ECSP099693A - Ligandos de receptor vainilloide novedosos y el uso de los mismos para la produccion de farmacos - Google Patents

Ligandos de receptor vainilloide novedosos y el uso de los mismos para la produccion de farmacos

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Publication number
ECSP099693A
ECSP099693A EC2009009693A ECSP099693A ECSP099693A EC SP099693 A ECSP099693 A EC SP099693A EC 2009009693 A EC2009009693 A EC 2009009693A EC SP099693 A ECSP099693 A EC SP099693A EC SP099693 A ECSP099693 A EC SP099693A
Authority
EC
Ecuador
Prior art keywords
production
vinylloid
pharmacos
new
same
Prior art date
Application number
EC2009009693A
Other languages
English (en)
Spanish (es)
Inventor
Derek Saunders
Jee Woo Lee
Vry Jean Marie Victor De
Thomas Christoph
Michael Przewosny
Robert Frank
Gregor Bahrenberg
Klaus Schiene
Bernd Saudermann
Original Assignee
Gruenenthal Chemie
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Gruenenthal Chemie filed Critical Gruenenthal Chemie
Publication of ECSP099693A publication Critical patent/ECSP099693A/es

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    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D213/00Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72Nitrogen atoms
    • C07D213/74Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
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    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
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    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4402Non condensed pyridines; Hydrogenated derivatives thereof only substituted in position 2, e.g. pheniramine, bisacodyl
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    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
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EC2009009693A 2007-04-16 2009-10-16 Ligandos de receptor vainilloide novedosos y el uso de los mismos para la produccion de farmacos ECSP099693A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE102007018151A DE102007018151A1 (de) 2007-04-16 2007-04-16 Neue Vanilloid-Rezeptor Liganden und ihre Verwendung zur Herstellung von Arzneimitteln

Publications (1)

Publication Number Publication Date
ECSP099693A true ECSP099693A (es) 2009-11-30

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Family Applications (1)

Application Number Title Priority Date Filing Date
EC2009009693A ECSP099693A (es) 2007-04-16 2009-10-16 Ligandos de receptor vainilloide novedosos y el uso de los mismos para la produccion de farmacos

Country Status (16)

Country Link
US (2) US8642775B2 (enExample)
EP (1) EP2146962A2 (enExample)
JP (1) JP5557734B2 (enExample)
KR (1) KR101497357B1 (enExample)
CN (1) CN101687799B (enExample)
BR (1) BRPI0810031A2 (enExample)
CA (1) CA2683910A1 (enExample)
CO (1) CO6220938A2 (enExample)
DE (1) DE102007018151A1 (enExample)
EC (1) ECSP099693A (enExample)
IL (1) IL201506A0 (enExample)
MX (1) MX2009011139A (enExample)
NZ (2) NZ580381A (enExample)
RU (1) RU2487120C2 (enExample)
WO (1) WO2008125337A2 (enExample)
ZA (1) ZA200907096B (enExample)

Families Citing this family (14)

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WO2008110351A2 (en) * 2007-03-15 2008-09-18 Dompe' Pha.R.Ma S.P.A. Use of (r) and (s)-2-aryl-propionic acid derivatives as antiseptic agents
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