EA199801015A1 - Производные пиперидинуксусной кислоты и их применение при лечении тромботических нарушений - Google Patents

Производные пиперидинуксусной кислоты и их применение при лечении тромботических нарушений

Info

Publication number
EA199801015A1
EA199801015A1 EA199801015A EA199801015A EA199801015A1 EA 199801015 A1 EA199801015 A1 EA 199801015A1 EA 199801015 A EA199801015 A EA 199801015A EA 199801015 A EA199801015 A EA 199801015A EA 199801015 A1 EA199801015 A1 EA 199801015A1
Authority
EA
Eurasian Patent Office
Prior art keywords
treatment
application
piperidinoxic
derivatives
acid
Prior art date
Application number
EA199801015A
Other languages
English (en)
Russian (ru)
Inventor
Дейвид Джордж Аллен
Колин Дейвид Элдред
Брайан Дейвид Джадкинс
Уильям Леонард Митчелл
Original Assignee
Глаксо Груп Лимитед
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GBGB9613017.4A external-priority patent/GB9613017D0/en
Priority claimed from GBGB9613095.0A external-priority patent/GB9613095D0/en
Priority claimed from GBGB9613018.2A external-priority patent/GB9613018D0/en
Application filed by Глаксо Груп Лимитед filed Critical Глаксо Груп Лимитед
Publication of EA199801015A1 publication Critical patent/EA199801015A1/ru

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4151,2-Diazoles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D453/00Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
EA199801015A 1996-06-21 1997-06-19 Производные пиперидинуксусной кислоты и их применение при лечении тромботических нарушений EA199801015A1 (ru)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
GBGB9613017.4A GB9613017D0 (en) 1996-06-21 1996-06-21 Therapeutic compounds
GBGB9613095.0A GB9613095D0 (en) 1996-06-21 1996-06-21 Therapeutic piperidines
GBGB9613018.2A GB9613018D0 (en) 1996-06-21 1996-06-21 Therapeutic indazoles
PCT/EP1997/003196 WO1997049699A1 (en) 1996-06-21 1997-06-19 Piperidine acetic acid derivatives and their use in the treatment of thrombotic disorders

Publications (1)

Publication Number Publication Date
EA199801015A1 true EA199801015A1 (ru) 1999-08-26

Family

ID=27268341

Family Applications (1)

Application Number Title Priority Date Filing Date
EA199801015A EA199801015A1 (ru) 1996-06-21 1997-06-19 Производные пиперидинуксусной кислоты и их применение при лечении тромботических нарушений

Country Status (17)

Country Link
EP (1) EP0912555A1 (cs)
JP (1) JP2000512648A (cs)
KR (1) KR20000022041A (cs)
AP (1) AP9801417A0 (cs)
AR (1) AR008245A1 (cs)
AU (1) AU3261197A (cs)
BR (1) BR9709930A (cs)
CA (1) CA2258753A1 (cs)
CZ (1) CZ424698A3 (cs)
EA (1) EA199801015A1 (cs)
ID (1) ID17052A (cs)
IL (1) IL127464A0 (cs)
IS (1) IS4924A (cs)
NO (1) NO985974L (cs)
PL (1) PL330797A1 (cs)
TR (1) TR199802665T2 (cs)
WO (1) WO1997049699A1 (cs)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7642278B2 (en) 2001-07-03 2010-01-05 Novartis Vaccines And Diagnostics, Inc. Indazole benzimidazole compounds
WO2003004488A1 (en) 2001-07-03 2003-01-16 Chiron Corporation Indazole benzimidazole compounds as tyrosine and serine/threonine kinase inhibitors
TW200401641A (en) * 2002-07-18 2004-02-01 Wyeth Corp 1-Heterocyclylalkyl-3-sulfonylindole or-indazole derivatives as 5-hydroxytryptamine-6 ligands
JP2006518385A (ja) * 2003-02-14 2006-08-10 ワイス 5−ヒドロキシトリプタミン−6リガンドとしてのヘテロサイクリル−3−スルホニルインダゾール
EP2001865A1 (en) 2006-04-05 2008-12-17 Wyeth a Corporation of the State of Delaware Sulfonyl-3-heterocyclylindazole derivatives as 5-hydroxytryptamine-6 ligands
BRPI0806542A2 (pt) 2007-01-10 2014-04-22 Hoffmann La Roche Derivados de sulfonamida como inibidores de quimase
CN113655155A (zh) * 2021-07-28 2021-11-16 任贤金 一种测定sph3127有关物质的方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE4124942A1 (de) * 1991-07-27 1993-01-28 Thomae Gmbh Dr K 5-gliedrige heterocyclen, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel
TW221996B (cs) * 1991-11-14 1994-04-01 Glaxo Group Ltd
GB9208740D0 (en) * 1992-04-23 1992-06-10 Glaxo Group Ltd Chemical compounds

Also Published As

Publication number Publication date
NO985974L (no) 1999-02-17
KR20000022041A (ko) 2000-04-25
AR008245A1 (es) 1999-12-29
IL127464A0 (en) 1999-10-28
AU3261197A (en) 1998-01-14
JP2000512648A (ja) 2000-09-26
NO985974D0 (no) 1998-12-18
IS4924A (is) 1998-12-15
WO1997049699A1 (en) 1997-12-31
PL330797A1 (en) 1999-06-07
BR9709930A (pt) 1999-08-10
ID17052A (id) 1997-12-04
AP9801417A0 (en) 1998-12-31
TR199802665T2 (xx) 1999-03-22
EP0912555A1 (en) 1999-05-06
CA2258753A1 (en) 1997-12-31
CZ424698A3 (cs) 1999-05-12

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