AR008245A1 - Derivados de acido acetico, uso de los mismos en la fabricacion de un agente terapeutico y proceso para preparar dichos derivados - Google Patents
Derivados de acido acetico, uso de los mismos en la fabricacion de un agente terapeutico y proceso para preparar dichos derivadosInfo
- Publication number
- AR008245A1 AR008245A1 ARP970102676A ARP970102676A AR008245A1 AR 008245 A1 AR008245 A1 AR 008245A1 AR P970102676 A ARP970102676 A AR P970102676A AR P970102676 A ARP970102676 A AR P970102676A AR 008245 A1 AR008245 A1 AR 008245A1
- Authority
- AR
- Argentina
- Prior art keywords
- derivatives
- prepare
- manufacture
- acetic acid
- therapeutic agent
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
- C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
Compuestos de la fórmula (I) o una sal, solvato o derivado del mismo funcional fisiológicamente, en el cual: X representa ya sea CH2-CCCH2 o CH=CH;Y representa un grupo de fórmula (II); R0 representa SO2Me o CONH2, y R1 es SO2Me, a procesos para su preparación, a composicones farmacéuticas quecontienen tales compuestos y a su uso en la preparación de agentes para el tratamiento de desórdenes trombóticos.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GBGB9613018.2A GB9613018D0 (en) | 1996-06-21 | 1996-06-21 | Therapeutic indazoles |
GBGB9613095.0A GB9613095D0 (en) | 1996-06-21 | 1996-06-21 | Therapeutic piperidines |
GBGB9613017.4A GB9613017D0 (en) | 1996-06-21 | 1996-06-21 | Therapeutic compounds |
Publications (1)
Publication Number | Publication Date |
---|---|
AR008245A1 true AR008245A1 (es) | 1999-12-29 |
Family
ID=27268341
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP970102676A AR008245A1 (es) | 1996-06-21 | 1997-06-18 | Derivados de acido acetico, uso de los mismos en la fabricacion de un agente terapeutico y proceso para preparar dichos derivados |
Country Status (17)
Country | Link |
---|---|
EP (1) | EP0912555A1 (es) |
JP (1) | JP2000512648A (es) |
KR (1) | KR20000022041A (es) |
AP (1) | AP9801417A0 (es) |
AR (1) | AR008245A1 (es) |
AU (1) | AU3261197A (es) |
BR (1) | BR9709930A (es) |
CA (1) | CA2258753A1 (es) |
CZ (1) | CZ424698A3 (es) |
EA (1) | EA199801015A1 (es) |
ID (1) | ID17052A (es) |
IL (1) | IL127464A0 (es) |
IS (1) | IS4924A (es) |
NO (1) | NO985974L (es) |
PL (1) | PL330797A1 (es) |
TR (1) | TR199802665T2 (es) |
WO (1) | WO1997049699A1 (es) |
Families Citing this family (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US7642278B2 (en) | 2001-07-03 | 2010-01-05 | Novartis Vaccines And Diagnostics, Inc. | Indazole benzimidazole compounds |
US7064215B2 (en) | 2001-07-03 | 2006-06-20 | Chiron Corporation | Indazole benzimidazole compounds |
TW200401641A (en) | 2002-07-18 | 2004-02-01 | Wyeth Corp | 1-Heterocyclylalkyl-3-sulfonylindole or-indazole derivatives as 5-hydroxytryptamine-6 ligands |
WO2004074243A2 (en) * | 2003-02-14 | 2004-09-02 | Wyeth | Heterocyclyl-3-sulfonylindazoles as 5-hydroxytryptamine-6 ligands |
WO2007117413A1 (en) | 2006-04-05 | 2007-10-18 | Wyeth | Sulfonyl-3-heterocyclylindazole derivatives as 5-hydroxytryptamine-6 ligands |
CN101578265B (zh) | 2007-01-10 | 2013-05-08 | 霍夫曼-拉罗奇有限公司 | 用作糜蛋白酶抑制剂的磺酰胺衍生物 |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE4124942A1 (de) * | 1991-07-27 | 1993-01-28 | Thomae Gmbh Dr K | 5-gliedrige heterocyclen, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel |
JPH07501063A (ja) * | 1991-11-14 | 1995-02-02 | グラクソ、グループ、リミテッド | フィブリノーゲン依存性血小板凝集阻害剤としてのピペリジン酢酸誘導体 |
GB9208740D0 (en) * | 1992-04-23 | 1992-06-10 | Glaxo Group Ltd | Chemical compounds |
-
1997
- 1997-06-18 AR ARP970102676A patent/AR008245A1/es unknown
- 1997-06-19 PL PL97330797A patent/PL330797A1/xx unknown
- 1997-06-19 CZ CZ984246A patent/CZ424698A3/cs unknown
- 1997-06-19 IL IL12746497A patent/IL127464A0/xx unknown
- 1997-06-19 TR TR1998/02665T patent/TR199802665T2/xx unknown
- 1997-06-19 EP EP97928243A patent/EP0912555A1/en not_active Withdrawn
- 1997-06-19 KR KR1019980710439A patent/KR20000022041A/ko not_active Application Discontinuation
- 1997-06-19 AU AU32611/97A patent/AU3261197A/en not_active Abandoned
- 1997-06-19 ID IDP972092A patent/ID17052A/id unknown
- 1997-06-19 EA EA199801015A patent/EA199801015A1/ru unknown
- 1997-06-19 AP APAP/P/1998/001417A patent/AP9801417A0/en unknown
- 1997-06-19 CA CA002258753A patent/CA2258753A1/en not_active Abandoned
- 1997-06-19 WO PCT/EP1997/003196 patent/WO1997049699A1/en not_active Application Discontinuation
- 1997-06-19 BR BR9709930A patent/BR9709930A/pt not_active Application Discontinuation
- 1997-06-19 JP JP10502284A patent/JP2000512648A/ja active Pending
-
1998
- 1998-12-15 IS IS4924A patent/IS4924A/is unknown
- 1998-12-18 NO NO985974A patent/NO985974L/no not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
JP2000512648A (ja) | 2000-09-26 |
IS4924A (is) | 1998-12-15 |
ID17052A (id) | 1997-12-04 |
CZ424698A3 (cs) | 1999-05-12 |
CA2258753A1 (en) | 1997-12-31 |
IL127464A0 (en) | 1999-10-28 |
NO985974D0 (no) | 1998-12-18 |
AU3261197A (en) | 1998-01-14 |
EA199801015A1 (ru) | 1999-08-26 |
AP9801417A0 (en) | 1998-12-31 |
KR20000022041A (ko) | 2000-04-25 |
EP0912555A1 (en) | 1999-05-06 |
WO1997049699A1 (en) | 1997-12-31 |
PL330797A1 (en) | 1999-06-07 |
NO985974L (no) | 1999-02-17 |
BR9709930A (pt) | 1999-08-10 |
TR199802665T2 (xx) | 1999-03-22 |
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