EA200801243A1 - Фармацевтическое применение замещенных амидов - Google Patents
Фармацевтическое применение замещенных амидовInfo
- Publication number
- EA200801243A1 EA200801243A1 EA200801243A EA200801243A EA200801243A1 EA 200801243 A1 EA200801243 A1 EA 200801243A1 EA 200801243 A EA200801243 A EA 200801243A EA 200801243 A EA200801243 A EA 200801243A EA 200801243 A1 EA200801243 A1 EA 200801243A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- substituted amides
- compounds
- pharmaceutical application
- disclosed
- pharmaceutical compositions
- Prior art date
Links
Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/433—Thidiazoles
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Landscapes
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
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- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
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- Engineering & Computer Science (AREA)
- Diabetes (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
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- Endocrinology (AREA)
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- Hematology (AREA)
- Epidemiology (AREA)
- Cardiology (AREA)
- Oncology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Psychiatry (AREA)
- Heart & Thoracic Surgery (AREA)
- Obesity (AREA)
- Communicable Diseases (AREA)
- Rheumatology (AREA)
- Hospice & Palliative Care (AREA)
- Pulmonology (AREA)
- Urology & Nephrology (AREA)
- Pain & Pain Management (AREA)
- Immunology (AREA)
- Ophthalmology & Optometry (AREA)
- Dermatology (AREA)
- Reproductive Health (AREA)
- Gastroenterology & Hepatology (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP05110228 | 2005-11-01 | ||
EP06116808 | 2006-07-07 | ||
PCT/EP2006/068015 WO2007051810A2 (en) | 2005-11-01 | 2006-11-01 | Pharmaceutical use of substituted amides |
Publications (1)
Publication Number | Publication Date |
---|---|
EA200801243A1 true EA200801243A1 (ru) | 2008-10-30 |
Family
ID=37946770
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA200801243A EA200801243A1 (ru) | 2005-11-01 | 2006-11-01 | Фармацевтическое применение замещенных амидов |
Country Status (9)
Country | Link |
---|---|
US (1) | US20090124598A1 (de) |
EP (1) | EP1948190A2 (de) |
JP (1) | JP2009514818A (de) |
KR (1) | KR20080076916A (de) |
AU (1) | AU2006310518A1 (de) |
CA (1) | CA2627306A1 (de) |
EA (1) | EA200801243A1 (de) |
IL (1) | IL191035A0 (de) |
WO (1) | WO2007051810A2 (de) |
Families Citing this family (68)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US8138342B2 (en) * | 2004-10-12 | 2012-03-20 | High Point Pharmacueticals, LLC | 11β-hydroxysteroid dehydrogenase type 1 active spiro compounds |
JP2009513611A (ja) * | 2005-11-01 | 2009-04-02 | ハイ ポイント ファーマシューティカルズ,リミティド ライアビリティ カンパニー | 置換アミドの医薬用途 |
WO2007107550A1 (en) * | 2006-03-21 | 2007-09-27 | High Point Pharmaceuticals, Llc | Adamantane derivatives for the treatment of the metabolic syndrome |
CA2648074A1 (en) | 2006-04-07 | 2007-10-18 | High Point Pharmaceuticals, Llc | 11.beta.-hydroxysteroid dehydrogenase type 1 active compounds |
CA2649677A1 (en) * | 2006-05-01 | 2007-11-15 | Incyte Corporation | Tetrasubstituted ureas as modulators of 11-.beta. hydroxyl steroid dehydrogenase type 1 |
