ES2059212T3 - Antagonistas paf/h1 imidazopiridina. - Google Patents

Antagonistas paf/h1 imidazopiridina.

Info

Publication number
ES2059212T3
ES2059212T3 ES92902889T ES92902889T ES2059212T3 ES 2059212 T3 ES2059212 T3 ES 2059212T3 ES 92902889 T ES92902889 T ES 92902889T ES 92902889 T ES92902889 T ES 92902889T ES 2059212 T3 ES2059212 T3 ES 2059212T3
Authority
ES
Spain
Prior art keywords
imidazopyridine
paf
antagonists
ring
condensed
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES92902889T
Other languages
English (en)
Spanish (es)
Inventor
David Alker
Robert John Bass
Kelvin Cooper
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Corp Belgium
Pfizer Corp SRL
Original Assignee
Pfizer Corp Belgium
Pfizer Corp SRL
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Corp Belgium, Pfizer Corp SRL filed Critical Pfizer Corp Belgium
Application granted granted Critical
Publication of ES2059212T3 publication Critical patent/ES2059212T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Dermatology (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Cosmetics (AREA)
  • Prostheses (AREA)
  • Steroid Compounds (AREA)
ES92902889T 1991-02-13 1992-01-24 Antagonistas paf/h1 imidazopiridina. Expired - Lifetime ES2059212T3 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB919102997A GB9102997D0 (en) 1991-02-13 1991-02-13 Therapeutic agents

Publications (1)

Publication Number Publication Date
ES2059212T3 true ES2059212T3 (es) 1994-11-01

Family

ID=10689943

Family Applications (1)

Application Number Title Priority Date Filing Date
ES92902889T Expired - Lifetime ES2059212T3 (es) 1991-02-13 1992-01-24 Antagonistas paf/h1 imidazopiridina.

Country Status (29)

Country Link
US (1) US5358953A (Sortimente)
EP (1) EP0572425B1 (Sortimente)
JP (1) JP2506541B2 (Sortimente)
KR (1) KR970005302B1 (Sortimente)
CN (1) CN1040326C (Sortimente)
AT (1) ATE109482T1 (Sortimente)
AU (1) AU650322B2 (Sortimente)
BR (1) BR9205615A (Sortimente)
CA (1) CA2099381C (Sortimente)
CZ (1) CZ280504B6 (Sortimente)
DE (1) DE69200304T2 (Sortimente)
DK (1) DK0572425T3 (Sortimente)
EG (1) EG20085A (Sortimente)
ES (1) ES2059212T3 (Sortimente)
FI (1) FI933531L (Sortimente)
GB (1) GB9102997D0 (Sortimente)
HU (2) HUT65947A (Sortimente)
IE (1) IE65125B1 (Sortimente)
IL (1) IL100887A (Sortimente)
MX (1) MX9200589A (Sortimente)
MY (1) MY108437A (Sortimente)
NO (1) NO300592B1 (Sortimente)
NZ (1) NZ241597A (Sortimente)
PL (1) PL169304B1 (Sortimente)
RU (1) RU2114845C1 (Sortimente)
TW (1) TW227000B (Sortimente)
WO (1) WO1992014734A1 (Sortimente)
YU (1) YU48238B (Sortimente)
ZA (1) ZA921005B (Sortimente)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2042421B1 (es) * 1992-05-22 1994-08-01 Uriach & Cia Sa J Procedimiento para la obtencion de la 8-cloro-11-*1-*(5-metil-3-piridil)metil*-4-piperidiliden*-6,11-dihidro-5h-benzo*5,6*ciclohepta*1,2-b*piridina.
AU3186395A (en) * 1994-08-10 1996-03-07 British Biotech Pharmaceuticals Limited Imidazopyridine derivatives as dual histamine (h1) and platelet activating factor (paf) antagonists
ES2087038B1 (es) * 1994-11-07 1997-03-16 Uriach & Cia Sa J Nuevas piperidinas con actividad antagonista del paf.
US5567711A (en) * 1995-04-19 1996-10-22 Abbott Laboratories Indole-3-carbonyl and indole-3-sulfonyl derivatives as platelet activating factor antagonists
GB9508748D0 (en) * 1995-04-28 1995-06-14 British Biotech Pharm Benzimidazole derivatives
SK12798A3 (en) * 1995-08-05 1998-08-05 British Biotech Pharm Imidazopyridine derivatives, method for producing thereof, pharmaceutical composition containing same and their use
SE9801526D0 (sv) * 1998-04-29 1998-04-29 Astra Ab New compounds
CA2774959C (en) 2000-08-04 2016-05-31 Dmi Biosciences, Inc. Method of using diketopiperazines and composition containing them
EP2517722B1 (en) 2003-05-15 2016-03-02 Ampio Pharmaceuticals, Inc. Synthesis of diketopiperazines
US7687515B2 (en) * 2006-01-17 2010-03-30 N.V. Organon 6-phenyl-1H-imidazo[4,5-c]pyridine-4-carbonitrile derivatives
RU2475485C2 (ru) 2008-01-30 2013-02-20 Ниппон Дзоки Фармасьютикал Ко., Лтд. Производное пиперидина
JP5856843B2 (ja) 2008-05-27 2016-02-10 アンピオ ファーマシューティカルズ，インコーポレイテッド ジケトピペラジンを用いた医薬組成物
JP5978296B2 (ja) * 2011-06-28 2016-08-24 フジアン・ミンドン・レジュヴネイション・ファーマスーティカル・カンパニー・リミテッド 抗アレルギ性ベンゾシクロヘプタチオフェン誘導体
EA028343B1 (ru) 2011-10-10 2017-11-30 Ампио Фармасьютикалз, Инк. Лечение дегенеративного заболевания сустава
PH12014500686A1 (en) 2011-10-10 2020-12-18 Ampio Pharmaceuticals Inc Implantable medical devices with increased immune tolerance, and methods for making and implanting
MX355446B (es) * 2011-10-28 2018-04-18 Ampio Pharmaceuticals Inc Tratamiento de rinitis.
US9808454B2 (en) 2013-03-15 2017-11-07 Ampio Pharmaceuticals, Inc. Compositions for the mobilization, homing, expansion and differentiation of stem cells and methods of using the same
EP3183240A4 (en) 2014-08-18 2018-06-27 Ampio Pharmaceuticals, Inc. Treatment of joint conditions
EP3310375A4 (en) 2015-06-22 2019-02-20 Ampio Pharmaceuticals, Inc. USE OF LOW-MOLECULAR FRACTIONS OF HUMAN SERUMALBUMINE IN THE TREATMENT OF ILLNESSES
CN113880801A (zh) * 2020-07-03 2022-01-04 合肥医工医药股份有限公司 一类三环化合物、其制备方法及其医药用途

