EA020923B1 - Производные димерного 1-арилпиразола - Google Patents

Производные димерного 1-арилпиразола Download PDF

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Publication number
EA020923B1
EA020923B1 EA201100800A EA201100800A EA020923B1 EA 020923 B1 EA020923 B1 EA 020923B1 EA 201100800 A EA201100800 A EA 201100800A EA 201100800 A EA201100800 A EA 201100800A EA 020923 B1 EA020923 B1 EA 020923B1
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EA
Eurasian Patent Office
Prior art keywords
composition
compounds
independently represent
group
compound
Prior art date
Application number
EA201100800A
Other languages
English (en)
Russian (ru)
Other versions
EA201100800A1 (ru
Inventor
Чарльз К. Менг
Original Assignee
Мериал Лимитед
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Publication date
Application filed by Мериал Лимитед filed Critical Мериал Лимитед
Publication of EA201100800A1 publication Critical patent/EA201100800A1/ru
Publication of EA020923B1 publication Critical patent/EA020923B1/ru

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/18—One oxygen or sulfur atom
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/56—1,2-Diazoles; Hydrogenated 1,2-diazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/14—Ectoparasiticides, e.g. scabicides

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pest Control & Pesticides (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Public Health (AREA)
  • Agronomy & Crop Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Plant Pathology (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
EA201100800A 2008-11-19 2009-11-18 Производные димерного 1-арилпиразола EA020923B1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US11602108P 2008-11-19 2008-11-19
PCT/US2009/064981 WO2010059719A2 (en) 2008-11-19 2009-11-18 Dimeric 1-arylpyrazole derivatives

Publications (2)

Publication Number Publication Date
EA201100800A1 EA201100800A1 (ru) 2011-12-30
EA020923B1 true EA020923B1 (ru) 2015-02-27

Family

ID=42034586

Family Applications (1)

Application Number Title Priority Date Filing Date
EA201100800A EA020923B1 (ru) 2008-11-19 2009-11-18 Производные димерного 1-арилпиразола

Country Status (12)

Country Link
US (1) US8642636B2 (cg-RX-API-DMAC7.html)
EP (1) EP2364300B1 (cg-RX-API-DMAC7.html)
JP (1) JP2012509338A (cg-RX-API-DMAC7.html)
CN (1) CN102264706A (cg-RX-API-DMAC7.html)
AU (1) AU2009316710B2 (cg-RX-API-DMAC7.html)
BR (1) BRPI0922042B1 (cg-RX-API-DMAC7.html)
CA (2) CA2743553C (cg-RX-API-DMAC7.html)
EA (1) EA020923B1 (cg-RX-API-DMAC7.html)
ES (1) ES2605811T3 (cg-RX-API-DMAC7.html)
MX (1) MX2011005214A (cg-RX-API-DMAC7.html)
NZ (1) NZ592985A (cg-RX-API-DMAC7.html)
WO (1) WO2010059719A2 (cg-RX-API-DMAC7.html)

