CY1109655T1 - Συνδεση των παραγωγων κινουκλιδινης στους μουσκαρινικους υποδοχεις μ3 - Google Patents
Συνδεση των παραγωγων κινουκλιδινης στους μουσκαρινικους υποδοχεις μ3Info
- Publication number
- CY1109655T1 CY1109655T1 CY20091101230T CY091101230T CY1109655T1 CY 1109655 T1 CY1109655 T1 CY 1109655T1 CY 20091101230 T CY20091101230 T CY 20091101230T CY 091101230 T CY091101230 T CY 091101230T CY 1109655 T1 CY1109655 T1 CY 1109655T1
- Authority
- CY
- Cyprus
- Prior art keywords
- kinoclidin
- muscaric
- producers
- receptors
- connection
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 abstract 3
- 102000007202 Muscarinic M3 Receptor Human genes 0.000 abstract 1
- 108010008405 Muscarinic M3 Receptor Proteins 0.000 abstract 1
- 230000001404 mediated effect Effects 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 239000000825 pharmaceutical preparation Substances 0.000 abstract 1
- 238000002360 preparation method Methods 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
- C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/02—Nasal agents, e.g. decongestants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/06—Antipsoriatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Abstract
Οι ενώσεις του χημικού τύπου (Ι), σε μορφή άλατος ή διιοντική μορφή στις οποίες οι R1, R2, R3 και R4 έχουν τις ερμηνείες που ορίστηκαν στην περιγραφή, είναι χρήσιμες στη θεραπεία καταστάσεων οι οποίες μεσολαβούνται από τον μουσκαρινικό υποδοχέα Μ3. Περιγράφονται επίσης τα φαρμακευτικά σκευάσματα τα οποία περιέχουν τις ενώσεις αυτές και μια διαδικασία για την παρασκευή των ενώσεων αυτών.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB0310232 | 2003-05-02 | ||
GB0324887A GB0324887D0 (en) | 2003-10-24 | 2003-10-24 | Organic compounds |
EP04730519A EP1631569B1 (en) | 2003-05-02 | 2004-04-30 | Quinuclidine derivatives binding to mucarinic m3 receptors |
Publications (1)
Publication Number | Publication Date |
---|---|
CY1109655T1 true CY1109655T1 (el) | 2014-08-13 |
Family
ID=33420896
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CY20091101230T CY1109655T1 (el) | 2003-05-02 | 2009-11-25 | Συνδεση των παραγωγων κινουκλιδινης στους μουσκαρινικους υποδοχεις μ3 |
Country Status (32)
Country | Link |
---|---|
US (2) | US20070060563A1 (el) |
EP (1) | EP1631569B1 (el) |
JP (1) | JP4416786B2 (el) |
KR (1) | KR100896544B1 (el) |
AR (1) | AR044134A1 (el) |
AT (1) | ATE440840T1 (el) |
AU (1) | AU2004234069B2 (el) |
BR (1) | BRPI0410238A (el) |
CA (1) | CA2523436C (el) |
CL (1) | CL2004000918A1 (el) |
CO (1) | CO5700782A2 (el) |
CY (1) | CY1109655T1 (el) |
DE (1) | DE602004022805D1 (el) |
DK (1) | DK1631569T3 (el) |
EC (1) | ECSP056134A (el) |
ES (1) | ES2331185T3 (el) |
HK (1) | HK1087704A1 (el) |
HR (1) | HRP20050933A2 (el) |
IL (1) | IL171591A (el) |
IS (1) | IS2746B (el) |
MA (1) | MA27775A1 (el) |
MX (1) | MXPA05011739A (el) |
MY (1) | MY142652A (el) |
NO (1) | NO20055688L (el) |
NZ (1) | NZ542995A (el) |
PE (1) | PE20050465A1 (el) |
PL (1) | PL1631569T3 (el) |
PT (1) | PT1631569E (el) |
RU (1) | RU2363700C2 (el) |
SI (1) | SI1631569T1 (el) |
TW (1) | TWI340139B (el) |
