EA201200016A1 - Лечение приливов, вазомоторных симптомов и ночной потливости с помощью предшественников половых стероидов в комбинации с избирательными (селективными) модуляторами эстрогеновых рецепторов - Google Patents

Лечение приливов, вазомоторных симптомов и ночной потливости с помощью предшественников половых стероидов в комбинации с избирательными (селективными) модуляторами эстрогеновых рецепторов

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Publication number
EA201200016A1
EA201200016A1 EA201200016A EA201200016A EA201200016A1 EA 201200016 A1 EA201200016 A1 EA 201200016A1 EA 201200016 A EA201200016 A EA 201200016A EA 201200016 A EA201200016 A EA 201200016A EA 201200016 A1 EA201200016 A1 EA 201200016A1
Authority
EA
Eurasian Patent Office
Prior art keywords
estrogen receptors
vasomotor symptoms
selective
night
electoral
Prior art date
Application number
EA201200016A
Other languages
English (en)
Russian (ru)
Inventor
Фернанд Лабри
Original Assignee
Эндорешерш, Инк.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43306950&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=EA201200016(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Эндорешерш, Инк. filed Critical Эндорешерш, Инк.
Publication of EA201200016A1 publication Critical patent/EA201200016A1/xx

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    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • A61K31/568—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in positions 10 and 13 by a chain having at least one carbon atom, e.g. androstanes, e.g. testosterone
    • A61K31/5685—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in positions 10 and 13 by a chain having at least one carbon atom, e.g. androstanes, e.g. testosterone having an oxo group in position 17, e.g. androsterone
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    • A61K31/138—Aryloxyalkylamines, e.g. propranolol, tamoxifen, phenoxybenzamine
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    • A61K31/19—Carboxylic acids, e.g. valproic acid
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  • Hematology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
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  • Gynecology & Obstetrics (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Rheumatology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Anesthesiology (AREA)
  • Psychiatry (AREA)
  • Hospice & Palliative Care (AREA)
  • Emergency Medicine (AREA)
  • Pregnancy & Childbirth (AREA)
  • Vascular Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
EA201200016A 2009-06-16 2010-06-16 Лечение приливов, вазомоторных симптомов и ночной потливости с помощью предшественников половых стероидов в комбинации с избирательными (селективными) модуляторами эстрогеновых рецепторов EA201200016A1 (ru)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US18754909P 2009-06-16 2009-06-16
US12/791,174 US20100317635A1 (en) 2009-06-16 2010-06-01 Treatment of hot flushes, vasomotor symptoms, and night sweats with sex steroid precursors in combination with selective estrogen receptor modulators
PCT/CA2010/000898 WO2010145010A1 (en) 2009-06-16 2010-06-16 Treatment of hot flushes, vasomotor symptoms, and night sweats with sex steroid precursors in combination with selective estrogen receptor modulators

Publications (1)

Publication Number Publication Date
EA201200016A1 true EA201200016A1 (ru) 2012-08-30

Family

ID=43306950

Family Applications (1)

Application Number Title Priority Date Filing Date
EA201200016A EA201200016A1 (ru) 2009-06-16 2010-06-16 Лечение приливов, вазомоторных симптомов и ночной потливости с помощью предшественников половых стероидов в комбинации с избирательными (селективными) модуляторами эстрогеновых рецепторов

Country Status (20)

Country Link
US (4) US20100317635A1 (ko)
EP (3) EP3682880A1 (ko)
JP (4) JP2012530074A (ko)
KR (10) KR20170078879A (ko)
CN (3) CN104352504A (ko)
AR (1) AR077119A1 (ko)
AU (1) AU2010262722A1 (ko)
BR (1) BRPI1011561A2 (ko)
CA (2) CA2893236A1 (ko)
CL (1) CL2011003172A1 (ko)
EA (1) EA201200016A1 (ko)
HK (1) HK1204550A1 (ko)
IL (2) IL216963A (ko)
MA (1) MA33434B1 (ko)
MX (1) MX338290B (ko)
NZ (1) NZ597583A (ko)
SG (3) SG10201705761YA (ko)
TW (1) TWI612044B (ko)
WO (1) WO2010145010A1 (ko)
ZA (1) ZA201109198B (ko)

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US10179107B2 (en) 2011-07-19 2019-01-15 Pantarhei Bioscience B.V. Tablet containing dehydroepiandrosterone (DHEA)
BR112014014124A2 (pt) 2011-12-14 2017-08-22 Seragon Pharmaceutical Inc Moduladores do receptor de estrogênio fluorados e usos dos mesmos
PE20150099A1 (es) 2011-12-16 2015-01-30 Olema Pharmaceuticals Inc Compuestos novedosos de benzopirano, composiciones y usos de los mismos
US20150071857A1 (en) * 2012-03-07 2015-03-12 Ligand Pharmaceuticals, Inc. Steroid hormone and cholesterol pathways as one unified homeostatic system
WO2014008159A1 (en) * 2012-07-03 2014-01-09 The University Of North Carolina At Chapel Hill Selective estrogen receptor degraders for treatment of tamoxifen resistant tumors
WO2014203129A1 (en) 2013-06-19 2014-12-24 Olema Pharmaceuticals, Inc. Combinations of benzopyran compounds, compositions and uses thereof
WO2014203132A1 (en) 2013-06-19 2014-12-24 Olema Pharmaceuticals, Inc. Substituted benzopyran compounds, compositions and uses thereof
CN103739456A (zh) * 2013-12-03 2014-04-23 镇江圣安医药有限公司 2-（对-（（z-4-氯-1,2-二苯基-1-丁烯基）苯氧基）乙醇的新型衍生物及其应用
US9744177B2 (en) 2014-03-10 2017-08-29 Endorecherche, Inc. Treatment of male androgen deficiency symptoms or diseases with sex steroid precursor combined with SERM
WO2016174011A1 (en) * 2015-04-28 2016-11-03 Cutech Srl Compositions comprising valerian extracts
AU2016347679B2 (en) * 2015-10-27 2020-06-25 Sun Pharma Advanced Research Company Limited Novel heterocyclic antiestrogens
WO2017162206A1 (zh) * 2016-03-25 2017-09-28 南京明德新药研发股份有限公司 作为雌激素受体降解剂的吲哚并取代哌啶类化合物
PL3449017T3 (pl) * 2016-04-29 2022-06-27 Board Of Regents, The University Of Texas System Ukierunkowane pomiary aktywności transkrypcyjnej związanej z receptorami hormonów
CN109640958B (zh) * 2016-05-20 2022-11-22 蔚蓝生物技术股份有限公司 包含选择性雌激素受体调节剂(serm)的阴道递送系统及其用途
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