US20090306048A1 (en) * | 2006-06-16 | 2009-12-10 | John Paul Kilburn | Pharmaceutical use of substituted piperidine carboxamides |
EP2044073A1 (de) * | 2006-07-13 | 2009-04-08 | High Point Pharmaceuticals, LLC | Verbindungen mit wirkung an der 11beta-hydroxysteroiddehydrogenase vom typ 1 |
EP1878721A1 (de) * | 2006-07-13 | 2008-01-16 | Novo Nordisk A/S | 4-Piperidylbenzamide als Inhibitoren der 11-beta-hydroxysteroiddehydrogenase Typ 1 |
RU2009108280A (ru) | 2006-08-08 | 2010-09-20 | Санофи-Авентис (Fr) | Ариламиноарилалкилзамещенные имидазолидин-2,4-дионы, способы их получения, содержащие эти соединения лекарственные средства и их применение |
WO2008101885A1 (en) * | 2007-02-23 | 2008-08-28 | High Point Pharmaceuticals, Llc | N-adamantyl benzamides as inhibitors of 11-beta-hydroxysteroid dehydrogenase |
JP2010519242A (ja) * | 2007-02-23 | 2010-06-03 | ハイ ポイント ファーマシューティカルズ,リミティド ライアビリティ カンパニー | 新規化合物 |
WO2008101886A1 (en) * | 2007-02-23 | 2008-08-28 | High Point Pharmaceuticals, Llc | N-adamantyl benzamides as inhibitors of 11-beta-hydroxysteroid dehydrogenase |
EA016951B1 (ru) | 2007-02-23 | 2012-08-30 | ХАЙ ПОЙНТ ФАРМАСЬЮТИКАЛЗ, ЭлЭлСи | N-АДАМАНТИЛБЕНЗАМИДЫ В КАЧЕСТВЕ ИНГИБИТОРОВ 11-β-ГИДРОКСИСТЕРОИДДЕГИДРОГЕНАЗЫ |
CA2678577A1 (en) | 2007-02-26 | 2008-09-04 | Vitae Pharmaceuticals, Inc. | Cyclic urea and carbamate inhibitors of 11.beta.-hydroxysteroid dehydrogenase 1 |
CN101652359A (zh) * | 2007-03-09 | 2010-02-17 | 高点制药有限责任公司 | 作为羟类固醇脱氢酶抑制剂的吲哚-和苯并咪唑酰胺类 |
CA2681934A1 (en) * | 2007-03-28 | 2008-10-02 | High Point Pharmaceuticals, Llc | 11beta-hsd1 active compounds |
ES2399912T3 (es) * | 2007-04-11 | 2013-04-04 | High Point Pharmaceuticals, Llc | Nuevos compuestos |
JP2010526777A (ja) * | 2007-04-24 | 2010-08-05 | ハイ ポイント ファーマシューティカルズ,リミティド ライアビリティ カンパニー | 置換アミドの医薬用途 |
EP2025674A1 (de) | 2007-08-15 | 2009-02-18 | sanofi-aventis | Substituierte Tetrahydronaphthaline, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel |
AR069207A1 (es) | 2007-11-07 | 2010-01-06 | Vitae Pharmaceuticals Inc | Ureas ciclicas como inhibidores de la 11 beta - hidroxi-esteroide deshidrogenasa 1 |
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-
2006
- 2006-11-01 EP EP06819214A patent/EP1948190A2/de not_active Withdrawn
- 2006-11-01 KR KR1020087012901A patent/KR20080076916A/ko not_active Application Discontinuation
- 2006-11-01 WO PCT/EP2006/068015 patent/WO2007051810A2/en active Application Filing
- 2006-11-01 US US12/092,230 patent/US20090124598A1/en not_active Abandoned
- 2006-11-01 CA CA002627306A patent/CA2627306A1/en not_active Abandoned
- 2006-11-01 JP JP2008537121A patent/JP2009514818A/ja not_active Withdrawn
- 2006-11-01 EA EA200801243A patent/EA200801243A1/xx unknown
- 2006-11-01 AU AU2006310518A patent/AU2006310518A1/en not_active Abandoned
-
2008
- 2008-04-27 IL IL191035A patent/IL191035A0/en unknown
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US20090124598A1 (en) | 2009-05-14 |
CA2627306A1 (en) | 2007-05-10 |
WO2007051810A3 (en) | 2008-01-24 |
JP2009514818A (ja) | 2009-04-09 |
WO2007051810A2 (en) | 2007-05-10 |
IL191035A0 (en) | 2009-08-03 |
AU2006310518A1 (en) | 2007-05-10 |
KR20080076916A (ko) | 2008-08-20 |
EP1948190A2 (de) | 2008-07-30 |
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