BRPI0511308A - moduladores seletivos receptores de androgênio e seus métodos de uso - Google Patents

moduladores seletivos receptores de androgênio e seus métodos de uso

Info

Publication number
BRPI0511308A
BRPI0511308A BRPI0511308-3A BRPI0511308A BRPI0511308A BR PI0511308 A BRPI0511308 A BR PI0511308A BR PI0511308 A BRPI0511308 A BR PI0511308A BR PI0511308 A BRPI0511308 A BR PI0511308A
Authority
BR
Brazil
Prior art keywords
bone
disorder
androgen receptor
selective androgen
promoting
Prior art date
Application number
BRPI0511308-3A
Other languages
English (en)
Inventor
James T Dalton
Duane D Miller
Karen A Veverka
Original Assignee
Univ Tennessee Res Foundation
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US10/861,923 external-priority patent/US8008348B2/en
Priority claimed from US10/863,524 external-priority patent/US20050038110A1/en
Priority claimed from US10/961,380 external-priority patent/US20060019931A1/en
Application filed by Univ Tennessee Res Foundation filed Critical Univ Tennessee Res Foundation
Publication of BRPI0511308A publication Critical patent/BRPI0511308A/pt
Publication of BRPI0511308B1 publication Critical patent/BRPI0511308B1/pt
Publication of BRPI0511308B8 publication Critical patent/BRPI0511308B8/pt

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    • C07C255/49—Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
    • C07C255/58—Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton containing cyano groups and singly-bound nitrogen atoms, not being further bound to other hetero atoms, bound to the carbon skeleton
    • C07C255/60—Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton containing cyano groups and singly-bound nitrogen atoms, not being further bound to other hetero atoms, bound to the carbon skeleton at least one of the singly-bound nitrogen atoms being acylated
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Abstract

MODULADORES SELETIVOS RECEPTORES DE ANDROGêNIO E SEUS MéTODOS DE USO Esta invenção provê compostos MSRA e seu uso no tratamento de uma variedade de doenças ou condições em um indivíduo, incluindo, entre elas, uma doença e/ou enfermidade de degeneração dos músculos ou uma doença e/ou enfermidade relacionada aos ossos.
BRPI0511308A 2004-06-07 2005-06-07 moduladores seletivos receptores de androgênio e seus métodos de uso BRPI0511308B8 (pt)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US10/861,923 2004-06-07
US10/861,923 US8008348B2 (en) 2001-12-06 2004-06-07 Treating muscle wasting with selective androgen receptor modulators
US10/863,524 US20050038110A1 (en) 2000-08-24 2004-06-09 Selective androgen receptor modulators and methods of use thereof
US10/863,524 2004-06-09
US10/961,380 US20060019931A1 (en) 2003-10-14 2004-10-12 Treating bone-related disorders with selective androgen receptor modulators
US10/961,380 2004-10-12
PCT/US2005/019788 WO2005120483A2 (en) 2004-06-07 2005-06-07 Selective androgen receptor modulators and methods of use thereof

Publications (3)

Publication Number Publication Date
BRPI0511308A true BRPI0511308A (pt) 2007-12-04
BRPI0511308B1 BRPI0511308B1 (pt) 2019-07-02
BRPI0511308B8 BRPI0511308B8 (pt) 2021-05-25

Family

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Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0511308A BRPI0511308B8 (pt) 2004-06-07 2005-06-07 moduladores seletivos receptores de androgênio e seus métodos de uso

Country Status (14)

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EP (2) EP2289872B1 (pt)
JP (2) JP4201818B2 (pt)
AT (1) ATE552235T1 (pt)
AU (1) AU2005251781C1 (pt)
BR (1) BRPI0511308B8 (pt)
CA (1) CA2543827C (pt)
CY (1) CY1120469T1 (pt)
DK (1) DK2289872T3 (pt)
EA (2) EA011306B8 (pt)
GE (1) GEP20094851B (pt)
IL (1) IL178716A (pt)
MX (1) MXPA06013958A (pt)
PL (2) PL2289872T3 (pt)
WO (1) WO2005120483A2 (pt)

Families Citing this family (34)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8853266B2 (en) * 2001-12-06 2014-10-07 University Of Tennessee Research Foundation Selective androgen receptor modulators for treating diabetes
US8309603B2 (en) 2004-06-07 2012-11-13 University Of Tennessee Research Foundation SARMs and method of use thereof
US9884038B2 (en) 2004-06-07 2018-02-06 University Of Tennessee Research Foundation Selective androgen receptor modulator and methods of use thereof
PL2289872T3 (pl) * 2004-06-07 2017-12-29 University Of Tennessee Research Foundation Medyczne zastosowania selektywnego modulatora receptora androgenowego
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