal ulcer |
| JPH0717621B2 (ja) * | 1986-03-07 | 1995-03-01 | 日本バイエルアグロケム株式会社 | 新規ヘテロ環式化合物 |
| JPH07121909B2 (ja) * | 1986-09-10 | 1995-12-25 | 日本バイエルアグロケム株式会社 | 新規複素環式化合物及び殺虫剤 |
-
1999
- 1999-01-28 DE DE19904310A patent/DE19904310A1/de not_active Withdrawn
-
2000
- 2000-01-17 ES ES00100235T patent/ES2179798T3/es not_active Expired - Lifetime
- 2000-01-17 AT AT00100235T patent/ATE221530T1/de active
- 2000-01-17 DK DK00100235T patent/DK1024140T3/da active
- 2000-01-17 DE DE50000320T patent/DE50000320D1/de not_active Expired - Lifetime
- 2000-01-17 EP EP00100235A patent/EP1024140B1/de not_active Expired - Lifetime
- 2000-01-18 JP JP2000009059A patent/JP2000219688A/ja active Pending
- 2000-01-20 KR KR1020000002597A patent/KR100632521B1/ko active IP Right Grant
- 2000-01-20 US US09/488,436 patent/US6211379B1/en not_active Expired - Lifetime
- 2000-01-26 IL IL13422800A patent/IL134228A/en not_active IP Right Cessation
- 2000-01-27 BR BRPI0000184-8A patent/BR0000184B1/pt not_active IP Right Cessation
- 2000-01-27 ZA ZA200000357A patent/ZA200000357B/xx unknown
- 2000-01-27 CZ CZ20000322A patent/CZ297921B6/cs not_active IP Right Cessation
- 2000-01-28 HU HU0000366A patent/HU225245B1/hu not_active IP Right Cessation
- 2000-01-28 CN CNB001045075A patent/CN1161354C/zh not_active Expired - Lifetime
-
2001
- 2001-03-30 HK HK01102337A patent/HK1031871A1/xx not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| BR0000184A (pt) | 2000-09-05 |
| DE19904310A1 (de) | 2000-08-03 |
| HUP0000366A2 (hu) | 2000-12-28 |
| EP1024140B1 (de) | 2002-07-31 |
| DE50000320D1 (de) | 2002-09-05 |
| BR0000184B1 (pt) | 2010-10-19 |
| US6211379B1 (en) | 2001-04-03 |
| CZ2000322A3 (cs) | 2000-09-13 |
| IL134228A (en) | 2002-11-10 |
| HK1031871A1 (en) | 2001-06-29 |
| EP1024140A1 (de) | 2000-08-02 |
| ATE221530T1 (de) | 2002-08-15 |
| KR100632521B1 (ko) | 2006-10-09 |
| CN1161354C (zh) | 2004-08-11 |
| DK1024140T3 (da) | 2002-11-04 |
| HU225245B1 (en) | 2006-08-28 |
| KR20010006582A (ko) | 2001-01-26 |
| JP2000219688A (ja) | 2000-08-08 |
| IL134228A0 (en) | 2001-04-30 |
| ZA200000357B (en) | 2000-08-15 |
| CZ297921B6 (cs) | 2007-05-02 |
| HUP0000366A3 (en) | 2001-12-28 |
| CN1269363A (zh) | 2000-10-11 |
| HU0000366D0 (en) | 2000-04-28 |
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