EA201001371A1 - Конденсированные пиримидиноновые соединения как модуляторы trpv3 - Google Patents

Конденсированные пиримидиноновые соединения как модуляторы trpv3

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Publication number
EA201001371A1
EA201001371A1 EA201001371A EA201001371A EA201001371A1 EA 201001371 A1 EA201001371 A1 EA 201001371A1 EA 201001371 A EA201001371 A EA 201001371A EA 201001371 A EA201001371 A EA 201001371A EA 201001371 A1 EA201001371 A1 EA 201001371A1
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EA
Eurasian Patent Office
Prior art keywords
trpv3
modulators
pyrimidine compounds
condensed pyrimidine
conditions
Prior art date
Application number
EA201001371A
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English (en)
Inventor
Лингам В.С. Прасада Рао
Чаудхари Сачин Сундарлал
Томас Абрахам
Кхайраткар-Джоши Неелима
Каттиге Видья Дж.
Original Assignee
Гленмарк Фармасьютикалс, С.А.
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Application filed by Гленмарк Фармасьютикалс, С.А. filed Critical Гленмарк Фармасьютикалс, С.А.
Publication of EA201001371A1 publication Critical patent/EA201001371A1/ru

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Abstract

Изобретение предусматривает модуляторы ванилоидных рецепторов преходящих потенциалов (TRPV). В частности, описанные тут соединения пригодны для лечения или профилактики заболеваний, состояний и/или расстройств, модулируемых TRPV3. Также предлагаются способы получения соединений, описанных тут, промежуточных соединений, используемых для их синтеза, их фармацевтические композиции, и способы лечения или профилактики заболеваний, состояний и/или расстройств, модулируемых TRPV3.
EA201001371A 2008-04-23 2009-04-15 Конденсированные пиримидиноновые соединения как модуляторы trpv3 EA201001371A1 (ru)

Applications Claiming Priority (9)

Application Number Priority Date Filing Date Title
IN902MU2008 2008-04-23
US5797108P 2008-06-02 2008-06-02
IN1201MU2008 2008-06-05
US7411208P 2008-06-19 2008-06-19
IN1687MU2008 2008-08-08
US9232408P 2008-08-27 2008-08-27
IN2174MU2008 2008-10-10
US11334408P 2008-11-11 2008-11-11
PCT/IB2009/005290 WO2009130560A1 (en) 2008-04-23 2009-04-15 Fused pyrimidineone compounds as trpv3 modulators

Publications (1)

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EA201001371A1 true EA201001371A1 (ru) 2011-08-30

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EA201001371A EA201001371A1 (ru) 2008-04-23 2009-04-15 Конденсированные пиримидиноновые соединения как модуляторы trpv3

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US (3) US8119647B2 (ru)
EP (2) EP2283017B1 (ru)
JP (1) JP5461525B2 (ru)
KR (1) KR20110005715A (ru)
CN (1) CN102015715A (ru)
AP (1) AP2010005408A0 (ru)
AU (1) AU2009239694B2 (ru)
BR (1) BRPI0910503A2 (ru)
CA (1) CA2720357A1 (ru)
EA (1) EA201001371A1 (ru)
GE (1) GEP20146026B (ru)
IL (1) IL208875A (ru)
MX (1) MX2010011028A (ru)
NZ (1) NZ595778A (ru)
WO (1) WO2009130560A1 (ru)
ZA (1) ZA201008347B (ru)

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