EA200602278A1 - Избирательные модуляторы андрогеновых рецепторов и способы их применения - Google Patents

Избирательные модуляторы андрогеновых рецепторов и способы их применения

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Publication number
EA200602278A1
EA200602278A1 EA200602278A EA200602278A EA200602278A1 EA 200602278 A1 EA200602278 A1 EA 200602278A1 EA 200602278 A EA200602278 A EA 200602278A EA 200602278 A EA200602278 A EA 200602278A EA 200602278 A1 EA200602278 A1 EA 200602278A1
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Eurasian Patent Office
Prior art keywords
bone
disorder
promoting
compounds
electional
Prior art date
Application number
EA200602278A
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English (en)
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EA011306B8 (ru
EA011306B1 (ru
Inventor
Джеймс Т. Далтон
Дуэйн Д. Миллер
Карен А. Веверка
Original Assignee
Юниверсити Оф Теннесси Рисерч Фаундейшн
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Publication date
Priority claimed from US10/861,923 external-priority patent/US8008348B2/en
Priority claimed from US10/863,524 external-priority patent/US20050038110A1/en
Priority claimed from US10/961,380 external-priority patent/US20060019931A1/en
Application filed by Юниверсити Оф Теннесси Рисерч Фаундейшн filed Critical Юниверсити Оф Теннесси Рисерч Фаундейшн
Publication of EA200602278A1 publication Critical patent/EA200602278A1/ru
Publication of EA011306B1 publication Critical patent/EA011306B1/ru
Publication of EA011306B8 publication Critical patent/EA011306B8/ru

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    • C07C255/58—Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton containing cyano groups and singly-bound nitrogen atoms, not being further bound to other hetero atoms, bound to the carbon skeleton
    • C07C255/60—Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton containing cyano groups and singly-bound nitrogen atoms, not being further bound to other hetero atoms, bound to the carbon skeleton at least one of the singly-bound nitrogen atoms being acylated
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Abstract

Изобретение относится к соединениям SARM и к их применению для лечения различных заболеваний или состояний у индивидуума, включая наряду с прочим истощающее мышцы заболевание и/или расстройство или связанное с костями заболевание и/или расстройство.
EA200602278A 2004-06-07 2005-06-07 Избирательные модуляторы андрогеновых рецепторов и способы их применения EA011306B8 (ru)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US10/861,923 US8008348B2 (en) 2001-12-06 2004-06-07 Treating muscle wasting with selective androgen receptor modulators
US10/863,524 US20050038110A1 (en) 2000-08-24 2004-06-09 Selective androgen receptor modulators and methods of use thereof
US10/961,380 US20060019931A1 (en) 2003-10-14 2004-10-12 Treating bone-related disorders with selective androgen receptor modulators
PCT/US2005/019788 WO2005120483A2 (en) 2004-06-07 2005-06-07 Selective androgen receptor modulators and methods of use thereof

Publications (3)

Publication Number Publication Date
EA200602278A1 true EA200602278A1 (ru) 2007-04-27
EA011306B1 EA011306B1 (ru) 2009-02-27
EA011306B8 EA011306B8 (ru) 2012-10-30

Family

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Family Applications (2)

Application Number Title Priority Date Filing Date
EA200802181A EA018699B1 (ru) 2004-06-07 2005-06-07 Применение соединения селективного модулятора андрогеновых рецепторов
EA200602278A EA011306B8 (ru) 2004-06-07 2005-06-07 Избирательные модуляторы андрогеновых рецепторов и способы их применения

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EA200802181A EA018699B1 (ru) 2004-06-07 2005-06-07 Применение соединения селективного модулятора андрогеновых рецепторов

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EP (2) EP2289872B1 (ru)
JP (2) JP4201818B2 (ru)
AT (1) ATE552235T1 (ru)
AU (1) AU2005251781C1 (ru)
BR (1) BRPI0511308B8 (ru)
CA (1) CA2543827C (ru)
CY (1) CY1120469T1 (ru)
DK (1) DK2289872T3 (ru)
EA (2) EA018699B1 (ru)
GE (1) GEP20094851B (ru)
IL (1) IL178716A (ru)
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US9884038B2 (en) 2004-06-07 2018-02-06 University Of Tennessee Research Foundation Selective androgen receptor modulator and methods of use thereof
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IL178716A0 (en) 2007-02-11
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EP1753417B1 (en) 2012-04-04
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WO2005120483A3 (en) 2006-08-03
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EP2289872A3 (en) 2013-01-09
CY1120469T1 (el) 2019-07-10
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AU2005251781B2 (en) 2007-09-13
EP1753417A2 (en) 2007-02-21
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IL178716A (en) 2014-04-30
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EA200802181A1 (ru) 2009-02-27
WO2005120483A2 (en) 2005-12-22
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ATE552235T1 (de) 2012-04-15
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