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL132137C (Sortimente) * 1963-04-24
EP0404797B1 (en) * 1988-03-15 1995-02-01 G.D. Searle & Co. 1H/3H-[4-(N,N-CYCLOALKYL AND/OR BRANCHED-ALKYLCARBOXAMIDO) -BENZYL]IMIDAZO[4,5-c]PYRIDINES AS PAF ANTAGONISTS
NZ228889A (en) * 1988-04-28 1991-09-25 Schering Corp Fused tri- or tetracyclic heterocyclic compounds and pharmaceutical compositions
US5250681A (en) * 1988-06-02 1993-10-05 Ajinomoto Co., Inc. Piperidine derivatives and hypotensives containing the same
US5114919A (en) * 1990-02-26 1992-05-19 Merck & Co., Inc. Adjuncts in cancer chemotherapy
ES2061247T3 (es) * 1990-05-09 1994-12-01 Pfizer Imidazo (4,5-c) piridinas con actividad antagonista del paf.

Also Published As

Publication number Publication date
IE920449A1 (en) 1992-08-12
MX9200589A (es) 1992-10-01
FI933531A7 (fi) 1993-08-10
MY108437A (en) 1996-09-30
HU211202A9 (en) 1995-11-28
DE69200304D1 (de) 1994-09-08
BR9205615A (pt) 1994-05-17
CN1064275A (zh) 1992-09-09
EG20085A (en) 1997-05-31
WO1992014734A1 (en) 1992-09-03
CZ280504B6 (cs) 1996-02-14
EP0572425A1 (en) 1993-12-08
YU14392A (sh) 1994-11-15
CN1040326C (zh) 1998-10-21
HU9302327D0 (en) 1993-10-28
EP0572425B1 (en) 1994-08-03
CA2099381A1 (en) 1992-08-14
NO300592B1 (no) 1997-06-23
DE69200304T2 (de) 1994-12-08
NO932889L (no) 1993-08-13
CS42592A3 (en) 1992-09-16
PL169304B1 (pl) 1996-06-28
JPH06504992A (ja) 1994-06-09
ZA921005B (en) 1993-08-12
FI933531A0 (fi) 1993-08-10
AU650322B2 (en) 1994-06-16
IL100887A (en) 1996-01-19
YU48238B (sh) 1997-08-22
HUT65947A (en) 1994-08-29
TW227000B (Sortimente) 1994-07-21
US5358953A (en) 1994-10-25
JP2506541B2 (ja) 1996-06-12
IL100887A0 (en) 1992-11-15
CA2099381C (en) 1996-07-09
KR970005302B1 (ko) 1997-04-15
IE65125B1 (en) 1995-10-04
NZ241597A (en) 1993-04-28
DK0572425T3 (da) 1994-09-12
AU1168392A (en) 1992-09-15
RU2114845C1 (ru) 1998-07-10
NO932889D0 (no) 1993-08-13
GB9102997D0 (en) 1991-03-27
FI933531L (fi) 1993-08-10
ATE109482T1 (de) 1994-08-15

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