WO (1) | WO2004096800A2 (el) |
Families Citing this family (30)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ES2239546B1 (es) * | 2004-03-15 | 2006-12-01 | Almirall Prodesfarma, S.A. | Nuevos esteres de quinuclidina cuaternizados. |
GB0410712D0 (en) | 2004-05-13 | 2004-06-16 | Novartis Ag | Organic compounds |
GB0424284D0 (en) | 2004-11-02 | 2004-12-01 | Novartis Ag | Organic compounds |
GB0428416D0 (en) * | 2004-12-24 | 2005-02-02 | Novartis Ag | Organic compounds |
GB0601951D0 (en) | 2006-01-31 | 2006-03-15 | Novartis Ag | Organic compounds |
EP1900737A1 (en) * | 2006-08-31 | 2008-03-19 | Novartis AG | Polymorph of (R)-3-(2-hydroxy-2,2-diphenyl-acetoxy)-1-(isoxazol-3-ylcarbamoyl-methyl)-1-azonia-bicyclo-[2.2.2]octane bromide |
EP1894568A1 (en) * | 2006-08-31 | 2008-03-05 | Novartis AG | Pharmaceutical compositions for the treatment of inflammatory or obstructive airway diseases |
TW200825084A (en) * | 2006-11-14 | 2008-06-16 | Astrazeneca Ab | New compounds 521 |
CN101610813A (zh) * | 2006-12-19 | 2009-12-23 | 阿斯利康(瑞典)有限公司 | 作为毒蕈碱受体拮抗剂的奎核醇衍生物 |
EP1950196A1 (de) * | 2007-01-29 | 2008-07-30 | Boehringer Ingelheim Pharma GmbH & Co. KG | Verfahren zur Herstellung von Ammoniumhexafluorophosphaten |
PL2197841T3 (pl) * | 2007-09-07 | 2012-04-30 | Theravance Inc | Związki zawierające guanidynę przydatne jako antagoniści receptorów |
JP2011506477A (ja) | 2007-12-14 | 2011-03-03 | セラヴァンス, インコーポレーテッド | ムスカリン受容体拮抗薬として有用なアミジン含有化合物 |
KR20100113557A (ko) | 2008-01-11 | 2010-10-21 | 노파르티스 아게 | 키나제 억제제로서의 피리미딘 |
NZ589091A (en) * | 2008-05-13 | 2011-07-29 | Astrazeneca Ab | Quinuclidine derivatives as muscarinic m3 receptor antagonists |
GB0808709D0 (en) * | 2008-05-13 | 2008-06-18 | Astrazeneca Ab | New combination 295 |
RU2010147881A (ru) * | 2008-05-13 | 2012-06-20 | Астразенека Аб (Se) | ФАРМАЦЕВТИЧЕСКИЙ ПРОДУКТ, СОДЕРЖАЩИЙ АНТАГОНИСТ МУСКАРИНОВОГО РЕЦЕПТОРА И АГОНИСТ β2-АДРЕНОРЕЦЕПТОРА |
US20090326004A1 (en) | 2008-06-03 | 2009-12-31 | Ranbaxy Laboratories Limited | Muscarinic receptor antagonists |
WO2009153536A1 (en) * | 2008-06-17 | 2009-12-23 | Argenta Discovery Limited | 1-aza-bicyclo [2.2.2] octane derivatives useful as muscarinic receptor antagonists |
GB0811100D0 (en) * | 2008-06-17 | 2008-07-23 | Astrazeneca Ab | New combination |
CA2803459A1 (en) * | 2010-06-22 | 2011-12-29 | Chiesi Farmaceutici S.P.A. | Alkaloid aminoester derivatives and medicinal compositions thereof |
US8637516B2 (en) | 2010-09-09 | 2014-01-28 | Irm Llc | Compounds and compositions as TRK inhibitors |
WO2012034095A1 (en) | 2010-09-09 | 2012-03-15 | Irm Llc | Compounds and compositions as trk inhibitors |
PE20140378A1 (es) | 2011-02-25 | 2014-03-28 | Irm Llc | Compuestos y composiciones como inhibidores de la trk |
JP2011195593A (ja) * | 2011-06-30 | 2011-10-06 | Astrazeneca Ab | ムスカリンm3受容体アンタゴニストとしてのキヌクリジン誘導体 |
RU2628082C2 (ru) * | 2011-12-30 | 2017-08-14 | КЬЕЗИ ФАРМАЧЕУТИЧИ С.п.А. | Хинуклидиновые эфиры 1-азагетероциклилуксусной кислоты в качестве антимускариновых средств, способ их получения и их лекарственные композиции |
