EA200000689A1 - Способ получения пароксетин гидрохлорида - Google Patents
Способ получения пароксетин гидрохлоридаInfo
- Publication number
- EA200000689A1 EA200000689A1 EA200000689A EA200000689A EA200000689A1 EA 200000689 A1 EA200000689 A1 EA 200000689A1 EA 200000689 A EA200000689 A EA 200000689A EA 200000689 A EA200000689 A EA 200000689A EA 200000689 A1 EA200000689 A1 EA 200000689A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- hydrochloride
- paroxethine
- obtaining
- propan
- paroxetine hydrochloride
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
(57) Настоящее изобретение раскрывает способ получения пропан-2-ол сольвата пароксетин гидрохлорида, включающий образование раствора пароксетин гидрохлорида в смеси пропан-2-ола и эффективного сорастворителя и кристаллизацию пропан-2-ол сольвата пароксетин гидрохлорида из раствора.Международная заявка была опубликована вместе с отчетом о международном поиске.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GBGB9726907.0A GB9726907D0 (en) | 1997-12-19 | 1997-12-19 | Novel compounds |
PCT/GB1998/003836 WO1999032484A1 (en) | 1997-12-19 | 1998-12-18 | Process for the preparation of paroxetine hydrochloride |
Publications (1)
Publication Number | Publication Date |
---|---|
EA200000689A1 true EA200000689A1 (ru) | 2000-12-25 |
Family
ID=10823933
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA200000689A EA200000689A1 (ru) | 1997-12-19 | 1998-12-18 | Способ получения пароксетин гидрохлорида |
Country Status (20)
Country | Link |
---|---|
EP (1) | EP1042318A1 (ru) |
JP (1) | JP2001526288A (ru) |
KR (1) | KR20010033317A (ru) |
CN (1) | CN1281448A (ru) |
AP (1) | AP2000001836A0 (ru) |
AU (1) | AU1769899A (ru) |
BG (1) | BG104604A (ru) |
BR (1) | BR9813638A (ru) |
CA (1) | CA2315066A1 (ru) |
EA (1) | EA200000689A1 (ru) |
GB (1) | GB9726907D0 (ru) |
HU (1) | HUP0004503A3 (ru) |
ID (1) | ID24733A (ru) |
IL (1) | IL136590A0 (ru) |
NO (1) | NO20003145D0 (ru) |
OA (1) | OA11635A (ru) |
PL (1) | PL341358A1 (ru) |
SK (1) | SK9242000A3 (ru) |
TR (1) | TR200001933T2 (ru) |
WO (1) | WO1999032484A1 (ru) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB9919001D0 (en) * | 1999-08-12 | 1999-10-13 | Smithkline Beecham Plc | Novel process |
GB9923439D0 (en) * | 1999-10-04 | 1999-12-08 | Smithkline Beecham Plc | Novel process |
NL1017421C2 (nl) | 2001-02-21 | 2002-01-15 | Synthon Bv | Werkwijze voor het vervaardigen van paroxetine. |
JP2005524656A (ja) * | 2002-02-22 | 2005-08-18 | テバ ファーマシューティカル インダストリーズ リミティド | 新規中間物質を用いるパロキセチンの調製 |
KR100672184B1 (ko) | 2004-09-21 | 2007-01-19 | 주식회사종근당 | 파록세틴의 콜린산 또는 콜린산 유도체 염 |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0223403B1 (en) * | 1985-10-25 | 1993-08-04 | Beecham Group Plc | Piperidine derivative, its preparation, and its use as medicament |
SK283608B6 (sk) * | 1995-02-06 | 2003-10-07 | Smithkline Beecham Plc | Bezvodý hydrochlorid paroxetínu, spôsob jeho výroby a použitie |
CA2187128A1 (en) * | 1996-10-04 | 1997-06-26 | K. S. Keshava Murthy | New and useful polymorph of anhydrous paroxetine hydrochloride |
-
1997
- 1997-12-19 GB GBGB9726907.0A patent/GB9726907D0/en not_active Ceased
-
1998
- 1998-12-18 KR KR1020007006764A patent/KR20010033317A/ko not_active Application Discontinuation
- 1998-12-18 EA EA200000689A patent/EA200000689A1/ru unknown
- 1998-12-18 TR TR2000/01933T patent/TR200001933T2/xx unknown
- 1998-12-18 SK SK924-2000A patent/SK9242000A3/sk unknown
- 1998-12-18 WO PCT/GB1998/003836 patent/WO1999032484A1/en not_active Application Discontinuation
- 1998-12-18 AP APAP/P/2000/001836A patent/AP2000001836A0/en unknown
- 1998-12-18 OA OA1200000182A patent/OA11635A/en unknown
- 1998-12-18 CN CN98811920A patent/CN1281448A/zh active Pending
- 1998-12-18 AU AU17698/99A patent/AU1769899A/en not_active Abandoned
- 1998-12-18 PL PL98341358A patent/PL341358A1/xx unknown
- 1998-12-18 JP JP2000525421A patent/JP2001526288A/ja active Pending
- 1998-12-18 CA CA002315066A patent/CA2315066A1/en not_active Abandoned
- 1998-12-18 IL IL13659098A patent/IL136590A0/xx unknown
- 1998-12-18 HU HU0004503A patent/HUP0004503A3/hu unknown
- 1998-12-18 ID IDW20001158A patent/ID24733A/id unknown
- 1998-12-18 BR BR9813638-0A patent/BR9813638A/pt not_active Application Discontinuation
- 1998-12-18 EP EP98962563A patent/EP1042318A1/en not_active Withdrawn
-
2000
- 2000-06-16 NO NO20003145A patent/NO20003145D0/no not_active Application Discontinuation
- 2000-07-13 BG BG104604A patent/BG104604A/xx unknown
Also Published As
Publication number | Publication date |
---|---|
OA11635A (en) | 2004-11-22 |
BR9813638A (pt) | 2000-10-17 |
AP2000001836A0 (en) | 2000-06-30 |
TR200001933T2 (tr) | 2000-12-21 |
HUP0004503A3 (en) | 2002-04-29 |
NO20003145L (no) | 2000-06-16 |
AU1769899A (en) | 1999-07-12 |
EP1042318A1 (en) | 2000-10-11 |
ID24733A (id) | 2000-08-03 |
SK9242000A3 (en) | 2001-01-18 |
KR20010033317A (ko) | 2001-04-25 |
PL341358A1 (en) | 2001-04-09 |
BG104604A (en) | 2001-03-30 |
IL136590A0 (en) | 2001-06-14 |
NO20003145D0 (no) | 2000-06-16 |
JP2001526288A (ja) | 2001-12-18 |
CN1281448A (zh) | 2001-01-24 |
CA2315066A1 (en) | 1999-07-01 |
HUP0004503A2 (hu) | 2002-03-28 |
GB9726907D0 (en) | 1998-02-18 |
WO1999032484A1 (en) | 1999-07-01 |
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