ECSP034754A - Derivados de beta-carbolina y su uso farmaceutico contra depresion y ansiedad - Google Patents

Derivados de beta-carbolina y su uso farmaceutico contra depresion y ansiedad

Info

Publication number
ECSP034754A
ECSP034754A EC2003004754A ECSP034754A ECSP034754A EC SP034754 A ECSP034754 A EC SP034754A EC 2003004754 A EC2003004754 A EC 2003004754A EC SP034754 A ECSP034754 A EC SP034754A EC SP034754 A ECSP034754 A EC SP034754A
Authority
EC
Ecuador
Prior art keywords
carbolina
anxiety
beta
derivatives
pharmaceutical use
Prior art date
Application number
EC2003004754A
Other languages
English (en)
Spanish (es)
Inventor
Konstanze Hurth
Thomas J Troxler
Daniel Hoyer
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of ECSP034754A publication Critical patent/ECSP034754A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/22Anxiolytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Psychiatry (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pain & Pain Management (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
EC2003004754A 2001-04-03 2003-08-27 Derivados de beta-carbolina y su uso farmaceutico contra depresion y ansiedad ECSP034754A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB0108337.7A GB0108337D0 (en) 2001-04-03 2001-04-03 Organic compounds

Publications (1)

Publication Number Publication Date
ECSP034754A true ECSP034754A (es) 2003-10-28

Family

ID=9912165

Family Applications (1)

Application Number Title Priority Date Filing Date
EC2003004754A ECSP034754A (es) 2001-04-03 2003-08-27 Derivados de beta-carbolina y su uso farmaceutico contra depresion y ansiedad

Country Status (27)

Country Link
US (1) US6861430B2 (OSRAM)
EP (1) EP1377578B1 (OSRAM)
JP (1) JP4405732B2 (OSRAM)
KR (1) KR100564840B1 (OSRAM)
CN (1) CN1309721C (OSRAM)
AR (1) AR035451A1 (OSRAM)
AT (1) ATE517104T1 (OSRAM)
AU (1) AU2002316828B2 (OSRAM)
BR (1) BR0208566B1 (OSRAM)
CA (1) CA2440014C (OSRAM)
CZ (1) CZ295992B6 (OSRAM)
EC (1) ECSP034754A (OSRAM)
ES (1) ES2368389T3 (OSRAM)
GB (1) GB0108337D0 (OSRAM)
HU (1) HUP0400317A3 (OSRAM)
IL (1) IL157545A0 (OSRAM)
MX (1) MXPA03009057A (OSRAM)
MY (1) MY134026A (OSRAM)
NO (1) NO20034413D0 (OSRAM)
NZ (1) NZ528370A (OSRAM)
PE (1) PE20021018A1 (OSRAM)
PL (1) PL210861B1 (OSRAM)
PT (1) PT1377578E (OSRAM)
RU (1) RU2003130644A (OSRAM)
SK (1) SK12222003A3 (OSRAM)
WO (1) WO2002081471A1 (OSRAM)
ZA (1) ZA200306108B (OSRAM)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE10164139A1 (de) 2001-12-27 2003-07-10 Bayer Ag 2-Heteroarylcarbonsäureamide
US7872133B2 (en) 2003-06-23 2011-01-18 Ono Pharmaceutical Co., Ltd. Tricyclic heterocycle compound
AR051780A1 (es) * 2004-11-29 2007-02-07 Japan Tobacco Inc Compuestos en anillo fusionados que contienen nitrogeno y utilizacion de los mismos
PT1829874E (pt) 2004-12-22 2014-04-10 Ono Pharmaceutical Co Composto tricíclico e sua utilização
US7879859B2 (en) 2005-11-21 2011-02-01 Merck Sharp & Dohme Corp. Diagnosis and treatment of type 2 diabetes and other disorders
WO2007062175A2 (en) * 2005-11-21 2007-05-31 Amgen Inc. Spiro-substituted tricyclic heterocycles cxcr3 antagonists
JP2010533712A (ja) * 2007-07-19 2010-10-28 メルク・シャープ・エンド・ドーム・コーポレイション 抗糖尿病化合物としてのベータカルボリン誘導体
WO2009016329A1 (en) * 2007-07-31 2009-02-05 Cambridge Enterprise Limited Use of gabaa receptor antagonists to treat cognitive impairment in patients with psychiatric conditions
US8338604B2 (en) 2008-06-20 2012-12-25 Bristol-Myers Squibb Company Imidazopyridine and imidazopyrazine compounds useful as kinase inhibitors
CA2744278C (en) 2008-11-19 2015-09-08 Envivo Pharmaceuticals, Inc. Treatment of cognitive disorders with (r)-7-chloro-n-(quinuclidin-3-yl)benzo[b]thiophene-2-carboxamide and pharmaceutically acceptable salts thereof
TW201028414A (en) 2009-01-16 2010-08-01 Merck Sharp & Dohme Oxadiazole beta carboline derivatives as antidiabetic compounds
CN102695414A (zh) 2010-01-15 2012-09-26 默沙东公司 作为抗糖尿病化合物的噁二唑β-咔啉衍生物
CN103221411B (zh) 2010-05-17 2016-05-11 富瑞姆制药公司 (R)-7-氯-N-(奎宁环-3-基)苯并[b]噻吩-2-甲酰胺盐酸盐单水合物的晶型
CA2872005A1 (en) 2012-05-08 2013-11-14 Forum Pharmaceuticals, Inc. Methods of maintaining, treating or improving cognitive function
CN111349096B (zh) * 2020-04-14 2021-03-09 石河子大学 一种吲哚类化合物及其制备方法、应用
KR102467844B1 (ko) 2021-04-21 2022-11-16 삼성전자주식회사 솔리드 스테이트 드라이브 장치 및 이를 포함하는 데이터 저장 장치

