EA200300388A1 - 1-аминоалкилциклогексаны в качестве трипаноцидных агентов - Google Patents
1-аминоалкилциклогексаны в качестве трипаноцидных агентовInfo
- Publication number
- EA200300388A1 EA200300388A1 EA200300388A EA200300388A EA200300388A1 EA 200300388 A1 EA200300388 A1 EA 200300388A1 EA 200300388 A EA200300388 A EA 200300388A EA 200300388 A EA200300388 A EA 200300388A EA 200300388 A1 EA200300388 A1 EA 200300388A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- agents
- tripanocidal
- cyclohexanes
- aminoalkyl
- methods
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/16—Amides, e.g. hydroxamic acids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
Landscapes
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Tropical Medicine & Parasitology (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Некоторые 1-аминоалкилциклогексаны являются противотрипаносомозными агентами и трипаноцидами. Раскрыты их фармацевтические композиции, используемые для этой цели, и способы их получения, а также способы лечения с их помощью трипаносомоза.Международная заявка была опубликована вместе с отчетом о международном поиске.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US09/664,629 US6602862B1 (en) | 2000-09-19 | 2000-09-19 | 1-Amino-alkylcyclohexanes as trypanocidal agents |
PCT/EP2001/010731 WO2002024186A1 (en) | 2000-09-19 | 2001-09-14 | 1-amino-alkylcyclohexanes as trypanocidal agents |
Publications (2)
Publication Number | Publication Date |
---|---|
EA200300388A1 true EA200300388A1 (ru) | 2003-08-28 |
EA005499B1 EA005499B1 (ru) | 2005-02-24 |
Family
ID=24666769
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA200300388A EA005499B1 (ru) | 2000-09-19 | 2001-09-14 | 1-аминоалкилциклогексаны в качестве трипаноцидных агентов |
Country Status (25)
Country | Link |
---|---|
US (1) | US6602862B1 (ru) |
EP (1) | EP1318800B1 (ru) |
JP (1) | JP2004509144A (ru) |
KR (1) | KR100570373B1 (ru) |
CN (1) | CN1283239C (ru) |
AR (1) | AR030750A1 (ru) |
AT (1) | ATE287708T1 (ru) |
AU (2) | AU2001287740B2 (ru) |
CA (1) | CA2420056C (ru) |
CZ (1) | CZ2003776A3 (ru) |
DE (1) | DE60108650T2 (ru) |
EA (1) | EA005499B1 (ru) |
ES (1) | ES2233679T3 (ru) |
GE (1) | GEP20053480B (ru) |
HK (1) | HK1058151A1 (ru) |
HU (1) | HUP0302497A3 (ru) |
IL (2) | IL154867A0 (ru) |
MX (1) | MXPA03001790A (ru) |
NO (1) | NO20031239L (ru) |
PL (1) | PL361428A1 (ru) |
PT (1) | PT1318800E (ru) |
TW (1) | TWI297605B (ru) |
UA (1) | UA73609C2 (ru) |
WO (1) | WO2002024186A1 (ru) |
ZA (1) | ZA200107649B (ru) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6444702B1 (en) | 2000-02-22 | 2002-09-03 | Neuromolecular, Inc. | Aminoadamantane derivatives as therapeutic agents |
BRPI1012669A2 (pt) * | 2009-06-29 | 2016-04-05 | Merz Pharma Gmbh & Co Kgaa | metodo de preparacao de 3,3,5,5-tetrametliciclohexanona, método de preparção de 1-amino-1,3,3,5,5,-pentametilciclohexano ou um sal farmaceuticamente aceitável do mesmo e composto |
CN102241678B (zh) | 2011-04-26 | 2014-10-29 | 辽宁利锋科技开发有限公司 | 含有脂环结构化合物的抗肿瘤作用与应用 |
PL2826856T3 (pl) * | 2013-07-16 | 2016-06-30 | Sia Latima | Genetycznie stabilny onkolityczny wirus RNA, sposób jego wytwarzania i zastosowanie |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU673736B2 (en) | 1993-04-13 | 1996-11-21 | Novartis Ag | Ornithine decarboxylase inhibiting cyclic aminooxy compounds |
US6071966A (en) * | 1997-06-30 | 2000-06-06 | Merz + Co. Gmbh & Co. | 1-amino-alkylcyclohexane NMDA receptor antagonists |
