EA200201253A1 - Фунгицидные 5-фенил-замещенные 2-(цианоамино)пиримидины - Google Patents

Фунгицидные 5-фенил-замещенные 2-(цианоамино)пиримидины

Info

Publication number
EA200201253A1
EA200201253A1 EA200201253A EA200201253A EA200201253A1 EA 200201253 A1 EA200201253 A1 EA 200201253A1 EA 200201253 A EA200201253 A EA 200201253A EA 200201253 A EA200201253 A EA 200201253A EA 200201253 A1 EA200201253 A1 EA 200201253A1
Authority
EA
Eurasian Patent Office
Prior art keywords
substituted
alkyl
hydrogen
phenyl
compounds
Prior art date
Application number
EA200201253A
Other languages
English (en)
Other versions
EA005927B1 (ru
Inventor
Клаус-Юрген Пес
Вальдемар Пфренгле
Гейвин Хеффернан
Original Assignee
Басф Акциенгезельшафт
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Басф Акциенгезельшафт filed Critical Басф Акциенгезельшафт
Publication of EA200201253A1 publication Critical patent/EA200201253A1/ru
Publication of EA005927B1 publication Critical patent/EA005927B1/ru

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48—Two nitrogen atoms
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/40—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having a double or triple bond to nitrogen, e.g. cyanates, cyanamides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32—One oxygen, sulfur or nitrogen atom
    • C07D239/38—One sulfur atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

Пиримидины формулы (I)в которой Rозначает водород или алкил, галоалкил, алкенил, алкинил, алкадиенил, алкокси, циклоалкил, фенил, 5- или 6-членный гетероарил или 5- или 6-членный гетероциклил, содержащие 1-4 атома азота или 1-3 атома азота и один атом серы или кислорода, или триалкилсилил, формил или алкоксикарбонил,причем группы Rне замещены или замещены указанными в описании заместителями;Rозначает фенил, циклоалкил или 5- или 6-членный гетероарил, содержащий 1-4 атома азота или 1-3 атома азота и один атом серы или кислорода, которые не замещены или замещены;Rозначает водород, галоген или алкил, алкокси, алкилтио, алкиламино или диалкиламино, которые не замещены или замещены;Rозначает водород или алкил, алкенил или алкинил, которые не замещены или замещены, иХ означает кислород, серу, группу NRили простую связь, причем Rозначает водород или алкил; илиRи Rвместе с размещенным между ними атомом азота образуют гетероцикл;способы и промежуточные соединения для получения данных соединений, композиции, содержащие данные соединения, и применение данных соединений для борьбы с фитопатогенными грибами.Международная заявка была опубликована вместе с отчетом о международном поиске.
EA200201253A 2000-06-13 2001-06-11 Фунгицидные 5-фенил-замещенные 2-(цианоамино)пиримидины EA005927B1 (ru)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US21126200P 2000-06-13 2000-06-13
US23163200P 2000-09-11 2000-09-11
PCT/EP2001/006565 WO2001096314A1 (en) 2000-06-13 2001-06-11 Fungicidal 5-phenyl substituted 2-(cyanoamino) pyrimidines

Publications (2)

Publication Number Publication Date
EA200201253A1 true EA200201253A1 (ru) 2003-04-24
EA005927B1 EA005927B1 (ru) 2005-08-25

Family

ID=26905995

Family Applications (1)

Application Number Title Priority Date Filing Date
EA200201253A EA005927B1 (ru) 2000-06-13 2001-06-11 Фунгицидные 5-фенил-замещенные 2-(цианоамино)пиримидины

Country Status (19)

Country Link
US (5) US6632821B2 (ru)
EP (1) EP1289963B1 (ru)
JP (1) JP2004503542A (ru)
KR (1) KR20030011894A (ru)
CN (1) CN1279027C (ru)
AT (1) ATE303367T1 (ru)
AU (1) AU778913B2 (ru)
BR (1) BR0111594A (ru)
CA (1) CA2412010A1 (ru)
CZ (1) CZ20024041A3 (ru)
DE (1) DE60113104D1 (ru)
EA (1) EA005927B1 (ru)
ES (1) ES2246330T3 (ru)
HU (1) HUP0300649A3 (ru)
IL (2) IL153016A0 (ru)
MX (1) MXPA02012073A (ru)
PL (1) PL362551A1 (ru)
SK (1) SK17452002A3 (ru)
WO (1) WO2001096314A1 (ru)

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JP2006518717A (ja) * 2003-02-06 2006-08-17 ビーエーエスエフ　アクチェンゲゼルシャフト ピリミジン類、製造およびそれの使用
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ATE432077T1 (de) 2003-09-24 2009-06-15 Wyeth Corp 5-arylpyrimidine als anti-krebs-mittel
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EP2326627A1 (en) * 2008-08-20 2011-06-01 Schering Corporation Substituted pyridine and pyrimidine derivatives and their use in treating viral infections
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Also Published As

Publication number Publication date
KR20030011894A (ko) 2003-02-11
MXPA02012073A (es) 2003-04-25
US20050282828A1 (en) 2005-12-22
HUP0300649A3 (en) 2003-10-28
CA2412010A1 (en) 2001-12-20
US6943252B2 (en) 2005-09-13
US20070208037A1 (en) 2007-09-06
HUP0300649A2 (hu) 2003-07-28
BR0111594A (pt) 2003-04-15
US20050282847A1 (en) 2005-12-22
JP2004503542A (ja) 2004-02-05
IL153016A0 (en) 2003-06-24
US20030088096A1 (en) 2003-05-08
EA005927B1 (ru) 2005-08-25
EP1289963B1 (en) 2005-08-31
DE60113104D1 (de) 2005-10-06
ES2246330T3 (es) 2006-02-16
CN1279027C (zh) 2006-10-11
AU7056401A (en) 2001-12-24
EP1289963A1 (en) 2003-03-12
CZ20024041A3 (cs) 2003-04-16
US6632821B2 (en) 2003-10-14
AU778913B2 (en) 2004-12-23
US20040147744A1 (en) 2004-07-29
US7230104B2 (en) 2007-06-12
ATE303367T1 (de) 2005-09-15
IL176276A0 (en) 2006-10-05
CN1443174A (zh) 2003-09-17
PL362551A1 (en) 2004-11-02
WO2001096314A1 (en) 2001-12-20
SK17452002A3 (sk) 2003-06-03

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