US9687488B2 (en) | 2012-05-03 | 2017-06-27 | St. Louis College Of Pharmacy | Compositions and methods for increasing neurotrophic peptides |
TWI647227B (zh) * | 2013-02-28 | 2019-01-11 | 日商安斯泰來製藥股份有限公司 | 2-醯胺噻唑衍生物或其鹽 |
CZ306791B6 (cs) | 2013-10-29 | 2017-07-12 | Zentiva, K.S. | Průmyslově využitelný způsob přípravy aklidinium bromidu o vysoké čistotě |
PT108370B (pt) * | 2015-03-30 | 2018-10-25 | Hovione Farm S A | Processo de preparação de brometo de aclidínio |
ES2897697T3 (es) | 2015-07-03 | 2022-03-02 | Novartis Ag | Inhalador adaptado para leer información almacenada en un medio de almacenamiento de datos de un recipiente |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB1219606A (en) * | 1968-07-15 | 1971-01-20 | Rech S Et D Applic Scient Soge | Quinuclidinol derivatives and preparation thereof |
DK534178A (da) * | 1977-12-16 | 1979-06-17 | Interx Research Corp | Anticholinerge midler med sektrtionshaemmende virkning |
ES2165768B1 (es) * | 1999-07-14 | 2003-04-01 | Almirall Prodesfarma Sa | Nuevos derivados de quinuclidina y composiciones farmaceuticas que los contienen. |
AU2001271027B2 (en) * | 2000-07-11 | 2005-07-07 | Msd K.K. | Ester derivatives |
DK1353919T3 (da) * | 2000-12-28 | 2006-11-20 | Almirall Prodesfarma Ag | Hidtil ukendte quinuclidinderivater og medicinale sammensætninger indeholdende samme |
IL162596A0 (en) * | 2001-12-20 | 2005-11-20 | S A L V A T Lab Sa | 1-Alkyl-1-azoniabicyclo Ä2.2.2Ü octane carbamate derivatives and their use as muscarinic receptor ntagonists |
GB0424284D0 (en) * | 2004-11-02 | 2004-12-01 | Novartis Ag | Organic compounds |
EP1900737A1 (en) * | 2006-08-31 | 2008-03-19 | Novartis AG | Polymorph of (R)-3-(2-hydroxy-2,2-diphenyl-acetoxy)-1-(isoxazol-3-ylcarbamoyl-methyl)-1-azonia-bicyclo-[2.2.2]octane bromide |
-
2004
- 2004-04-29 AR ARP040101468A patent/AR044134A1/es not_active Application Discontinuation
- 2004-04-30 ES ES04730519T patent/ES2331185T3/es not_active Expired - Lifetime
- 2004-04-30 WO PCT/EP2004/004605 patent/WO2004096800A2/en active Application Filing
- 2004-04-30 US US10/554,558 patent/US20070060563A1/en not_active Abandoned
- 2004-04-30 AU AU2004234069A patent/AU2004234069B2/en not_active Ceased
- 2004-04-30 EP EP04730519A patent/EP1631569B1/en not_active Expired - Lifetime
- 2004-04-30 CL CL200400918A patent/CL2004000918A1/es unknown
- 2004-04-30 TW TW093112339A patent/TWI340139B/zh not_active IP Right Cessation
- 2004-04-30 MX MXPA05011739A patent/MXPA05011739A/es active IP Right Grant
- 2004-04-30 KR KR1020057020776A patent/KR100896544B1/ko not_active IP Right Cessation
- 2004-04-30 PE PE2004000435A patent/PE20050465A1/es not_active Application Discontinuation
- 2004-04-30 CA CA2523436A patent/CA2523436C/en not_active Expired - Fee Related
- 2004-04-30 RU RU2005137360/04A patent/RU2363700C2/ru not_active IP Right Cessation
- 2004-04-30 DE DE602004022805T patent/DE602004022805D1/de not_active Expired - Lifetime
- 2004-04-30 NZ NZ542995A patent/NZ542995A/en not_active IP Right Cessation
- 2004-04-30 BR BRPI0410238-0A patent/BRPI0410238A/pt not_active IP Right Cessation
- 2004-04-30 AT AT04730519T patent/ATE440840T1/de active
- 2004-04-30 PT PT04730519T patent/PT1631569E/pt unknown