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE4118741A1 (de) * 1991-06-05 1992-12-10 Schering Ag Neue hetaryloxy-(beta)-carboline, deren herstellung und verwendung in arzneimitteln
US6057340A (en) * 1998-02-03 2000-05-02 American Home Products Corporation Oxazole derivatives as serotonin-1A receptor agonists
DE69904595T2 (de) 1998-06-12 2003-11-27 Societe De Conseils De Recherches Et D'applications Scientifiques S.A., Paris Betacarbolinverbindungen

Also Published As

Publication number Publication date
NO20034413L (no) 2003-10-02
RU2003130644A (ru) 2005-04-10
KR100564840B1 (ko) 2006-03-28
NO20034413D0 (no) 2003-10-02
CA2440014C (en) 2010-11-23
CZ20032655A3 (cs) 2003-12-17
GB0108337D0 (en) 2001-05-23
PL210861B1 (pl) 2012-03-30
AR035451A1 (es) 2004-05-26
SK12222003A3 (sk) 2004-06-08
KR20040008150A (ko) 2004-01-28
CA2440014A1 (en) 2002-10-17
CZ295992B6 (cs) 2005-12-14
JP2004525178A (ja) 2004-08-19
CN1309721C (zh) 2007-04-11
HUP0400317A3 (en) 2007-10-29
BR0208566A (pt) 2004-03-30
ATE517104T1 (de) 2011-08-15
PE20021018A1 (es) 2003-01-13
AU2002316828B2 (en) 2006-05-11
WO2002081471A1 (en) 2002-10-17
ES2368389T3 (es) 2011-11-16
PT1377578E (pt) 2011-09-23
NZ528370A (en) 2005-10-28
JP4405732B2 (ja) 2010-01-27
US6861430B2 (en) 2005-03-01
EP1377578B1 (en) 2011-07-20
IL157545A0 (en) 2004-03-28
ZA200306108B (en) 2004-07-05
CN1500090A (zh) 2004-05-26
EP1377578A1 (en) 2004-01-07
US20040132735A1 (en) 2004-07-08
PL362571A1 (en) 2004-11-02
MXPA03009057A (es) 2004-02-12
MY134026A (en) 2007-11-30
BR0208566B1 (pt) 2013-12-24
HUP0400317A2 (hu) 2004-09-28

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