EA201270749A1 - Композиции с вирусным ингибитором для терапевтического применения in vivo, включающие сочетание (-)-карвона, (+) карвона, гераниола и дополнительного эфиромасличного компонента - Google Patents

Композиции с вирусным ингибитором для терапевтического применения in vivo, включающие сочетание (-)-карвона, (+) карвона, гераниола и дополнительного эфиромасличного компонента

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Publication number
EA201270749A1
EA201270749A1 EA201270749A EA201270749A EA201270749A1 EA 201270749 A1 EA201270749 A1 EA 201270749A1 EA 201270749 A EA201270749 A EA 201270749A EA 201270749 A EA201270749 A EA 201270749A EA 201270749 A1 EA201270749 A1 EA 201270749A1
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Eurasian Patent Office
Prior art keywords
carvon
geraniol
combination
essential oil
vivo
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EA201270749A
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English (en)
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EA025278B1 (ru
EA025278B9 (ru
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Кристин Коппен
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Сеса Альянс С.А.
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Application filed by Сеса Альянс С.А. filed Critical Сеса Альянс С.А.
Publication of EA201270749A1 publication Critical patent/EA201270749A1/ru
Publication of EA025278B1 publication Critical patent/EA025278B1/ru
Publication of EA025278B9 publication Critical patent/EA025278B9/ru

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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/12Ketones
    • A61K31/122Ketones having the oxygen directly attached to a ring, e.g. quinones, vitamin K1, anthralin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/045Hydroxy compounds, e.g. alcohols; Salts thereof, e.g. alcoholates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/075Ethers or acetals
    • A61K31/085Ethers or acetals having an ether linkage to aromatic ring nuclear carbon
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/14Quaternary ammonium compounds, e.g. edrophonium, choline
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/16Amides, e.g. hydroxamic acids
    • A61K31/18Sulfonamides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/336Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having three-membered rings, e.g. oxirane, fumagillin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/16Antivirals for RNA viruses for influenza or rhinoviruses
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/20Antivirals for DNA viruses
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/20Antivirals for DNA viruses
    • A61P31/22Antivirals for DNA viruses for herpes viruses
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02ATECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Virology (AREA)
  • Epidemiology (AREA)
  • Communicable Diseases (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Molecular Biology (AREA)
  • Biotechnology (AREA)
  • Engineering & Computer Science (AREA)
  • Pulmonology (AREA)
  • AIDS & HIV (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Micro-Organisms Or Cultivation Processes Thereof (AREA)

Abstract

Настоящее изобретение относится к антивирусной композиции, включающей следующие компоненты: R-(-)-2-метил-5-(проп-1-ен-2-ил)-циклогекс-2-енон (также именуемый (-)-карвоном) и S-(+)-2-метил-5-(проп-1-ен-2-ил)-циклогекс-2-енон (также именуемый (+)-карвоном), и (2Е)-3,7-диметилоктан-2,6-диен-1-ол (также именуемый транс-гераниолом) в сочетании по меньшей мере с еще одним компонентом, избранным из эфиромасличных компонентов для применения в лечении и профилактике расстройств, вызванных вирусами с ДНК и заключенными в оболочку, вирусами с ДНК и не заключенными в оболочку, вирусами с РНК и заключенными в оболочку, вирусами с РНК и не заключенными в оболочку.
EA201270749A 2010-03-26 2011-03-28 Антивирусная композиция против заключенных или незаключенных в оболочку днк- или рнк-вирусов EA025278B9 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP10157930A EP2368547B1 (en) 2010-03-26 2010-03-26 Antiviral compositions comprising geraniol and carvone
PCT/EP2011/054758 WO2011117424A1 (en) 2010-03-26 2011-03-28 Viral inhibitor compositions for in vivo therapeutic use comprising a combination of (-) -carvone, geraniol and a further essential oil component

Publications (3)

Publication Number Publication Date
EA201270749A1 true EA201270749A1 (ru) 2013-03-29
EA025278B1 EA025278B1 (ru) 2016-12-30
EA025278B9 EA025278B9 (ru) 2017-03-31

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EA201270749A EA025278B9 (ru) 2010-03-26 2011-03-28 Антивирусная композиция против заключенных или незаключенных в оболочку днк- или рнк-вирусов

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US (2) US8980945B2 (ru)
EP (2) EP2368547B1 (ru)
JP (1) JP5342085B2 (ru)
KR (1) KR101340260B1 (ru)
CN (1) CN102946876B (ru)
AU (1) AU2011231511B2 (ru)
BR (1) BR112012024260B1 (ru)
CA (1) CA2790087C (ru)
CL (1) CL2012002606A1 (ru)
CO (1) CO6602166A2 (ru)
CY (3) CY1113449T1 (ru)
DK (2) DK2368547T3 (ru)
EA (1) EA025278B9 (ru)
ES (2) ES2392938T3 (ru)
HK (1) HK1176019A1 (ru)
HR (2) HRP20120964T1 (ru)
HU (1) HUE026121T2 (ru)
IL (1) IL222048A (ru)
LU (1) LU91805B1 (ru)
MA (1) MA34074B1 (ru)
ME (1) ME02035B (ru)
MX (1) MX346412B (ru)
MY (2) MY153104A (ru)
NZ (1) NZ602602A (ru)
PE (2) PE20130065A1 (ru)
PL (2) PL2368547T3 (ru)
PT (2) PT2368547E (ru)
RS (2) RS52544B (ru)
SG (1) SG184039A1 (ru)
SI (2) SI2368547T1 (ru)
SM (2) SMT201200062B (ru)
TN (2) TN2012000444A1 (ru)
UA (1) UA102497C2 (ru)
WO (1) WO2011117424A1 (ru)
ZA (2) ZA201208116B (ru)

