EA199901045A3 - Новые гидразидные соединения, способ их получения и содержащие их фармацевтические композиции - Google Patents

Новые гидразидные соединения, способ их получения и содержащие их фармацевтические композиции

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Publication number
EA199901045A3
EA199901045A3 EA199901045A EA199901045A EA199901045A3 EA 199901045 A3 EA199901045 A3 EA 199901045A3 EA 199901045 A EA199901045 A EA 199901045A EA 199901045 A EA199901045 A EA 199901045A EA 199901045 A3 EA199901045 A3 EA 199901045A3
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Eurasian Patent Office
Prior art keywords
group
alkylene
description
preparation
pharmaceutical compositions
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EA199901045A
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English (en)
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EA002442B1 (ru
EA199901045A2 (ru
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Вега Антонио Монхе
Мораса Игнанио Альдана
Даниель-Энри Кеньяр
Жак Дюо
Зюана Одиль Делла
Жан Бутэн
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Адир Э Компани
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Publication of EA199901045A2 publication Critical patent/EA199901045A2/ru
Publication of EA199901045A3 publication Critical patent/EA199901045A3/ru
Publication of EA002442B1 publication Critical patent/EA002442B1/ru

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Abstract

Соединения формулы (I)R-NH-A-CO-NH-NH-(W)-Z (I)где n равен 0 или 1,W обозначает группу -CO- или группу S(O), где r равен 0, 1 или 2,Z обозначает группу, выбранную из арила, арилалкила, гетероарила и гетероарилалкила, каждый из которых является необязательно замещенным,R обозначает группу, выбранную изZ-T-CO-, Z-O-T-CO-, Z-T-O-CO-, Z-T-S(O)-где Z, T и q имеют определенные в описании значения,A обозначает алкиленовую, алкениленовую или алкиниленовую группу, каждая из которых имеет 3-8 атомов углерода, алкиленциклоалкиленовую группу, циклоалкиленалкиленовую группу или алкиленциклоалкиленалкиленовую, алкиленариленовую группу, ариленалкиленовую группу, алкиленариленалкиленовую группу, группу, где Bимеет определенные в описании значения, или A образует с соседним атомом азота группуопределенную в описании.Лекарственные препараты.
EA199901045A 1998-12-17 1999-12-16 Новые гидразидные соединения, способ их получения и содержащие их фармацевтические композиции EA002442B1 (ru)

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Application Number Priority Date Filing Date Title
ES009802626A ES2161594B1 (es) 1998-12-17 1998-12-17 Nuevos derivados de la hidrazida, su procedimiento de preparacion y las composiciones farmaceuticas que los contienen.

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EA199901045A2 EA199901045A2 (ru) 2000-06-26
EA199901045A3 true EA199901045A3 (ru) 2000-10-30
EA002442B1 EA002442B1 (ru) 2002-04-25

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US (2) US6172108B1 (ru)
EP (1) EP1010691A3 (ru)
JP (1) JP3445204B2 (ru)
KR (1) KR100428686B1 (ru)
CN (1) CN1260345A (ru)
AU (1) AU763555B2 (ru)
BR (1) BR9907429A (ru)
CA (1) CA2292246A1 (ru)
EA (1) EA002442B1 (ru)
ES (1) ES2161594B1 (ru)
HU (1) HUP9904630A3 (ru)
NO (1) NO314399B1 (ru)
NZ (1) NZ501849A (ru)
PL (1) PL337253A1 (ru)
ZA (1) ZA997733B (ru)

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MXPA02004985A (es) * 1999-11-26 2003-10-14 Shionogi & Co Antagonistas del neuropeptido y, y5.
ES2187334B1 (es) * 2001-01-17 2004-09-16 Les Laboratoires Servier Nuevos derivados de la hidrazida, su procedimiento de preparacion y las composiciones farmaceuticas que los contienen.
TWI297335B (en) 2001-07-10 2008-06-01 Synta Pharmaceuticals Corp Taxol enhancer compounds
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TWI252847B (en) * 2001-07-10 2006-04-11 Synta Pharmaceuticals Corp Synthesis of taxol enhancers
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ES2161594A1 (es) 2001-12-01
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US6271247B1 (en) 2001-08-07
HUP9904630A2 (hu) 2000-08-28
US6172108B1 (en) 2001-01-09
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ES2161594B1 (es) 2003-04-01
EA002442B1 (ru) 2002-04-25
EA199901045A2 (ru) 2000-06-26
CA2292246A1 (fr) 2000-06-17
ZA997733B (en) 2000-06-29
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PL337253A1 (en) 2000-06-19
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