ES2018667B3 - Derivados del acido 4-qionolon-3-carboxilico, procedimiento para su obtencion y preparados farmaceuticos que los contienen. - Google Patents

Derivados del acido 4-qionolon-3-carboxilico, procedimiento para su obtencion y preparados farmaceuticos que los contienen.

Info

Publication number
ES2018667B3
ES2018667B3 ES87109461T ES87109461T ES2018667B3 ES 2018667 B3 ES2018667 B3 ES 2018667B3 ES 87109461 T ES87109461 T ES 87109461T ES 87109461 T ES87109461 T ES 87109461T ES 2018667 B3 ES2018667 B3 ES 2018667B3
Authority
ES
Spain
Prior art keywords
qionolon
carboxilico
derivatives
procedure
obtaining
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES87109461T
Other languages
English (en)
Inventor
Fritz Sauter
Ulrich Jordis
Manfred Rudolf
Josef Wieser
Karl Baumann
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Chemie Linz GmbH
Original Assignee
Chemie Linz GmbH
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Chemie Linz GmbH filed Critical Chemie Linz GmbH
Application granted granted Critical
Publication of ES2018667B3 publication Critical patent/ES2018667B3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/80—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
    • C07D211/84—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen directly attached to ring carbon atoms
    • C07D211/86—Oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/08—Bridged systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyridine Compounds (AREA)
ES87109461T 1986-07-04 1987-07-01 Derivados del acido 4-qionolon-3-carboxilico, procedimiento para su obtencion y preparados farmaceuticos que los contienen. Expired - Lifetime ES2018667B3 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE3622509 1986-07-04

Publications (1)

Publication Number Publication Date
ES2018667B3 true ES2018667B3 (es) 1991-05-01

Family

ID=6304401

Family Applications (1)

Application Number Title Priority Date Filing Date
ES87109461T Expired - Lifetime ES2018667B3 (es) 1986-07-04 1987-07-01 Derivados del acido 4-qionolon-3-carboxilico, procedimiento para su obtencion y preparados farmaceuticos que los contienen.

Country Status (24)

Country Link
US (1) US5045549A (es)
EP (1) EP0251308B1 (es)
JP (1) JPH07103123B2 (es)
KR (1) KR880001595A (es)
AR (1) AR245450A1 (es)
AT (1) ATE58538T1 (es)
AU (1) AU608515B2 (es)
CS (1) CS277415B6 (es)
DD (1) DD262428A1 (es)
DE (1) DE3766299D1 (es)
DK (1) DK342187A (es)
ES (1) ES2018667B3 (es)
FI (1) FI88506C (es)
GR (1) GR3001097T3 (es)
HU (1) HU197907B (es)
IL (1) IL83049A (es)
MY (1) MY101261A (es)
NO (1) NO166130C (es)
NZ (1) NZ220950A (es)
PH (1) PH24239A (es)
PT (1) PT85257B (es)
SU (1) SU1551248A3 (es)
YU (1) YU45039B (es)
ZA (1) ZA874849B (es)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IN166416B (es) * 1985-09-18 1990-05-05 Pfizer
SI8810667A8 (en) * 1987-04-08 1996-04-30 Chinoin Gyogyszer Es Vegyeszet Anhydride of quinoline carboxylic acid of boron acid and process for their production.
JPH02131453A (ja) * 1988-04-15 1990-05-21 Asahi Glass Co Ltd ２―クロロ―４，５―ジフルオロベンゾイルアクリル酸誘導体
JPH072679B2 (ja) * 1988-04-15 1995-01-18 旭硝子株式会社 ２―クロロ―４，５―ジフルオロ安息香酸誘導体
WO1989012055A1 (en) * 1988-06-08 1989-12-14 Kyorin Pharmaceutical Co., Ltd. Antitumor agent
JPH02298946A (ja) * 1989-05-15 1990-12-11 Johoku Seihan Center:Kk 製版・版下作製材および製版・版下作製における貼付方法
EP0449445A3 (en) * 1990-03-27 1993-08-25 Pfizer Inc. Preparation of beta-ketoesters useful in preparing quinolone antibiotics
DE69132256T2 (de) 1990-04-18 2001-01-25 Procter & Gamble Pharma Antimikrobielle chinolonyl-lactame
FR2692577B1 (fr) * 1992-05-26 1996-02-02 Bouchara Sa Nouvelles quinolones fluorees, leur procede de preparation et les compositions pharmaceutiques en renfermant.
TW252107B (es) * 1993-08-27 1995-07-21 Hokuriku Pharmacetical Co Ltd
ES2092963B1 (es) * 1995-04-12 1997-12-16 Sint Quimica Sa Procedimiento para la preparacion del acido 1-ciclopropil-6-fluoro-1, 4-dihidro-7-(1s,4s)-5-metil-2,5-diazabiciclo(2.2.1) hept-2-il)-4-oxo-3-quinolincarboxilico y sus sales.
SE0003795D0 (sv) 2000-10-20 2000-10-20 Astrazeneca Ab Pharmaceutically useful compounds
WO2011031745A1 (en) 2009-09-09 2011-03-17 Achaogen, Inc. Antibacterial fluoroquinolone analogs