TW593225B (en) | 1997-06-30 | 2004-06-21 | Merz Pharma Gmbh & Co Kgaa | 1-amino-alkylcyclohexane NMDA receptor antagonists |
US6093743A (en) * | 1998-06-23 | 2000-07-25 | Medinox Inc. | Therapeutic methods employing disulfide derivatives of dithiocarbamates and compositions useful therefor |
-
2000
- 2000-09-19 US US09/664,629 patent/US6602862B1/en not_active Expired - Fee Related
-
2001
- 2001-09-04 TW TW090121900A patent/TWI297605B/zh active
- 2001-09-14 JP JP2002528257A patent/JP2004509144A/ja active Pending
- 2001-09-14 AT AT01967349T patent/ATE287708T1/de not_active IP Right Cessation
- 2001-09-14 IL IL15486701A patent/IL154867A0/xx unknown
- 2001-09-14 GE GE5127A patent/GEP20053480B/en unknown
- 2001-09-14 AU AU2001287740A patent/AU2001287740B2/en not_active Ceased
- 2001-09-14 CZ CZ2003776A patent/CZ2003776A3/cs unknown
- 2001-09-14 CA CA002420056A patent/CA2420056C/en not_active Expired - Fee Related
- 2001-09-14 ES ES01967349T patent/ES2233679T3/es not_active Expired - Lifetime
- 2001-09-14 AU AU8774001A patent/AU8774001A/xx active Pending
- 2001-09-14 DE DE60108650T patent/DE60108650T2/de not_active Expired - Fee Related
- 2001-09-14 CN CNB018159524A patent/CN1283239C/zh not_active Expired - Fee Related
- 2001-09-14 HU HU0302497A patent/HUP0302497A3/hu unknown
- 2001-09-14 WO PCT/EP2001/010731 patent/WO2002024186A1/en active IP Right Grant
- 2001-09-14 EP EP01967349A patent/EP1318800B1/en not_active Expired - Lifetime
- 2001-09-14 PT PT01967349T patent/PT1318800E/pt unknown
- 2001-09-14 UA UA2003043559A patent/UA73609C2/uk unknown
- 2001-09-14 PL PL36142801A patent/PL361428A1/xx unknown
- 2001-09-14 MX MXPA03001790A patent/MXPA03001790A/es active IP Right Grant
- 2001-09-14 KR KR1020037004009A patent/KR100570373B1/ko not_active IP Right Cessation
- 2001-09-14 EA EA200300388A patent/EA005499B1/ru not_active IP Right Cessation
- 2001-09-17 ZA ZA200107649A patent/ZA200107649B/xx unknown
- 2001-09-17 AR ARP010104388A patent/AR030750A1/es unknown
-
2003
- 2003-03-11 IL IL154867A patent/IL154867A/en not_active IP Right Cessation
- 2003-03-18 NO NO20031239A patent/NO20031239L/no not_active Application Discontinuation
-
2004
- 2004-02-13 HK HK04100992A patent/HK1058151A1/xx not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
CN1283239C (zh) | 2006-11-08 |
HK1058151A1 (en) | 2004-05-07 |
HUP0302497A3 (en) | 2005-08-29 |
NO20031239D0 (no) | 2003-03-18 |
PL361428A1 (en) | 2004-10-04 |
KR20030045079A (ko) | 2003-06-09 |
CA2420056A1 (en) | 2002-03-28 |
EP1318800A1 (en) | 2003-06-18 |
ZA200107649B (en) | 2002-05-14 |
DE60108650D1 (en) | 2005-03-03 |
HUP0302497A2 (hu) | 2003-12-29 |
US6602862B1 (en) | 2003-08-05 |
GEP20053480B (en) | 2005-03-25 |
KR100570373B1 (ko) | 2006-04-24 |
CN1461213A (zh) | 2003-12-10 |
AU8774001A (en) | 2002-04-02 |
CZ2003776A3 (en) | 2004-03-17 |
EP1318800B1 (en) | 2005-01-26 |
WO2002024186A1 (en) | 2002-03-28 |
ES2233679T3 (es) | 2005-06-16 |
EA005499B1 (ru) | 2005-02-24 |
NO20031239L (no) | 2003-03-18 |
PT1318800E (pt) | 2005-05-31 |
AU2001287740B2 (en) | 2005-01-27 |
UA73609C2 (en) | 2005-08-15 |
IL154867A0 (en) | 2003-10-31 |
CA2420056C (en) | 2007-11-13 |
MXPA03001790A (es) | 2004-11-01 |
ATE287708T1 (de) | 2005-02-15 |
TWI297605B (en) | 2008-06-11 |
AR030750A1 (es) | 2003-09-03 |
IL154867A (en) | 2009-08-03 |
DE60108650T2 (de) | 2006-01-19 |
JP2004509144A (ja) | 2004-03-25 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
MM4A | Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s) |
Designated state(s): AM AZ BY KZ KG MD TJ TM RU |