EA200000689A1 - Способ получения пароксетин гидрохлорида - Google Patents

Способ получения пароксетин гидрохлорида

Info

Publication number
EA200000689A1
EA200000689A1 EA200000689A EA200000689A EA200000689A1 EA 200000689 A1 EA200000689 A1 EA 200000689A1 EA 200000689 A EA200000689 A EA 200000689A EA 200000689 A EA200000689 A EA 200000689A EA 200000689 A1 EA200000689 A1 EA 200000689A1
Authority
EA
Eurasian Patent Office
Prior art keywords
hydrochloride
paroxethine
obtaining
propan
paroxetine hydrochloride
Prior art date
Application number
EA200000689A
Other languages
English (en)
Russian (ru)
Inventor
Нил Уорд
Алан Дэвид Джоунс
Original Assignee
Смитклайн Бичам Плс
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Смитклайн Бичам Плс filed Critical Смитклайн Бичам Плс
Publication of EA200000689A1 publication Critical patent/EA200000689A1/ru

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
EA200000689A 1997-12-19 1998-12-18 Способ получения пароксетин гидрохлорида EA200000689A1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB9726907.0A GB9726907D0 (en) 1997-12-19 1997-12-19 Novel compounds
PCT/GB1998/003836 WO1999032484A1 (en) 1997-12-19 1998-12-18 Process for the preparation of paroxetine hydrochloride

Publications (1)

Publication Number Publication Date
EA200000689A1 true EA200000689A1 (ru) 2000-12-25

Family

ID=10823933

Family Applications (1)

Application Number Title Priority Date Filing Date
EA200000689A EA200000689A1 (ru) 1997-12-19 1998-12-18 Способ получения пароксетин гидрохлорида

Country Status (20)

Country Link
EP (1) EP1042318A1 (no)
JP (1) JP2001526288A (no)
KR (1) KR20010033317A (no)
CN (1) CN1281448A (no)
AP (1) AP2000001836A0 (no)
AU (1) AU1769899A (no)
BG (1) BG104604A (no)
BR (1) BR9813638A (no)
CA (1) CA2315066A1 (no)
EA (1) EA200000689A1 (no)
GB (1) GB9726907D0 (no)
HU (1) HUP0004503A3 (no)
ID (1) ID24733A (no)
IL (1) IL136590A0 (no)
NO (1) NO20003145L (no)
OA (1) OA11635A (no)
PL (1) PL341358A1 (no)
SK (1) SK9242000A3 (no)
TR (1) TR200001933T2 (no)
WO (1) WO1999032484A1 (no)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9919001D0 (en) * 1999-08-12 1999-10-13 Smithkline Beecham Plc Novel process
GB9923439D0 (en) * 1999-10-04 1999-12-08 Smithkline Beecham Plc Novel process
NL1017421C2 (nl) 2001-02-21 2002-01-15 Synthon Bv Werkwijze voor het vervaardigen van paroxetine.
JP2005524656A (ja) * 2002-02-22 2005-08-18 テバ ファーマシューティカル インダストリーズ リミティド 新規中間物質を用いるパロキセチンの調製
KR100672184B1 (ko) 2004-09-21 2007-01-19 주식회사종근당 파록세틴의 콜린산 또는 콜린산 유도체 염

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0223403B1 (en) * 1985-10-25 1993-08-04 Beecham Group Plc Piperidine derivative, its preparation, and its use as medicament
SK283608B6 (sk) * 1995-02-06 2003-10-07 Smithkline Beecham Plc Bezvodý hydrochlorid paroxetínu, spôsob jeho výroby a použitie
CA2187128A1 (en) * 1996-10-04 1997-06-26 K. S. Keshava Murthy New and useful polymorph of anhydrous paroxetine hydrochloride

Also Published As

Publication number Publication date
HUP0004503A2 (hu) 2002-03-28
EP1042318A1 (en) 2000-10-11
ID24733A (id) 2000-08-03
SK9242000A3 (en) 2001-01-18
OA11635A (en) 2004-11-22
AU1769899A (en) 1999-07-12
BR9813638A (pt) 2000-10-17
GB9726907D0 (en) 1998-02-18
IL136590A0 (en) 2001-06-14
WO1999032484A1 (en) 1999-07-01
KR20010033317A (ko) 2001-04-25
CN1281448A (zh) 2001-01-24
TR200001933T2 (tr) 2000-12-21
AP2000001836A0 (en) 2000-06-30
CA2315066A1 (en) 1999-07-01
HUP0004503A3 (en) 2002-04-29
NO20003145D0 (no) 2000-06-16
JP2001526288A (ja) 2001-12-18
NO20003145L (no) 2000-06-16
PL341358A1 (en) 2001-04-09
BG104604A (en) 2001-03-30

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