EA020923B1 - Производные димерного 1-арилпиразола - Google Patents

Производные димерного 1-арилпиразола Download PDF

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Publication number
EA020923B1
EA020923B1 EA201100800A EA201100800A EA020923B1 EA 020923 B1 EA020923 B1 EA 020923B1 EA 201100800 A EA201100800 A EA 201100800A EA 201100800 A EA201100800 A EA 201100800A EA 020923 B1 EA020923 B1 EA 020923B1
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EA
Eurasian Patent Office
Prior art keywords
composition
compounds
independently represent
group
compound
Prior art date
Application number
EA201100800A
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English (en)
Russian (ru)
Other versions
EA201100800A1 (ru
Inventor
Чарльз К. Менг
Original Assignee
Мериал Лимитед
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Application filed by Мериал Лимитед filed Critical Мериал Лимитед
Publication of EA201100800A1 publication Critical patent/EA201100800A1/ru
Publication of EA020923B1 publication Critical patent/EA020923B1/ru

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/18—One oxygen or sulfur atom
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/56—1,2-Diazoles; Hydrogenated 1,2-diazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/14—Ectoparasiticides, e.g. scabicides

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pest Control & Pesticides (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Public Health (AREA)
  • Agronomy & Crop Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Plant Pathology (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
EA201100800A 2008-11-19 2009-11-18 Производные димерного 1-арилпиразола EA020923B1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US11602108P 2008-11-19 2008-11-19
PCT/US2009/064981 WO2010059719A2 (en) 2008-11-19 2009-11-18 Dimeric 1-arylpyrazole derivatives

Publications (2)

Publication Number Publication Date
EA201100800A1 EA201100800A1 (ru) 2011-12-30
EA020923B1 true EA020923B1 (ru) 2015-02-27

Family

ID=42034586

Family Applications (1)

Application Number Title Priority Date Filing Date
EA201100800A EA020923B1 (ru) 2008-11-19 2009-11-18 Производные димерного 1-арилпиразола

Country Status (12)

Country Link
US (1) US8642636B2 (enExample)
EP (1) EP2364300B1 (enExample)
JP (1) JP2012509338A (enExample)
CN (1) CN102264706A (enExample)
AU (1) AU2009316710B2 (enExample)
BR (1) BRPI0922042B1 (enExample)
CA (2) CA2952443C (enExample)
EA (1) EA020923B1 (enExample)
ES (1) ES2605811T3 (enExample)
MX (1) MX2011005214A (enExample)
NZ (1) NZ592985A (enExample)
WO (1) WO2010059719A2 (enExample)

Families Citing this family (25)