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ES2615738T3 (es) 2011-05-13 2017-06-08 Array Biopharma, Inc. Compuestos de pirrolidinil urea, pirrolidinil tiourea y pirrolidinil guanidina como inhibidores de trkA quinasa
US9981959B2 (en) 2012-11-13 2018-05-29 Array Biopharma Inc. Thiazolyl and oxazolyl urea, thiourea, guanidine and cyanoguanidine compounds as TrkA kinase inhibitors
WO2014078331A1 (en) 2012-11-13 2014-05-22 Array Biopharma Inc. N-(arylalkyl)-n'-pyrazolyl-urea, thiourea, guanidine and cyanoguanidine compounds as trka kinase inhibitors
PL2920166T3 (pl) 2012-11-13 2017-05-31 Array Biopharma, Inc. Bicykliczne związki mocznika, tiomocznika, guanidyny i cyjanoguanidyny przydatne w leczeniu bólu
WO2014078372A1 (en) 2012-11-13 2014-05-22 Array Biopharma Inc. Pyrrolidinyl urea, thiourea, guanidine and cyanoguanidine compounds as trka kinase inhibitors
US9790210B2 (en) 2012-11-13 2017-10-17 Array Biopharma Inc. N-(monocyclic aryl),N'-pyrazolyl-urea, thiourea, guanidine and cyanoguanidine compounds as TrkA kinase inhibitors
WO2014078408A1 (en) 2012-11-13 2014-05-22 Array Biopharma Inc. Bicyclic heteroaryl urea, thiourea, guanidine and cyanoguanidine compounds as trka kinase inhibitors
US9546156B2 (en) 2012-11-13 2017-01-17 Array Biopharma Inc. N-bicyclic aryl,N'-pyrazolyl urea, thiourea, guanidine cyanoguanidine compounds as TrkA kinase inhibitors
ME02990B (me) 2012-11-13 2018-10-20 Array Biopharma Inc Jedinjenja n-pirolidinil, n'-pirazolil- uree, tiouree, guanidina i cijanoguanidina kао inhibitori trka kinaze
WO2014078417A1 (en) 2012-11-13 2014-05-22 Array Biopharma Inc. Pyrazolyl urea, thiourea, guanidine and cyanoguanidine compounds as trka kinase inhibitors
WO2014078378A1 (en) 2012-11-13 2014-05-22 Array Biopharma Inc. Pyrrolidinyl urea, thiourea, guanidine and cyanoguanidine compounds as trka kinase inhibitors
JP2016164125A (ja) * 2013-07-02 2016-09-08 国立大学法人帯広畜産大学 バベシア症の治療剤及び予防剤
RU2719489C2 (ru) 2014-05-15 2020-04-17 Эррэй Биофарма Инк. 1-((3S,4R)-4-(3-ФТОРФЕНИЛ)-1-(2-МЕТОКСИЭТИЛ)ПИРРОЛИДИН-3-ИЛ)-3-(4-МЕТИЛ-3-(2-МЕТИЛПИРИМИДИН-5-ИЛ)-1-ФЕНИЛ-1Н-ПИРАЗОЛ-5-ИЛ)МОЧЕВИНА В КАЧЕСТВЕ ИНГИБИТОРА TrkA КИНАЗЫ
WO2017195173A1 (en) 2016-05-12 2017-11-16 Verdesian Life Sciences, U.S., Llc Compositions for controlling enzyme-induced urea decomposition
MY201375A (en) 2017-03-28 2024-02-20 Verdesian Life Sciences Us Llc Triarylmethane compounds for controlling enzyme-induced urea decomposition
ES3047398T3 (en) 2018-11-06 2025-12-03 Corteva Agriscience Llc Safened compositions comprising pyridine carboxylate herbicides and cloquintocet
LT3876726T (lt) * 2018-11-06 2025-03-10 Corteva Agriscience Llc Kompozicijos, apimančios piridino karboksilato herbicidus ir azolo karboksilato herbicidų antidotus
MX2021005341A (es) 2018-11-07 2021-06-30 Corteva Agriscience Llc Composiciones que comprenden herbicidas de carboxilato de piridina con herbicidas de inhibidores de acetolactato sintasa (als).
WO2020096929A1 (en) 2018-11-07 2020-05-14 Dow Agrosciences Llc Compositions comprising pyridine carboxylate herbicides with photosystem ii and optional hppd inhibitor herbicides
PL3876729T3 (pl) 2018-11-07 2025-04-14 Corteva Agriscience Llc Kompozycje zawierające herbicyd pirydynokarboksylanowy oraz herbicydy będące inhibitorami oksydazy protoporfirynogenu (protox)
ES3041637T3 (en) 2018-11-07 2025-11-13 Corteva Agriscience Llc Compositions comprising pyridine carboxylate herbicides and 4-hydroxyphenyl-pyruvate dioxygenase (hppd) inhibitor herbicides
AU2019387370A1 (en) 2018-11-30 2021-06-10 Nuvation Bio Inc. Pyrrole and pyrazole compounds and methods of use thereof
CA3185969A1 (en) 2020-07-24 2022-01-27 Jean Marie Defauw Process for making an isoxazoline compound and intermediate thereof

