EA201190004A1 - Конденсированные имидазол карбоксамиды в качестве модуляторов trpv3 - Google Patents

Конденсированные имидазол карбоксамиды в качестве модуляторов trpv3

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Publication number
EA201190004A1
EA201190004A1 EA201190004A EA201190004A EA201190004A1 EA 201190004 A1 EA201190004 A1 EA 201190004A1 EA 201190004 A EA201190004 A EA 201190004A EA 201190004 A EA201190004 A EA 201190004A EA 201190004 A1 EA201190004 A1 EA 201190004A1
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EA
Eurasian Patent Office
Prior art keywords
trpv3
methods
imidazole carboxamide
condensed imidazole
modulators
Prior art date
Application number
EA201190004A
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English (en)
Inventor
Сачин Сундарлал Чаудхари
Абрахам Томас
Ашок Бхаусахеб Кадам
Сачин Васантрао Дхоне
Суреш Махадев Кадам
Неелима Кхайраткар-Джоши
Видийа Ганапати Каттиге
Original Assignee
Гленмарк Фармасьютикалс, С.А.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
Application filed by Гленмарк Фармасьютикалс, С.А. filed Critical Гленмарк Фармасьютикалс, С.А.
Publication of EA201190004A1 publication Critical patent/EA201190004A1/ru

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Abstract

Данное изобретение относится к модуляторам активности рецептора транзиторного потенциала по ваниллоиду (TRPV) формулы (I). В частности, описанные здесь соединения полезны для лечения или предотвращения заболеваний, патологических состояний и/или нарушений, модулируемых действием TRPV3. Изобретение также относится к способам получения описываемых здесь соединений, способам получения используемых для их синтеза промежуточных соединений, фармацевтическим композициям и способам лечения или предотвращения заболеваний, патологических состояний и/или нарушений, модулируемых действием TRPV3.
EA201190004A 2008-12-15 2009-12-15 Конденсированные имидазол карбоксамиды в качестве модуляторов trpv3 EA201190004A1 (ru)

Applications Claiming Priority (9)

Application Number Priority Date Filing Date Title
IN2610MU2008 2008-12-15
US14113308P 2008-12-29 2008-12-29
IN145MU2009 2009-01-22
US15024809P 2009-02-05 2009-02-05
IN1397MU2009 2009-06-10
US22161509P 2009-06-30 2009-06-30
IN1730MU2009 2009-07-29
US23745609P 2009-08-27 2009-08-27
PCT/IB2009/007951 WO2010070452A1 (en) 2008-12-15 2009-12-15 Fused imidazole carboxamides as trpv3 modulators

Publications (1)

Publication Number Publication Date
EA201190004A1 true EA201190004A1 (ru) 2012-11-30

Family

ID=42241253

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EA201190004A EA201190004A1 (ru) 2008-12-15 2009-12-15 Конденсированные имидазол карбоксамиды в качестве модуляторов trpv3

Country Status (12)

Country Link
US (1) US8318928B2 (ru)
EP (1) EP2367825A1 (ru)
JP (1) JP2012512151A (ru)
AR (1) AR076830A1 (ru)
AU (1) AU2009329192A1 (ru)
CA (1) CA2746077A1 (ru)
EA (1) EA201190004A1 (ru)
GE (1) GEP20146099B (ru)
MX (1) MX2011006132A (ru)
NZ (1) NZ595777A (ru)
TW (1) TW201022283A (ru)
WO (1) WO2010070452A1 (ru)

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CA2807538A1 (en) * 2010-08-10 2012-02-16 Abbvie Inc. Novel trpv3 modulators
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US8754101B2 (en) 2011-04-11 2014-06-17 Glaxo Group Limited N-cyclobutyl-imidazopyridine-methylamine as TRPV1 antagonists
WO2013062966A2 (en) 2011-10-24 2013-05-02 Abbvie Inc. Novel trpv3 modulators
WO2014015167A2 (en) * 2012-07-18 2014-01-23 University Of Notre Dame Du Lac 5,5-heteroaromatic anti-infective compounds
PL3552017T3 (pl) * 2016-12-09 2022-08-08 Denali Therapeutics Inc. Związki użyteczne jako inhibitory RIPK1

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Also Published As

Publication number Publication date
EP2367825A1 (en) 2011-09-28
AU2009329192A2 (en) 2012-03-29
US20100152192A1 (en) 2010-06-17
TW201022283A (en) 2010-06-16
JP2012512151A (ja) 2012-05-31
NZ595777A (en) 2013-07-26
GEP20146099B (en) 2014-05-27
MX2011006132A (es) 2011-09-01
US8318928B2 (en) 2012-11-27
CA2746077A1 (en) 2010-06-24
AU2009329192A1 (en) 2011-12-01
AR076830A1 (es) 2011-07-13
WO2010070452A1 (en) 2010-06-24

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