ZA200907096B - Novel vanilloid receptor ligands and the use thereof for the production of pharmaceuticals - Google Patents

Novel vanilloid receptor ligands and the use thereof for the production of pharmaceuticals

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Publication number
ZA200907096B
ZA200907096B ZA2009/07096A ZA200907096A ZA200907096B ZA 200907096 B ZA200907096 B ZA 200907096B ZA 2009/07096 A ZA2009/07096 A ZA 2009/07096A ZA 200907096 A ZA200907096 A ZA 200907096A ZA 200907096 B ZA200907096 B ZA 200907096B
Authority
ZA
South Africa
Prior art keywords
pharmaceuticals
production
receptor ligands
vanilloid receptor
novel vanilloid
Prior art date
Application number
ZA2009/07096A
Other languages
English (en)
Inventor
Robert Frank
Gregor Bahrenberg
Thomas Christoph
Klaus Schiene
Vry Jean De
Derek John Saunders
Michael Przewosny
Bernd Sundermann
Jeewoo Lee
Original Assignee
Gruenenthal Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Gruenenthal Gmbh filed Critical Gruenenthal Gmbh
Publication of ZA200907096B publication Critical patent/ZA200907096B/en

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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72—Nitrogen atoms
    • C07D213/74—Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
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ZA2009/07096A 2007-04-16 2009-10-12 Novel vanilloid receptor ligands and the use thereof for the production of pharmaceuticals ZA200907096B (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE102007018151A DE102007018151A1 (de) 2007-04-16 2007-04-16 Neue Vanilloid-Rezeptor Liganden und ihre Verwendung zur Herstellung von Arzneimitteln
PCT/EP2008/002994 WO2008125337A2 (de) 2007-04-16 2008-04-15 Neue vanilloid-rezeptor liganden und ihre verwendung zur herstellung von arzneimitteln

Publications (1)

Publication Number Publication Date
ZA200907096B true ZA200907096B (en) 2013-03-27

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ZA2009/07096A ZA200907096B (en) 2007-04-16 2009-10-12 Novel vanilloid receptor ligands and the use thereof for the production of pharmaceuticals

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US (2) US8642775B2 (enExample)
EP (1) EP2146962A2 (enExample)
JP (1) JP5557734B2 (enExample)
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WO2008125337A2 (de) 2008-10-23
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CO6220938A2 (es) 2010-11-19
US20080262039A1 (en) 2008-10-23
NZ580381A (en) 2012-05-25
CN101687799A (zh) 2010-03-31
CA2683910A1 (en) 2008-04-16
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AU2008238245A1 (en) 2008-10-23
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IL201506A0 (en) 2010-05-31
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JP5557734B2 (ja) 2014-07-23
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ECSP099693A (es) 2009-11-30
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CN101687799B (zh) 2014-07-23
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KR20100016594A (ko) 2010-02-12
KR101497357B1 (ko) 2015-03-02
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US8791268B2 (en) 2014-07-29
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