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MY173181A (en) 2011-05-13 2020-01-02 Array Biopharma Inc Pyrrolidinyl urea, pyrrolidinyl thiourea and pyrrolidinyl guanidine compounds as trka kinase inhibitors
WO2014078378A1 (en) 2012-11-13 2014-05-22 Array Biopharma Inc. Pyrrolidinyl urea, thiourea, guanidine and cyanoguanidine compounds as trka kinase inhibitors
US9822118B2 (en) 2012-11-13 2017-11-21 Array Biopharma Inc. Bicyclic heteroaryl urea, thiourea, guanidine and cyanoguanidine compounds as TrkA kinase inhibitors
US9790178B2 (en) 2012-11-13 2017-10-17 Array Biopharma Inc. Pyrrolidinyl urea, thiourea, guanidine and cyanoguanidine compounds as TrkA kinase inhibitors
EP2920166B1 (en) 2012-11-13 2016-11-02 Array Biopharma, Inc. Bicyclic urea, thiourea, guanidine and cyanoguanidine compounds useful for the treatment of pain
WO2014078325A1 (en) 2012-11-13 2014-05-22 Array Biopharma Inc. N-(monocyclic aryl),n'-pyrazolyl-urea, thiourea, guanidine and cyanoguanidine compounds as trka kinase inhibitors
WO2014078331A1 (en) 2012-11-13 2014-05-22 Array Biopharma Inc. N-(arylalkyl)-n'-pyrazolyl-urea, thiourea, guanidine and cyanoguanidine compounds as trka kinase inhibitors
WO2014078328A1 (en) 2012-11-13 2014-05-22 Array Biopharma Inc. N-bicyclic aryl,n'-pyrazolyl urea, thiourea, guanidine and cyanoguanidine compounds as trka kinase inhibitors
EP2922844B1 (en) 2012-11-13 2018-01-10 Array Biopharma, Inc. N-pyrrolidinyl, n'-pyrazolyl- urea, thiourea, guanidine and cyanoguanidine compounds as trka kinase inhibitors
US9981959B2 (en) 2012-11-13 2018-05-29 Array Biopharma Inc. Thiazolyl and oxazolyl urea, thiourea, guanidine and cyanoguanidine compounds as TrkA kinase inhibitors
US9809578B2 (en) 2012-11-13 2017-11-07 Array Biopharma Inc. Pyrazolyl urea, thiourea, guanidine and cyanoguanidine compounds as trkA kinase inhibitors
JP2016164125A (ja) * 2013-07-02 2016-09-08 国立大学法人帯広畜産大学 バベシア症の治療剤及び予防剤
LT3154959T (lt) 2014-05-15 2019-09-25 Array Biopharma, Inc. 1-((3s,4r)-4-(3-fluorfenil)-1-(2-metoksietil)pirolidin-3-il)-3-(4-metil-3-(2-metilpirimidin-5-il)-1-fenil-1h-pirazol-5-il)karbamidas kaip trka kinazės inhibitorius
US11384032B2 (en) 2016-05-12 2022-07-12 Verdesian Life Sciences, U.S., Llc Compositions for controlling enzyme-induced urea decomposition
WO2018183562A1 (en) 2017-03-28 2018-10-04 Verdesian Life Sciences, U.S., Llc Triarylmethane compounds for controlling enzyme-induced urea decomposition
WO2020096831A1 (en) 2018-11-06 2020-05-14 Dow Agrosciences Llc Safened compositions comprising pyridine carboxylate herbicides and cloquintocet
WO2020096832A1 (en) * 2018-11-06 2020-05-14 Dow Agrosciences Llc Compositions comprising pyridine carboxylate herbicides and azole carboxylate safeners
US12285012B2 (en) 2018-11-07 2025-04-29 Corteva Agriscience Llc Compositions comprising pyridine carboxylate herbicides with acetolactate synthase (ALS) inhibitor herbicides
EA202191265A1 (ru) 2018-11-07 2021-07-27 КОРТЕВА АГРИСАЙЕНС ЭлЭлСи Композиции, содержащие гербицид на основе пиридинкарбоксилата и гербициды, представляющие собой ингибиторы протопорфириногеноксидазы (protox)
BR112021008843A2 (pt) 2018-11-07 2021-08-17 Corteva Agriscience Llc composições que compreendem herbicidas de carboxilato de piridina com fotossistema ii e herbicidas inibidores da hppd opcionais
CN112996393B (zh) 2018-11-07 2023-05-12 科迪华农业科技有限责任公司 包含羧酸吡啶除草剂与合成生长素除草剂或生长素转运抑制剂的组合物
WO2020096936A1 (en) 2018-11-07 2020-05-14 Dow Agrosciences Llc Compositions comprising pyridine carboxylate herbicides and 4-hydroxyphenyl-pyruvate dioxygenase (hppd) inhibitor herbicides
EP3886854A4 (en) 2018-11-30 2022-07-06 Nuvation Bio Inc. Pyrrole and pyrazole compounds and methods of use thereof
KR20230043904A (ko) 2020-07-24 2023-03-31 엘랑코 유에스 인코포레이티드 이속사졸린 화합물 및 이의 중간체의 제조 공정
EP4208157A1 (en) 2020-09-04 2023-07-12 Elanco Us Inc. Palatable formulations

Citations (2)

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Publication number Priority date Publication date Assignee Title
US3966900A (en) * 1969-03-12 1976-06-29 Airwick Industries, Inc. Evaporator system comprising a stabilized pesticidal phosphoric acid ester and method for stabilizing such ester enclosed in an evaporator
US20070275976A1 (en) * 2004-06-26 2007-11-29 Stefan Schnatterer N-phenylpyrazole derivatives as pesticides