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TWI463979B (zh) * 2013-04-12 2014-12-11 Nat Defense Medical Ct 檸檬醛用於製備治療局部腎絲球硬化症之藥物的用途
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CN106727628A (zh) * 2016-12-17 2017-05-31 郑州郑先医药科技有限公司 一种治疗慢性腹泻的西药组合物
KR101970281B1 (ko) * 2017-07-28 2019-04-18 고려대학교 산학협력단 리나릴 아세테이트를 포함하는 올메사탄으로 유발된 장운동과다증의 예방 또는 치료용 조성물
CN107648488A (zh) * 2017-09-29 2018-02-02 陈晓阳 一种用于治疗慢性咽炎的丸剂
KR102118181B1 (ko) * 2018-06-12 2020-06-02 광주여자대학교 산학협력단 식물성 정유를 유효성분으로 포함하는 a형 인플루엔자 바이러스에 대한 항바이러스 조성물
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CN111012769B (zh) * 2019-12-05 2021-02-12 青海大学 一种用于治疗包虫病的药物组合物、药物制剂及乳剂制备方法
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CN114716327A (zh) * 2020-12-14 2022-07-08 中南民族大学 柏木醇衍生物、其制备方法及其应用
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JP7133820B1 (ja) * 2021-06-09 2022-09-09 塩野香料株式会社 コロナウイルス感染症予防用香料組成物及び結合阻害剤
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EA025278B1 (ru) 2016-12-30
CO6602166A2 (es) 2013-01-18
US8980945B2 (en) 2015-03-17
AU2011231511B2 (en) 2014-03-20
DK2555763T3 (da) 2014-08-04
PE20141008A1 (es) 2014-09-20
PE20130065A1 (es) 2013-03-08
LU91805B1 (fr) 2011-09-26
NZ602602A (en) 2012-12-21
KR101340260B1 (ko) 2013-12-10
CA2790087C (en) 2013-07-30
CY1113449T1 (el) 2016-06-22
SI2368547T1 (sl) 2013-01-31
RS53435B (en) 2014-12-31
EA025278B9 (ru) 2017-03-31
CN102946876A (zh) 2013-02-27
CA2790087A1 (en) 2011-09-29
PT2555763E (pt) 2014-08-04
MY153104A (en) 2014-12-31
KR20120128716A (ko) 2012-11-27
RS52544B (en) 2013-04-30
CL2012002606A1 (es) 2013-10-18
HRP20140706T1 (hr) 2014-09-12
JP2013523622A (ja) 2013-06-17
SI2555763T1 (sl) 2014-08-29
WO2011117424A1 (en) 2011-09-29
AU2011231511A1 (en) 2012-10-18
PL2555763T3 (pl) 2014-09-30
TN2012000444A1 (en) 2014-01-30
ZA201208116B (en) 2014-04-30
SG184039A1 (en) 2012-10-30
MX346412B (es) 2017-03-17
BR112012024260A2 (pt) 2016-07-12
ES2486765T3 (es) 2014-08-19
ME02035B (me) 2013-04-30
SMT201400104B (it) 2014-09-08
US20130225676A1 (en) 2013-08-29
IL222048A (en) 2014-09-30
MX2012010949A (es) 2013-01-29
TN2013000366A1 (en) 2015-01-20
SMT201200062B (it) 2013-03-08
EP2555763B1 (en) 2014-04-30
HRP20120964T1 (en) 2012-12-31
HUE026121T2 (en) 2016-05-30
CN102946876B (zh) 2016-04-06
EP2368547A1 (en) 2011-09-28
PT2368547E (pt) 2012-11-20
EP2368547B1 (en) 2012-09-12
HK1176019A1 (en) 2013-07-19
CY1119841T1 (el) 2018-06-27
MY158757A (en) 2016-11-15
EP2555763A1 (en) 2013-02-13
UA102497C2 (ru) 2013-07-10
MA34074B1 (fr) 2013-03-05
CY1115375T1 (el) 2017-01-04
ES2392938T3 (es) 2012-12-17
BR112012024260B1 (pt) 2019-12-31
PL2368547T3 (pl) 2013-02-28
US8883859B1 (en) 2014-11-11
DK2368547T3 (da) 2013-01-02
ZA201306926B (en) 2014-04-30
JP5342085B2 (ja) 2013-11-13

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