ES2052296T3 - Derivados de tieno(2,3-d)pirimidina. - Google Patents

Derivados de tieno(2,3-d)pirimidina.

Info

Publication number
ES2052296T3
ES2052296T3 ES91103547T ES91103547T ES2052296T3 ES 2052296 T3 ES2052296 T3 ES 2052296T3 ES 91103547 T ES91103547 T ES 91103547T ES 91103547 T ES91103547 T ES 91103547T ES 2052296 T3 ES2052296 T3 ES 2052296T3
Authority
ES
Spain
Prior art keywords
sub
rest
elevated
mean
hydroxy
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES91103547T
Other languages
English (en)
Inventor
Matthias Dr Wiesenfeldt
Karl-Heinz Dr Etzbach
Peter Dr Hofmeister
Christoph Dr Kuenast
Karl-Otto Dr Westphalen
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
BASF SE
Original Assignee
BASF SE
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by BASF SE filed Critical BASF SE
Application granted granted Critical
Publication of ES2052296T3 publication Critical patent/ES2052296T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Plant Pathology (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

Abstract

TIENO [2,3-D] DERIVADOS DE PIRIMIDINA DE LA FORMULA GENERAL I EN LA QUE LOS SUSTITUYENTES TIENEN EL SIGUIENTE SIGNIFICADO; R ELEVADO 1 HIDROGENO, C SUB 1-C SUB 5 ALQUILO, C SUB 1-C SUB 3 CLOROALQUILO, C SUB 3-C SUB 6 CICLOALQUILO, FENILO O BENCILO R (AL CUADRADO) FLUOR, CLORO, BROMO, YODO, HIDROXY, ACIDO, CIANO, TIOCIANATO, MERCAPTO, UN RESTO ORGANICO NO UNIDO SOBRE NITROGENO O UN RESTO NR ELEVADO 5 R ELEVADO 6, DEL QUE R ELEVADO 5 Y R ELEVADO 6 SIGNIFICAN HIDROGENO, AMINO O RESTO ORGANICO INDEPENDIENTES ENTRE ELLOS O CONJUNTAMENTE CON EL ATOMO DE NITROGENO FORMAN UN RESTO HETEROCICLICO CON 3 HASTA 8 CICLOATOMOS, CON LA RESERVA, DE QUE R (AL CUADRADO) NO SIGNIFICA FENOXI-C SUB 2-C SUB 3 ALQUILAMINO, R ELEVADO 3 CLORO, BROMO, HIDROXY O MERCAPTO, CON LA RESERVA, DE QUE R (AL CUADRADO) HIDROXI Y R ELEVADO 3 NO SIGNIFICAN BROMO SIMULTANEAMENTE Y DE QUE NO SIGNIFICA SIMULTANEAMENTE R ELEVADO 3 HIDROXI Y R ELEVADO 4 ALCOXICARBONILO O CARBOXY R ELEVADO 4 HIDROGENO, C SUB 1-C SUB 6 ALQUILO, C SUB 3-C SUB 6 MONO-, DI-, O TRIHALOGENURO DE ALQUILO, FENILO CIANO, FORMILO, HIDROXIIMINOMETILO, CARBOXY, ALCOXICARBONILO, AMINOCARBONILO O UN RESTO DE LA FORMULA CH=X POR LA CUAL X SOBRE RESTO UNIDO DE NITROGENO DE UN AMINO PRIMARIO O SOBRE EL RESTO UNIDO DE CARBONO ES UNA COMBINACION METILOACTIVA, ASI COMO LOS TAUTOMEROS DE ESTE TIENO[2,3-D] DERIVADOS DE PIRAMIDINA Y LAS SALES TOLERADAS DE PLANTAS UTILES DE ESTE DERIVADO Y SUS TAUTOMEROS. LAS COMBINACIONES I ENCUENTRAN UTILIZACION COMO INSECTICIDAS, REGULADORES DE CRECIMIENTO, Y HERBICIDAS
ES91103547T 1990-03-19 1991-03-08 Derivados de tieno(2,3-d)pirimidina. Expired - Lifetime ES2052296T3 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19904008726 DE4008726A1 (de) 1990-03-19 1990-03-19 Thieno(2,3-d)pyrimidinderivate

Publications (1)

Publication Number Publication Date
ES2052296T3 true ES2052296T3 (es) 1994-07-01

Family

ID=6402524

Family Applications (1)

Application Number Title Priority Date Filing Date
ES91103547T Expired - Lifetime ES2052296T3 (es) 1990-03-19 1991-03-08 Derivados de tieno(2,3-d)pirimidina.