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU784798B2 (en) * 1999-12-02 2006-06-22 Boehringer Ingelheim Animal Health USA Inc. Control of arthropods in animals
US7262214B2 (en) * 2003-02-26 2007-08-28 Merial Limited 1-N-arylpyrazole derivatives in prevention of arthropod-borne and mosquito-borne diseases

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3966900A (en) * 1969-03-12 1976-06-29 Airwick Industries, Inc. Evaporator system comprising a stabilized pesticidal phosphoric acid ester and method for stabilizing such ester enclosed in an evaporator
US20070275976A1 (en) * 2004-06-26 2007-11-29 Stefan Schnatterer N-phenylpyrazole derivatives as pesticides

Non-Patent Citations (5)

* Cited by examiner, † Cited by third party
Title
BOURGUIGNON J.: "IDENTICAL AND NONIDENTICAL TWIN DRUGS". PRACTICE OF MEDICINAL CHEMISTRY, 1 January 1996 (1996-01-01), pages 261-293, XP001248799, the whole document *
DATABASE BEILSTEIN 1996, XP002575606. Database accession no. 6036932, abstract & COUR, AGNETE LA; FINDEISEN, MATTHIAS; HAZELL, RITA; HENNIG, LOTHAR; OLSEN, CARL ERIK; SIMONSEN, OLE: J. CHEM. SOC., DALTON TRANSACTIONS: INORGANIC CHEMISTRY, vol. 16, 1996, pages 3437-3448 *
DATABASE BEILSTEIN. BEILSTEIN INSTITUTE FOR ORGANIC CHEMISTRY, FRANKFURT-MAIN, DE; 1959, XP002575607. Database accession no. 630245, abstract & FINAR; LORD: J. CHEM. SOC., 1959, pages 1819-1821 *
DATABASE BEILSTEIN. BEILSTEIN INSTITUTE FOR ORGANIC CHEMISTRY, FRANKFURT-MAIN, DE; 1996, XP002575604. Database accession no. 6010790, abstract & NIVOROZHKIN, ALEXANDER L.; TOFTLUND, HANS; JOERGENSEN, PER LAUGE; NIVOROZHKIN, LEONID E.: J. CHEM. SOC., DALTON TRANSACTIONS: INORG. CHEM., vol. 7, 1996, pages 1215-1222 *
DATABASE BEILSTEIN. BEILSTEIN INSTITUTE FOR ORGANIC CHEMISTRY, FRANKFURT-MAIN, DE; 1997, XP002575605. Database accession no. 6206504, abstract & AHLUWALIA, V. K.; SHARMA, POOJA; GOYAL, BINDU: IND. J. CHEM., SECTION B: ORGANIC CHEMISTRY INCLUDING MEDICINAL CHEMISTRY, vol. 36, 1997, pages 1059-1061 *

Also Published As

Publication number Publication date
EA201100800A1 (ru) 2011-12-30
JP2012509338A (ja) 2012-04-19
CA2952443C (en) 2019-04-02
AU2009316710A1 (en) 2010-05-27
BRPI0922042B1 (pt) 2020-01-28
CA2743553C (en) 2017-03-14
MX2011005214A (es) 2011-06-01
CN102264706A (zh) 2011-11-30
CA2952443A1 (en) 2010-05-27
EP2364300B1 (en) 2016-10-19
HK1160852A1 (en) 2012-08-17
EP2364300A2 (en) 2011-09-14
BRPI0922042A2 (pt) 2016-11-01
US8642636B2 (en) 2014-02-04
CA2743553A1 (en) 2010-05-27
ES2605811T3 (es) 2017-03-16
US20110245157A1 (en) 2011-10-06
WO2010059719A3 (en) 2010-11-18
AU2009316710B2 (en) 2015-08-06
WO2010059719A2 (en) 2010-05-27
NZ592985A (en) 2013-04-26

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MM4A Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s)

Designated state(s): AM AZ BY KZ KG MD TJ TM RU