EA200600055A1 - Агонисты рецептора меланокортина 4 (мк4 ) и их применение - Google Patents

Агонисты рецептора меланокортина 4 (мк4 ) и их применение

Info

Publication number
EA200600055A1
EA200600055A1 EA200600055A EA200600055A EA200600055A1 EA 200600055 A1 EA200600055 A1 EA 200600055A1 EA 200600055 A EA200600055 A EA 200600055A EA 200600055 A EA200600055 A EA 200600055A EA 200600055 A1 EA200600055 A1 EA 200600055A1
Authority
EA
Eurasian Patent Office
Prior art keywords
receptor
agonists
melanocortin
application
obesity
Prior art date
Application number
EA200600055A
Other languages
English (en)
Russian (ru)
Inventor
Дэвид Бенджамин Флора
Марк Луис Хеймэн
ДжиЭнн Л. Хертел
Хансен Максвелл Хсиунг
Джон Филип Майер
Дэвид Ли Смайли
Лян Цзэн Янь
Ляньшань Чжан
Original Assignee
Эли Лилли Энд Компани
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Эли Лилли Энд Компани filed Critical Эли Лилли Энд Компани
Publication of EA200600055A1 publication Critical patent/EA200600055A1/ru

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/665—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans derived from pro-opiomelanocortin, pro-enkephalin or pro-dynorphin
    • C07K14/68—Melanocyte-stimulating hormone [MSH]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/12—Cyclic peptides, e.g. bacitracins; Polymyxins; Gramicidins S, C; Tyrocidins A, B or C
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/48—Drugs for disorders of the endocrine system of the pancreatic hormones

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Endocrinology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Diabetes (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Epidemiology (AREA)
  • Immunology (AREA)
  • Hematology (AREA)
  • Zoology (AREA)
  • Reproductive Health (AREA)
  • Molecular Biology (AREA)
  • Obesity (AREA)
  • Genetics & Genomics (AREA)
  • Toxicology (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Gynecology & Obstetrics (AREA)
  • Emergency Medicine (AREA)
  • Child & Adolescent Psychology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Peptides Or Proteins (AREA)
EA200600055A 2003-06-19 2004-06-17 Агонисты рецептора меланокортина 4 (мк4 ) и их применение EA200600055A1 (ru)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US47974003P 2003-06-19 2003-06-19
US55734704P 2004-03-29 2004-03-29
US57073704P 2004-05-13 2004-05-13
US57067604P 2004-05-13 2004-05-13
PCT/US2004/016625 WO2005000339A2 (en) 2003-06-19 2004-06-17 Melanocortin receptor 4(mc4) agonists and their uses

Publications (1)

Publication Number Publication Date
EA200600055A1 true EA200600055A1 (ru) 2006-08-25

Family

ID=33556652

Family Applications (1)

Application Number Title Priority Date Filing Date
EA200600055A EA200600055A1 (ru) 2003-06-19 2004-06-17 Агонисты рецептора меланокортина 4 (мк4 ) и их применение

Country Status (17)

Country Link
US (1) US20070105759A1 (https=)
EP (1) EP1644023A2 (https=)
JP (1) JP2006527773A (https=)
KR (1) KR20060014444A (https=)
AR (1) AR044824A1 (https=)
AU (1) AU2004251616A1 (https=)
BR (1) BRPI0410731A (https=)
CA (1) CA2530024A1 (https=)
CR (1) CR8159A (https=)
EA (1) EA200600055A1 (https=)
EC (1) ECSP056236A (https=)
IL (1) IL171931A0 (https=)
MX (1) MXPA05013951A (https=)
NO (1) NO20060259L (https=)
PE (1) PE20050284A1 (https=)
TW (1) TW200514791A (https=)
WO (1) WO2005000339A2 (https=)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2725150C2 (ru) * 2013-03-15 2020-06-30 Ритм Фармасьютикалз, Инк. Пептидные композиции
RU2844779C2 (ru) * 2013-03-15 2025-08-06 Ритм Фармасьютикалз, Инк. Фармацевтические композиции

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WO2006073772A1 (en) * 2005-01-05 2006-07-13 Eli Lilly And Company Polyethylene glycol linked mc4r or mc3r agonist peptides
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TWI364290B (en) * 2007-05-25 2012-05-21 Ipsen Pharma Sas Melanocortin receptor ligands modifled with hydantoin
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EP2766349B1 (de) 2011-03-08 2016-06-01 Sanofi Mit carbozyklen oder heterozyklen substituierte oxathiazinderivate, verfahren zu deren herstellung, diese verbindungen enthaltende arzneimittel und deren verwendung
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Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2725150C2 (ru) * 2013-03-15 2020-06-30 Ритм Фармасьютикалз, Инк. Пептидные композиции
RU2844779C2 (ru) * 2013-03-15 2025-08-06 Ритм Фармасьютикалз, Инк. Фармацевтические композиции

Also Published As

Publication number Publication date
PE20050284A1 (es) 2005-05-20
CR8159A (es) 2006-02-09
WO2005000339A2 (en) 2005-01-06
CA2530024A1 (en) 2005-01-06
EP1644023A2 (en) 2006-04-12
US20070105759A1 (en) 2007-05-10
AU2004251616A1 (en) 2005-01-06
IL171931A0 (en) 2006-04-10
KR20060014444A (ko) 2006-02-15
ECSP056236A (es) 2006-04-19
WO2005000339A3 (en) 2005-02-03
JP2006527773A (ja) 2006-12-07
NO20060259L (no) 2006-03-14
TW200514791A (en) 2005-05-01
WO2005000339A8 (en) 2005-04-21
AR044824A1 (es) 2005-10-05
BRPI0410731A (pt) 2006-06-20
MXPA05013951A (es) 2006-02-24

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