HUP0300649A2 - Fungicid hatású 5-fenil-szubsztituált 2-(ciano-amino)-pirimidin-származékok, előállításuk és alkalmazásuk - Google Patents

Fungicid hatású 5-fenil-szubsztituált 2-(ciano-amino)-pirimidin-származékok, előállításuk és alkalmazásuk

Info

Publication number
HUP0300649A2
HUP0300649A2 HU0300649A HUP0300649A HUP0300649A2 HU P0300649 A2 HUP0300649 A2 HU P0300649A2 HU 0300649 A HU0300649 A HU 0300649A HU P0300649 A HUP0300649 A HU P0300649A HU P0300649 A2 HUP0300649 A2 HU P0300649A2
Authority
HU
Hungary
Prior art keywords
group
atom
optionally substituted
hydrogen atom
sulfur
Prior art date
Application number
HU0300649A
Other languages
English (en)
Inventor
Gavin Heffernan
Klaus-Jürgen Pees
Waldemar Pfrengle
Original Assignee
Basf Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Basf Ag filed Critical Basf Ag
Publication of HUP0300649A2 publication Critical patent/HUP0300649A2/hu
Publication of HUP0300649A3 publication Critical patent/HUP0300649A3/hu

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48—Two nitrogen atoms
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/40—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having a double or triple bond to nitrogen, e.g. cyanates, cyanamides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32—One oxygen, sulfur or nitrogen atom
    • C07D239/38—One sulfur atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

A találmány tárgyát az általános képletű pirimidinszármazékok - aholR1 hidrogénatom vagy adott esetben szubsztituált alkil-, halogén-alkil-, alkenil-, alkinil-, alkadienil-, alkoxi-, cikloalkil-,fenilcsoport vagy 1-4 vagy 1-3 nitrogénatomot és 1 kén- vagyoxigénatomot tartalmazó 5- vagy 6-tagú heteroaril-csoport vagy 5- vagy6-tagú heterociklusos vagy trialkil-szilil-, formil- vagy alkoxi-karbonil-csoport; R2 adott esetben szubsztituált fenil-, cikloalkil-,vagy l-4 vagy 1-3 nitrogénatomot és 1 kén- vagy oxigénatomottartalmazó 5- vagy 6-tagú heteroarilcsoport; R3 hidrogén-, halogénatomvagy adott esetben szubsztituált alkil-, alkoxi-, alkil-tio- vagyalkil-amino-csoport; R4 hidrogénatom vagy adott esetben szubsztituáltalkil-, alkenil- vagy alkinilcsoport; és X oxigénatom, kénatom, =N-R5általános képletű csoport vagy egyes kötés, ahol R5 hidrogénatom vagyalkilcsoport; vagy R1 és R5 egy közbülső nitrogénatommal együtt egyheterociklusos gyűrűt képez - és előállításuk, ezeket tartalmazókészítmények és káros gombák elleni alkalmazásuk képezik. Ó
HU0300649A 2000-06-13 2001-06-11 Fungicidal 5-phenyl substituted 2-(cyanoamino)pyrimidines, preparation and use thereof HUP0300649A3 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US21126200P 2000-06-13 2000-06-13
US23163200P 2000-09-11 2000-09-11
PCT/EP2001/006565 WO2001096314A1 (en) 2000-06-13 2001-06-11 Fungicidal 5-phenyl substituted 2-(cyanoamino) pyrimidines

Publications (2)

Publication Number Publication Date
HUP0300649A2 true HUP0300649A2 (hu) 2003-07-28
HUP0300649A3 HUP0300649A3 (en) 2003-10-28

Family

ID=26905995

Family Applications (1)

Application Number Title Priority Date Filing Date
HU0300649A HUP0300649A3 (en) 2000-06-13 2001-06-11 Fungicidal 5-phenyl substituted 2-(cyanoamino)pyrimidines, preparation and use thereof

Country Status (19)

Country Link
US (5) US6632821B2 (hu)
EP (1) EP1289963B1 (hu)
JP (1) JP2004503542A (hu)
KR (1) KR20030011894A (hu)
CN (1) CN1279027C (hu)
AT (1) ATE303367T1 (hu)
AU (1) AU778913B2 (hu)
BR (1) BR0111594A (hu)
CA (1) CA2412010A1 (hu)
CZ (1) CZ20024041A3 (hu)
DE (1) DE60113104D1 (hu)
EA (1) EA005927B1 (hu)
ES (1) ES2246330T3 (hu)
HU (1) HUP0300649A3 (hu)
IL (2) IL153016A0 (hu)
MX (1) MXPA02012073A (hu)
PL (1) PL362551A1 (hu)
SK (1) SK17452002A3 (hu)
WO (1) WO2001096314A1 (hu)