- 2004-04-30 JP JP2006505341A patent/JP4416786B2/ja not_active Expired - Fee Related
- 2004-04-30 MY MYPI20041637A patent/MY142652A/en unknown
- 2004-04-30 SI SI200431277T patent/SI1631569T1/sl unknown
- 2004-04-30 PL PL04730519T patent/PL1631569T3/pl unknown
- 2004-04-30 DK DK04730519T patent/DK1631569T3/da active
-
2005
- 2005-10-27 IL IL171591A patent/IL171591A/en not_active IP Right Cessation
- 2005-10-28 HR HR20050933A patent/HRP20050933A2/xx not_active Application Discontinuation
- 2005-11-01 EC EC2005006134A patent/ECSP056134A/es unknown
- 2005-11-03 CO CO05112195A patent/CO5700782A2/es not_active Application Discontinuation
- 2005-11-08 MA MA28583A patent/MA27775A1/fr unknown
- 2005-11-30 IS IS8158A patent/IS2746B/is unknown
- 2005-12-01 NO NO20055688A patent/NO20055688L/no not_active Application Discontinuation
-
2006
- 2006-07-17 HK HK06107974.9A patent/HK1087704A1/xx not_active IP Right Cessation
-
2009
- 2009-10-20 US US12/582,291 patent/US8168654B2/en not_active Expired - Fee Related
- 2009-11-25 CY CY20091101230T patent/CY1109655T1/el unknown
Also Published As
Similar Documents
Publication | Publication Date | Title |
---|---|---|
CY1109655T1 (el) | Συνδεση των παραγωγων κινουκλιδινης στους μουσκαρινικους υποδοχεις μ3 | |
CY1110952T1 (el) | Παραγωγα κινουκλιδινης και η χρηση αυτων ως μουσκαρινικοι ανταγωνιστες υποδοχεων μ3 | |
CY1108894T1 (el) | Νεα παραγωγα βενζιμιδαζολης | |
CY1105301T1 (el) | Αρυλοσυμπυκνωμενες αζαπολυκυκλικες ενωσεις | |
CY1107080T1 (el) | Υποκατεστημενες ινδολο-βασεις του mannich | |
CY1113450T1 (el) | Διαμινοπυριμιδινες ως ρ2χ3 και ρ2χ2/3 ανταγωνιστες | |
CY1107974T1 (el) | Παραγωγα κινολινης και κιναζολινης εχοντα συναφεια προς τους υποδοχεις τυπου 5ht1 | |
CY1108752T1 (el) | Παραγωγα πουρινης δρωντα ως αγωνιστες του α2α-υποδοχεα | |
CY1110332T1 (el) | Παραγωγα βενζιμιδαζολης, συνθεσεις που τα περιεχουν, παρασκευη αυτων και χρηση τους | |
CY1109015T1 (el) | Διφαινυλ ενωσεις χρησιμες ως ανταγωνιστες μουσκαρινικου υποδοχεα | |
SE0200920D0 (sv) | Novel compounds | |
TW200613243A (en) | Novel compounds | |
CY1111440T1 (el) | 5-χλωρο-3-(4-μεθανοσουλφονυλφαινυλ)-6'-μεθυλ-[2,3']διπυριδινυλ σε καθαρη κρυσταλλικη μορφη και διαδικασια για συνθεση | |
CY1111071T1 (el) | Φαρμακευτικες ενωσεις που περιεχουν τα παραγωγα αζετιδινης, τα νεα παραγωγα αζετιδινης και η παρασκευη τους | |
EA200600892A1 (ru) | Новые хинолиновые производные | |
SE0104140D0 (sv) | Novel Compounds | |
EA200701324A1 (ru) | Соединения пиридина для лечения заболеваний, опосредованных действием простагландина | |
SE0300480D0 (sv) | Novel compounds | |
CY1106486T1 (el) | Μεθοδος παρασκευης 2-(κινοξαλιν-5-υλσουλφονυλαμινο) βενζαμιδικων ενωσεων | |
CY1119407T1 (el) | Διαμορφωτες toy lxr | |
CY1107915T1 (el) | Τρικυκλικες σπιροπιπεριδινες ή σπιροπυρρολιδινες | |
ATE541839T1 (de) | Pyrrolidiniumderivate als m3-muskarinische rezeptoren | |
ES2368594T3 (es) | Derivados sustituidos de ciclohexilmetilo. | |
CY1105047T1 (el) | Ενωσεις πυριδοπυριμιδινονης, η μεθοδος παρασκευης τους και φαρμακευτικες συνθεσεις που τις περιεχουν | |
TW200626553A (en) | Novel compounds |