Family Cites Families (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4292317A (en) * 1977-09-20 1981-09-29 Laboratorie Roger Bellon 1,4-Dihydro-quinoline-3-carboxylic acid derivatives, process for their preparation and compositions containing them
DE2808070A1 (de) * 1978-02-24 1979-08-30 Bayer Ag Verfahren zur herstellung von 4-pyridon-3-carbonsaeuren und/oder deren derivaten
DE3267485D1 (en) * 1981-02-18 1986-01-02 Nippon Shinyaku Co Ltd Substituted carboxylic acid derivatives
US4499091A (en) * 1982-03-31 1985-02-12 Sterling Drug Inc. 1-Amino (or substituted amino)-1,4-dihydro-4-oxo-6-fluoro-7-heterylquinoline-3-carboxylic acids and their use as antibacterial agents
DE3363711D1 (en) * 1982-03-31 1986-07-03 Sterling Drug Inc New quinolone compounds and preparation thereof
NZ208470A (en) * 1983-07-18 1988-06-30 Abbott Lab 6-fluoro-1,4-dihydro-4-oxo-quinoline-3-carboxylic acid derivatives and antibacterial compositions containing such
US4730000A (en) * 1984-04-09 1988-03-08 Abbott Laboratories Quinoline antibacterial compounds
JPS6056959A (ja) * 1983-07-18 1985-04-02 アボツト　ラボラトリ−ズ キノリン抗菌性化合物
US4571396A (en) * 1984-04-16 1986-02-18 Warner-Lambert Company Antibacterial agents
EP0181521A1 (en) * 1984-10-19 1986-05-21 Otsuka Pharmaceutical Co., Ltd. Antimicrobial 1-substituted Phenyl-4-oxoquinoline-3-carboxylic acid compounds
US4578473A (en) * 1985-04-15 1986-03-25 Warner-Lambert Company Process for quinoline-3-carboxylic acid antibacterial agents
IN166416B (es) * 1985-09-18 1990-05-05 Pfizer
DE3601567A1 (de) * 1986-01-21 1987-07-23 Bayer Ag 7-(azabicycloalkyl)-chinoloncarbonsaeure- und -naphthyridon-carbonsaeure-derivate
US4962108A (en) * 1987-07-31 1990-10-09 Warner-Lambert Company Antibacterial quinoline compounds
US4923879A (en) * 1987-07-31 1990-05-08 Warner-Lambert Company 1,8-Naphthyridines and their use as antibacterial agents
US4962112A (en) * 1987-08-04 1990-10-09 Abbott Laboratories 7-(2-methyl-4-aminopyrrolidinyl)naphthryidine and quinoline compounds
US4780468A (en) * 1987-08-07 1988-10-25 Warner-Lambert Company 8-trifluoromethyl quinolones as antibacterial agents
US4851418A (en) * 1987-08-21 1989-07-25 Warner-Lambert Company Naphthyridine antibacterial agents containing an α-amino acid in the side chain of the 7-substituent
WO1989005643A1 (en) * 1987-12-18 1989-06-29 Pfizer Inc. Heterocyclic-substituted quinoline-carboxylic acids
US4920120A (en) * 1988-01-25 1990-04-24 Warner-Lambert Company Antibacterial agents

Also Published As

Publication number Publication date
YU45039B (en) 1991-06-30
FI88506C (fi) 1993-05-25
EP0251308B1 (de) 1990-11-22
YU124687A (en) 1988-12-31
AR245450A1 (es) 1994-01-31
HU197907B (en) 1989-06-28
GR3001097T3 (en) 1992-04-17
DE3766299D1 (de) 1991-01-03
IL83049A0 (en) 1987-12-31
PT85257A (en) 1987-08-01
EP0251308A1 (de) 1988-01-07
NO872778D0 (no) 1987-07-02
JPH07103123B2 (ja) 1995-11-08
FI872897A (fi) 1988-01-05
JPS6322580A (ja) 1988-01-30
AU7508087A (en) 1988-01-07
DK342187A (da) 1988-01-05
ZA874849B (en) 1988-03-30
AU608515B2 (en) 1991-04-11
CS277415B6 (en) 1993-03-17
NO166130C (no) 1991-06-05
NO166130B (no) 1991-02-25
FI88506B (fi) 1993-02-15
FI872897A0 (fi) 1987-07-01
HUT45060A (en) 1988-05-30
CS505587A3 (en) 1992-08-12
DK342187D0 (da) 1987-07-03
DD262428A1 (de) 1988-11-30
NZ220950A (en) 1990-07-26
US5045549A (en) 1991-09-03
SU1551248A3 (ru) 1990-03-15
MY101261A (en) 1991-08-17
ATE58538T1 (de) 1990-12-15
KR880001595A (ko) 1988-04-25
NO872778L (no) 1988-01-05
IL83049A (en) 1991-12-12
PH24239A (en) 1990-05-04
PT85257B (pt) 1990-03-30

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