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GB0126914D0 (en) * 2001-11-08 2002-01-02 Syngenta Ltd Fungicides
CA2467683C (en) * 2001-11-19 2011-09-27 Basf Aktiengesellschaft 5-phenylpyrimidines, agents comprising the same, method for production and use thereof
CN100357297C (zh) * 2003-02-06 2007-12-26 巴斯福股份公司 嘧啶、其生产方法及其用途
CN100445269C (zh) * 2003-04-04 2008-12-24 巴斯福股份公司 2-取代的嘧啶
BRPI0410482A (pt) * 2003-05-20 2006-06-13 Basf Ag composto, processo para preparar o mesmo, agente adequado para combater fungos nocivos, e, processo para combater fungos nocivos fitopatogênicos
WO2005012261A1 (de) 2003-07-24 2005-02-10 Basf Aktiengesellschaft 2-substituierte pyrimidine
DE602004021269D1 (de) 2003-09-24 2009-07-09 Wyeth Corp 5-arylpyrimidine als anti-krebs-mittel
DE10360370A1 (de) * 2003-12-22 2005-07-14 Bayer Cropscience Ag Triazolopyrimidine
DE102004003428A1 (de) * 2004-01-23 2005-08-11 Boehringer Ingelheim Pharma Gmbh & Co. Kg Neue langwirksame Beta-2-Agonisten, und deren Verwendung als Arzneimittel
DE102004003493A1 (de) * 2004-01-23 2005-08-11 Bayer Cropscience Ag 5-Phenylpyrimidine
JP2008513401A (ja) * 2004-09-17 2008-05-01 ビーエーエスエフ ソシエタス・ヨーロピア 植物の線虫病に対処するための２−置換ピリミジンの使用
US20080176744A1 (en) * 2005-03-10 2008-07-24 Basf Aktiengesellschaft Use of 4-Aminopyrimidines for Controlling Harmful Fungi, Novel 4-Aminopyrimidines, Processes for Their Preparation and Compositions Comprising Them
GB0512844D0 (en) * 2005-06-23 2005-08-03 Novartis Ag Organic compounds
CA2645779A1 (en) * 2006-03-27 2007-10-04 Basf Se Substituted 5-hetaryl-4-aminopyrimidines
WO2007113322A2 (de) * 2006-04-05 2007-10-11 Basf Se Substituierte 5-hetarylpyrimidine zur bekämpfung von pflanzenschädigenden pilzen und von krebserkrankungen
CL2007002231A1 (es) * 2006-08-02 2008-04-11 Basf Ag Uso de compuestos derivados de 5-(het) arilpirimidina para combatir hongos daninos; compuestos derivados de 5-(het) arilpirimidina; agente fungicida; y agente farmaceutico.
DE102007012908A1 (de) 2007-03-19 2008-09-25 Momentive Performance Materials Gmbh Neue Polyamid-Polysiloxan-Verbindungen
TWI409265B (zh) * 2008-08-20 2013-09-21 Merck Sharp & Dohme 經取代之吡啶及嘧啶衍生物及彼等於治療病毒感染之用途
AU2013361540B2 (en) * 2012-12-19 2017-02-02 Dow Agrosciences Llc Pesticidal compositions and processes related thereto
CN104892528A (zh) * 2014-12-10 2015-09-09 上海工程技术大学 一种2-硫代巴比妥酸衍生物的制备方法

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Also Published As

Publication number Publication date
CZ20024041A3 (cs) 2003-04-16
US7230104B2 (en) 2007-06-12
DE60113104D1 (de) 2005-10-06
US20050282828A1 (en) 2005-12-22
ATE303367T1 (de) 2005-09-15
CN1443174A (zh) 2003-09-17
WO2001096314A1 (en) 2001-12-20
MXPA02012073A (es) 2003-04-25
AU778913B2 (en) 2004-12-23
EA005927B1 (ru) 2005-08-25
CN1279027C (zh) 2006-10-11
IL153016A0 (en) 2003-06-24
EP1289963A1 (en) 2003-03-12
US20070208037A1 (en) 2007-09-06
SK17452002A3 (sk) 2003-06-03
EA200201253A1 (ru) 2003-04-24
BR0111594A (pt) 2003-04-15
JP2004503542A (ja) 2004-02-05
ES2246330T3 (es) 2006-02-16
IL176276A0 (en) 2006-10-05
HUP0300649A3 (en) 2003-10-28
AU7056401A (en) 2001-12-24
KR20030011894A (ko) 2003-02-11
US20050282847A1 (en) 2005-12-22
US20040147744A1 (en) 2004-07-29
US6943252B2 (en) 2005-09-13
EP1289963B1 (en) 2005-08-31
PL362551A1 (en) 2004-11-02
US6632821B2 (en) 2003-10-14
CA2412010A1 (en) 2001-12-20
US20030088096A1 (en) 2003-05-08

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