Country Status (6)

Country Link
EP (1) EP0447891B1 (es)
JP (1) JPH04217685A (es)
CA (1) CA2038521A1 (es)
DE (2) DE4008726A1 (es)
DK (1) DK0447891T3 (es)
ES (1) ES2052296T3 (es)

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US6503914B1 (en) * 2000-10-23 2003-01-07 Board Of Regents, The University Of Texas System Thienopyrimidine-based inhibitors of the Src family
US7427623B2 (en) 2001-09-11 2008-09-23 Smithkline Beecham Corporation 4-Amino-2,3-disubstituted thieno[2,3-d]pyrimidines and pharmacetical compositions thereof
WO2004013141A1 (en) 2002-08-06 2004-02-12 Astrazeneca Ab Condensed pyridines and pyrimidines with tie2 (tek) activity
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TW200410975A (en) * 2002-09-26 2004-07-01 Nihon Nohyaku Co Ltd New pesticide and method for using it, new substituted thienopyrimidine derivative, its intermediate, and method for producing it
ES2217956B1 (es) * 2003-01-23 2006-04-01 Almirall Prodesfarma, S.A. Nuevos derivados de 4-aminotieno(2,3-d)pirimidin-6-carbonitrilo.
ATE511511T1 (de) * 2003-03-31 2011-06-15 Trovis Pharmaceuticals Llc Neue piperidinylaminothienoä2,3-dü pyrimidinverbindungen
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US7419978B2 (en) 2003-10-22 2008-09-02 Bristol-Myers Squibb Company Phenyl-aniline substituted bicyclic compounds useful as kinase inhibitors
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JP5243960B2 (ja) 2005-10-21 2013-07-24 ダウ アグロサイエンシィズ エルエルシー 殺菌活性を有するチエノ−ピリミジン化合物
US7531482B2 (en) 2005-10-21 2009-05-12 Dow Agrosciences Llc Thieno-pyrimidine compounds having fungicidal activity
TWI417095B (zh) 2006-03-15 2013-12-01 Janssen Pharmaceuticals Inc １，４-二取代之３-氰基-吡啶酮衍生物及其作為ｍＧｌｕＲ２-受體之正向異位性調節劑之用途
CN101466716A (zh) 2006-04-07 2009-06-24 德维洛根股份公司 用于药物组合物的具有mnkl/mnk2抑制活性的噻吩并嘧啶
EA200802248A1 (ru) 2006-05-22 2009-06-30 Басф Се Способы применения соединений 4-амино-5-хлортиено[2,3-d]-пиримидина в качестве инсектицидов
EP1889847A1 (en) 2006-07-10 2008-02-20 DeveloGen Aktiengesellschaft Pyrrolopyrimidines for pharmaceutical compositions
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US9133209B2 (en) 2009-07-30 2015-09-15 Merial, Inc. Insecticidal 4-amino-thieno[2,3-D]-pyrimidine compounds and methods of their use
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TW201219401A (en) 2010-09-14 2012-05-16 Lexicon Pharmaceuticals Inc Bicyclic inhibitors of Notum Pectinacetylesterase and methods of their use
JP5852665B2 (ja) 2010-11-08 2016-02-03 ジヤンセン・フアーマシユーチカルズ・インコーポレーテツド １，２，４−トリアゾロ［４，３−ａ］ピリジン誘導体およびｍＧｌｕＲ２受容体のポジティブアロステリックモジュレーターとしてのそれらの使用
JP5852666B2 (ja) 2010-11-08 2016-02-03 ジヤンセン・フアーマシユーチカルズ・インコーポレーテツド １，２，４−トリアゾロ［４，３−ａ］ピリジン誘導体およびｍＧｌｕＲ２受容体のポジティブアロステリックモジュレーターとしてのそれらの使用
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JO3367B1 (ar) 2013-09-06 2019-03-13 Janssen Pharmaceutica Nv مركبات 2،1، 4- ثلاثي زولو [3،4-a] بيريدين واستخدامها بصفة منظمات تفارغية موجبة لمستقبلات ميجلور 2
FR3015483B1 (fr) * 2013-12-23 2016-01-01 Servier Lab Nouveaux derives de thienopyrimidine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
KR20200036063A (ko) 2014-01-21 2020-04-06 얀센 파마슈티카 엔.브이. 대사 조절형 글루탐산 작동성 수용체 제2아형의 양성 알로스테릭 조절제 또는 오르토스테릭 작동제를 포함하는 조합 및 그 용도
KR20220038826A (ko) 2014-01-21 2022-03-29 얀센 파마슈티카 엔.브이. 대사 조절형 글루탐산 작동성 수용체 제2아형의 양성 알로스테릭 조절제 또는 오르토스테릭 작동제를 포함하는 조합 및 그 용도
KR20180075228A (ko) * 2016-12-26 2018-07-04 한미약품 주식회사 싸이에노피리미딘 화합물의 신규 제조방법 및 중간체
RU2746282C1 (ru) * 2020-07-30 2021-04-12 Федеральное государственное бюджетное образовательное учреждение высшего образования "Кубанский государственный университет" (ФГБОУ ВО "КубГУ") Способ повышения урожайности озимой пшеницы

Family Cites Families (2)

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GB1570494A (en) * 1975-11-28 1980-07-02 Ici Ltd Thienopyrimidine derivatives and their use as pesticides
ZA782648B (en) * 1977-05-23 1979-06-27 Ici Australia Ltd The prevention,control or eradication of infestations of ixodid ticks

Also Published As

Publication number Publication date
EP0447891B1 (de) 1994-04-27
CA2038521A1 (en) 1991-09-20
EP0447891A1 (de) 1991-09-25
JPH04217685A (ja) 1992-08-07
DK0447891T3 (da) 1994-05-30
DE59101477D1 (de) 1994-06-01
DE4008726A1 (de) 1991-09-26

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