EA023697B1 - ПРИМЕНЕНИЕ КОМБИНАЦИИ ИЗ 7-(2,5-ДИГИДРО-4-ИМИДАЗО[1,2-а]ПИРИДИН-3-ИЛ-2,5-ДИОКСО-1Н-ПИРРОЛ-3-ИЛ)-9-ФТОР-1,2,3,4-ТЕТРАГИДРО-2-(1-ПИПЕРИДИНИЛКАРБОНИЛ)ПИРРОЛО[3,2,1-jk][1,4]БЕНЗОДИАЗЕПИНА И ХИМИОТЕРАПЕВТИЧЕСКОГО АГЕНТА ДЛЯ ПОЛУЧЕНИЯ ЛЕКАРСТВЕННОГО СРЕДСТВА ДЛЯ ЛЕЧЕНИЯ РАКА ЖЕЛУДКА - Google Patents
ПРИМЕНЕНИЕ КОМБИНАЦИИ ИЗ 7-(2,5-ДИГИДРО-4-ИМИДАЗО[1,2-а]ПИРИДИН-3-ИЛ-2,5-ДИОКСО-1Н-ПИРРОЛ-3-ИЛ)-9-ФТОР-1,2,3,4-ТЕТРАГИДРО-2-(1-ПИПЕРИДИНИЛКАРБОНИЛ)ПИРРОЛО[3,2,1-jk][1,4]БЕНЗОДИАЗЕПИНА И ХИМИОТЕРАПЕВТИЧЕСКОГО АГЕНТА ДЛЯ ПОЛУЧЕНИЯ ЛЕКАРСТВЕННОГО СРЕДСТВА ДЛЯ ЛЕЧЕНИЯ РАКА ЖЕЛУДКА Download PDFInfo
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- EA023697B1 EA023697B1 EA201201155A EA201201155A EA023697B1 EA 023697 B1 EA023697 B1 EA 023697B1 EA 201201155 A EA201201155 A EA 201201155A EA 201201155 A EA201201155 A EA 201201155A EA 023697 B1 EA023697 B1 EA 023697B1
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- EA
- Eurasian Patent Office
- Prior art keywords
- compound
- fluoro
- imidazo
- dihydro
- mmol
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Landscapes
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| EP2747761A1 (en) * | 2011-09-22 | 2014-07-02 | Bind Therapeutics, Inc. | Methods of treating cancers with therapeutic nanoparticles |
| TW201417817A (zh) * | 2012-09-25 | 2014-05-16 | Daiichi Sankyo Co Ltd | Ｇｓｋ３抑制劑與抗ｄｒ５抗體之組合 |
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| US10201540B2 (en) | 2016-03-02 | 2019-02-12 | Frequency Therapeutics, Inc. | Solubilized compositions for controlled proliferation of stem cells / generating inner ear hair cells using GSK3 inhibitors: I |
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| WO2018125746A1 (en) | 2016-12-30 | 2018-07-05 | Frequency Therapeutics, Inc. | 1h-pyrrole-2,5-dione compounds and methods of using them to induce self-renewal of stem/progenitor supporting cells |
| AU2020218366A1 (en) | 2019-02-08 | 2021-09-16 | Frequency Therapeutics, Inc. | Valproic acid compounds and Wnt agonists for treating ear disorders |
| AU2022285754A1 (en) * | 2021-06-03 | 2023-12-14 | University Of Cincinnati | Bzd-1 as a chemosensitizer of cancer |
| CN113956157B (zh) * | 2021-11-18 | 2024-05-03 | 西安都创医药科技有限公司 | 一种合成2-甲酰基-1-环丙烷甲酸乙酯的方法 |
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| GB8904161D0 (en) * | 1989-02-23 | 1989-04-05 | Hoffmann La Roche | Substituted pyrroles |
| KR0166088B1 (ko) * | 1990-01-23 | 1999-01-15 | . | 수용해도가 증가된 시클로덱스트린 유도체 및 이의 용도 |
| US5376645A (en) * | 1990-01-23 | 1994-12-27 | University Of Kansas | Derivatives of cyclodextrins exhibiting enhanced aqueous solubility and the use thereof |
| US7034013B2 (en) * | 2001-03-20 | 2006-04-25 | Cydex, Inc. | Formulations containing propofol and a sulfoalkyl ether cyclodextrin |
| KR100974770B1 (ko) * | 2002-03-05 | 2010-08-06 | 일라이 릴리 앤드 캄파니 | 키나제 억제제로서의 퓨린 유도체 |
| AR041291A1 (es) * | 2002-09-19 | 2005-05-11 | Schering Corp | Imidazopiridinas como inhibidores de quinasa dependientes de ciclina |
| CA2569091A1 (en) | 2004-07-09 | 2006-01-19 | Agency For Science, Technology And Research | Modulation of gsk-3.beta. and method of treating proliferative disorders |
| GB0418328D0 (en) * | 2004-08-17 | 2004-09-22 | Imp College Innovations Ltd | Cancer methods and medicaments |
| EP2460886B1 (en) * | 2005-05-04 | 2014-01-01 | University of South Florida | Predicting treatment response in cancer subjects |
| TWI428132B (zh) * | 2007-07-02 | 2014-03-01 | Lilly Co Eli | 癌症化療效果之強化 |
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