NO155226C - Fremgangsmaate for fremstilling av farmasoeytiske preparater inneholdende benzodiazepiner, dibenzotiepiner eller quinolinmetanolderivater. - Google Patents

Fremgangsmaate for fremstilling av farmasoeytiske preparater inneholdende benzodiazepiner, dibenzotiepiner eller quinolinmetanolderivater.

Info

Publication number
NO155226C
NO155226C NO801863A NO801863A NO155226C NO 155226 C NO155226 C NO 155226C NO 801863 A NO801863 A NO 801863A NO 801863 A NO801863 A NO 801863A NO 155226 C NO155226 C NO 155226C
Authority
NO
Norway
Prior art keywords
quinolinmetanol
dibenzotiepines
derivatives
procedure
preparation
Prior art date
Application number
NO801863A
Other languages
English (en)
Other versions
NO801863L (no
NO155226B (no
Inventor
Juerg Schrank
Hans Steffen
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of NO801863L publication Critical patent/NO801863L/no
Publication of NO155226B publication Critical patent/NO155226B/no
Publication of NO155226C publication Critical patent/NO155226C/no

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/10—Dispersions; Emulsions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/10—Dispersions; Emulsions
    • A61K9/127—Liposomes
    • A61K9/1277—Processes for preparing; Proliposomes
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Dispersion Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
NO801863A 1979-06-22 1980-06-20 Fremgangsmaate for fremstilling av farmasoeytiske preparater inneholdende benzodiazepiner, dibenzotiepiner eller quinolinmetanolderivater. NO155226C (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH586379 1979-06-22

Publications (3)

Publication Number Publication Date
NO801863L NO801863L (no) 1980-12-22
NO155226B NO155226B (no) 1986-11-24
NO155226C true NO155226C (no) 1987-03-04

Family

ID=4300559

Family Applications (1)

Application Number Title Priority Date Filing Date
NO801863A NO155226C (no) 1979-06-22 1980-06-20 Fremgangsmaate for fremstilling av farmasoeytiske preparater inneholdende benzodiazepiner, dibenzotiepiner eller quinolinmetanolderivater.

Country Status (21)

Country Link
US (1) US4411894A (no)
EP (1) EP0021337B1 (no)
JP (1) JPS567714A (no)
KR (1) KR850001301B1 (no)
AR (1) AR230178A1 (no)
AT (1) ATE5508T1 (no)
AU (1) AU534959B2 (no)
CA (1) CA1173360A (no)
DE (1) DE3065818D1 (no)
DK (1) DK155172C (no)
ES (1) ES8104720A1 (no)
FI (1) FI72875C (no)
HU (1) HU186296B (no)
IE (1) IE49615B1 (no)
IL (1) IL60326A (no)
MC (1) MC1336A1 (no)
NO (1) NO155226C (no)
NZ (1) NZ194047A (no)
PH (1) PH16795A (no)
PT (1) PT71436B (no)
ZA (1) ZA803567B (no)

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CA1264162A (en) * 1984-03-15 1990-01-02 Manfred Breuninger Glycerol ether phosphatides
JPS60208910A (ja) * 1984-03-31 1985-10-21 Green Cross Corp:The 水難溶性薬物・リン脂質複合体の製造方法
US4891208A (en) * 1985-04-10 1990-01-02 The Liposome Company, Inc. Steroidal liposomes
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US4880635B1 (en) * 1984-08-08 1996-07-02 Liposome Company Dehydrated liposomes
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US5736155A (en) * 1984-08-08 1998-04-07 The Liposome Company, Inc. Encapsulation of antineoplastic agents in liposomes
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US5252263A (en) * 1986-06-16 1993-10-12 The Liposome Company, Inc. Induction of asymmetry in vesicles
MX9203808A (es) * 1987-03-05 1992-07-01 Liposome Co Inc Formulaciones de alto contenido de medicamento: lipido, de agentes liposomicos-antineoplasticos.
US4950432A (en) * 1987-10-16 1990-08-21 Board Of Regents, The University Of Texas System Polyene microlide pre-liposomal powders
US4946683A (en) * 1987-11-18 1990-08-07 Vestar, Inc. Multiple step entrapment/loading procedure for preparing lipophilic drug-containing liposomes
JP2792702B2 (ja) * 1988-10-05 1998-09-03 ネクスター・フアーマシユーテイカルズ・インコーポレイテツド 乾燥時に改善された安定性を示すリポソームの調製方法
US5091187A (en) * 1990-04-26 1992-02-25 Haynes Duncan H Phospholipid-coated microcrystals: injectable formulations of water-insoluble drugs
US5246707A (en) * 1990-04-26 1993-09-21 Haynes Duncan H Sustained release delivery of water-soluble bio-molecules and drugs using phospholipid-coated microcrystals, microdroplets and high-concentration liposomes
US5091188A (en) * 1990-04-26 1992-02-25 Haynes Duncan H Phospholipid-coated microcrystals: injectable formulations of water-insoluble drugs
ATE138803T1 (de) * 1990-07-31 1996-06-15 Liposome Co Inc Anhäufung von aminosäuren und peptiden in liposomen
US5462740A (en) * 1993-09-17 1995-10-31 Athena Neurosciences, Inc. Rectally-administered, epileptic-seizure-inhibiting composition
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US6518412B1 (en) 1997-09-29 2003-02-11 Jean-Louis Dasseux Gene therapy approaches to supply apolipoprotein A-I agonists and their use to treat dyslipidemic disorders
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GB1575343A (en) * 1977-05-10 1980-09-17 Ici Ltd Method for preparing liposome compositions containing biologically active compounds
CH621479A5 (no) * 1977-08-05 1981-02-13 Battelle Memorial Institute

Also Published As

Publication number Publication date
NO801863L (no) 1980-12-22
ZA803567B (en) 1981-06-24
FI72875C (fi) 1987-08-10
ES492676A0 (es) 1981-05-16
IE49615B1 (en) 1985-10-30
DK155172C (da) 1989-09-18
AU5928980A (en) 1981-01-08
PT71436A (en) 1980-07-01
MC1336A1 (fr) 1981-04-21
ATE5508T1 (de) 1983-12-15
KR850001301B1 (ko) 1985-09-12
DK266680A (da) 1980-12-23
EP0021337A3 (en) 1981-04-22
PH16795A (en) 1984-02-28
DK155172B (da) 1989-02-27
HU186296B (en) 1985-07-29
FI801876A (fi) 1980-12-23
DE3065818D1 (en) 1984-01-12
IE801281L (en) 1980-12-22
JPS567714A (en) 1981-01-27
US4411894A (en) 1983-10-25
AU534959B2 (en) 1984-02-23
EP0021337B1 (de) 1983-12-07
NO155226B (no) 1986-11-24
KR830002327A (ko) 1983-05-28
IL60326A (en) 1983-09-30
CA1173360A (en) 1984-08-28
EP0021337A2 (de) 1981-01-07
ES8104720A1 (es) 1981-05-16
FI72875B (fi) 1987-04-30
PT71436B (en) 1981-10-23
AR230178A1 (es) 1984-03-01
IL60326A0 (en) 1980-09-16
NZ194047A (en) 1982-09-14

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