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3966900A (en) * 1969-03-12 1976-06-29 Airwick Industries, Inc. Evaporator system comprising a stabilized pesticidal phosphoric acid ester and method for stabilizing such ester enclosed in an evaporator
US20070275976A1 (en) * 2004-06-26 2007-11-29 Stefan Schnatterer N-phenylpyrazole derivatives as pesticides

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1237873B1 (en) * 1999-12-02 2013-04-03 Merial Limited Control of arthropods in animals
US7262214B2 (en) * 2003-02-26 2007-08-28 Merial Limited 1-N-arylpyrazole derivatives in prevention of arthropod-borne and mosquito-borne diseases

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3966900A (en) * 1969-03-12 1976-06-29 Airwick Industries, Inc. Evaporator system comprising a stabilized pesticidal phosphoric acid ester and method for stabilizing such ester enclosed in an evaporator
US20070275976A1 (en) * 2004-06-26 2007-11-29 Stefan Schnatterer N-phenylpyrazole derivatives as pesticides

Non-Patent Citations (5)

* Cited by examiner, † Cited by third party
Title
BOURGUIGNON J.: "IDENTICAL AND NONIDENTICAL TWIN DRUGS". PRACTICE OF MEDICINAL CHEMISTRY, 1 January 1996 (1996-01-01), pages 261-293, XP001248799, the whole document *
DATABASE BEILSTEIN 1996, XP002575606. Database accession no. 6036932, abstract & COUR, AGNETE LA; FINDEISEN, MATTHIAS; HAZELL, RITA; HENNIG, LOTHAR; OLSEN, CARL ERIK; SIMONSEN, OLE: J. CHEM. SOC., DALTON TRANSACTIONS: INORGANIC CHEMISTRY, vol. 16, 1996, pages 3437-3448 *
DATABASE BEILSTEIN. BEILSTEIN INSTITUTE FOR ORGANIC CHEMISTRY, FRANKFURT-MAIN, DE; 1959, XP002575607. Database accession no. 630245, abstract & FINAR; LORD: J. CHEM. SOC., 1959, pages 1819-1821 *
DATABASE BEILSTEIN. BEILSTEIN INSTITUTE FOR ORGANIC CHEMISTRY, FRANKFURT-MAIN, DE; 1996, XP002575604. Database accession no. 6010790, abstract & NIVOROZHKIN, ALEXANDER L.; TOFTLUND, HANS; JOERGENSEN, PER LAUGE; NIVOROZHKIN, LEONID E.: J. CHEM. SOC., DALTON TRANSACTIONS: INORG. CHEM., vol. 7, 1996, pages 1215-1222 *
DATABASE BEILSTEIN. BEILSTEIN INSTITUTE FOR ORGANIC CHEMISTRY, FRANKFURT-MAIN, DE; 1997, XP002575605. Database accession no. 6206504, abstract & AHLUWALIA, V. K.; SHARMA, POOJA; GOYAL, BINDU: IND. J. CHEM., SECTION B: ORGANIC CHEMISTRY INCLUDING MEDICINAL CHEMISTRY, vol. 36, 1997, pages 1059-1061 *

Also Published As

Publication number Publication date
EP2364300A2 (en) 2011-09-14
NZ592985A (en) 2013-04-26
BRPI0922042A2 (pt) 2016-11-01
JP2012509338A (ja) 2012-04-19
WO2010059719A2 (en) 2010-05-27
BRPI0922042B1 (pt) 2020-01-28
AU2009316710A1 (en) 2010-05-27
MX2011005214A (es) 2011-06-01
CA2743553A1 (en) 2010-05-27
EA201100800A1 (ru) 2011-12-30
EP2364300B1 (en) 2016-10-19
US8642636B2 (en) 2014-02-04
ES2605811T3 (es) 2017-03-16
CA2952443A1 (en) 2010-05-27
WO2010059719A3 (en) 2010-11-18
AU2009316710B2 (en) 2015-08-06
CN102264706A (zh) 2011-11-30
US20110245157A1 (en) 2011-10-06
CA2743553C (en) 2017-03-14
HK1160852A1 (en) 2012-08-17
CA2952443C (en) 2019-04-02

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MM4A Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s)

Designated state(s): AM AZ BY KZ KG MD TJ TM RU