EA002481B1 - Композиция на основе солюбилизированного сертралина - Google Patents

Композиция на основе солюбилизированного сертралина Download PDF

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Publication number
EA002481B1
EA002481B1 EA199900962A EA199900962A EA002481B1 EA 002481 B1 EA002481 B1 EA 002481B1 EA 199900962 A EA199900962 A EA 199900962A EA 199900962 A EA199900962 A EA 199900962A EA 002481 B1 EA002481 B1 EA 002481B1
Authority
EA
Eurasian Patent Office
Prior art keywords
composition
sertraline
solubilizing agent
concentration
matter
Prior art date
Application number
EA199900962A
Other languages
English (en)
Russian (ru)
Other versions
EA199900962A1 (ru
Inventor
Дуэйн Томас Фризен
Скотт Макс Хербиг
Рави Майсор Шенкер
Джеймс Блэр Вест
Original Assignee
Пфайзер Продактс Инк.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=21971159&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=EA002481(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Пфайзер Продактс Инк. filed Critical Пфайзер Продактс Инк.
Publication of EA199900962A1 publication Critical patent/EA199900962A1/ru
Publication of EA002481B1 publication Critical patent/EA002481B1/ru

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0002—Galenical forms characterised by the drug release technique; Application systems commanded by energy
    • A61K9/0004—Osmotic delivery systems; Sustained release driven by osmosis, thermal energy or gas
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2009—Inorganic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/02—Inorganic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/12—Carboxylic acids; Salts or anhydrides thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/14—Esters of carboxylic acids, e.g. fatty acid monoglycerides, medium-chain triglycerides, parabens or PEG fatty acid esters
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/16—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing nitrogen, e.g. nitro-, nitroso-, azo-compounds, nitriles, cyanates
    • A61K47/18—Amines; Amides; Ureas; Quaternary ammonium compounds; Amino acids; Oligopeptides having up to five amino acids
    • A61K47/183—Amino acids, e.g. glycine, EDTA or aspartame

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Inorganic Chemistry (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
EA199900962A 1997-07-01 1998-06-15 Композиция на основе солюбилизированного сертралина EA002481B1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US5141397P 1997-07-01 1997-07-01
PCT/IB1998/000933 WO1999001120A1 (en) 1997-07-01 1998-06-15 Solubilized sertraline compositions

Publications (2)

Publication Number Publication Date
EA199900962A1 EA199900962A1 (ru) 2000-08-28
EA002481B1 true EA002481B1 (ru) 2002-06-27

Family

ID=21971159

Family Applications (1)

Application Number Title Priority Date Filing Date
EA199900962A EA002481B1 (ru) 1997-07-01 1998-06-15 Композиция на основе солюбилизированного сертралина

Country Status (34)

Country Link
EP (1) EP0999829A1 (no)
JP (1) JP2000514100A (no)
KR (1) KR100366373B1 (no)
CN (1) CN1261794A (no)
AP (1) AP1192A (no)
AR (3) AR015917A1 (no)
AU (1) AU742535B2 (no)
BG (1) BG103918A (no)
BR (1) BR9810739A (no)
CA (1) CA2290974C (no)
CO (1) CO4940495A1 (no)
DZ (1) DZ2548A1 (no)
EA (1) EA002481B1 (no)
HN (1) HN1998000102A (no)
HR (1) HRP980377A2 (no)
HU (1) HUP0002236A3 (no)
ID (1) ID23429A (no)
IL (1) IL133076A (no)
IS (1) IS5260A (no)
MA (1) MA24587A1 (no)
NO (1) NO996520L (no)
OA (1) OA11243A (no)
PA (1) PA8454301A1 (no)
PE (1) PE97199A1 (no)
PL (1) PL337804A1 (no)
SK (1) SK181099A3 (no)
TN (1) TNSN98124A1 (no)
TR (1) TR199903297T2 (no)
TW (1) TW550087B (no)
UA (1) UA67741C2 (no)
UY (1) UY25071A1 (no)
WO (1) WO1999001120A1 (no)
YU (1) YU68299A (no)
ZA (1) ZA985708B (no)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GEP20053427B (en) 1999-12-23 2005-01-25 Pfizer Prod Inc Pharmaceutical Compositions Providing Enhanced Drug Concentrations
US20030086972A1 (en) * 2000-08-09 2003-05-08 Appel Leah E. Hydrogel-driven drug dosage form
MXPA03001771A (es) 2000-08-30 2003-06-04 Pfizer Prod Inc Formulaciones de liberacion sostenida para secretagogos de hormona del crecimiento.
US20040191207A1 (en) * 2003-03-31 2004-09-30 Lipari John M. Alpha-hydroxy acid ester drug delivery compositions and methods of use
KR101500020B1 (ko) * 2007-03-12 2015-03-06 디에스엠 아이피 어셋츠 비.브이. 미용 조성물
JPWO2011081117A1 (ja) * 2009-12-29 2013-05-09 興和株式会社 経口投与用固形医薬組成物
CN102711763A (zh) * 2009-12-29 2012-10-03 兴和株式会社 口服用医药组合物
CN109908354A (zh) * 2017-12-12 2019-06-21 万特制药(海南)有限公司 盐酸舍曲林口服浓缩液及其制备工艺

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4803076A (en) * 1986-09-04 1989-02-07 Pfizer Inc. Controlled release device for an active substance
ATE96999T1 (de) * 1989-08-30 1993-11-15 Pfizer Verwendung von sertralin zur behandlung von abhaengigkeiten von chemischen stoffen.
ZA97976B (en) * 1996-04-05 1997-08-18 Alza Corp Uniform drug delivery theraphy.

Also Published As

Publication number Publication date
WO1999001120A1 (en) 1999-01-14
MA24587A1 (fr) 1998-12-31
HN1998000102A (es) 1999-01-08
BG103918A (en) 2000-07-31
HRP980377A2 (en) 1999-04-30
TR199903297T2 (xx) 2000-07-21
AR015917A1 (es) 2001-05-30
IS5260A (is) 1999-11-19
ZA985708B (en) 2000-01-10
BR9810739A (pt) 2000-09-12
AP1192A (en) 2003-07-23
NO996520L (no) 2000-02-29
UA67741C2 (uk) 2004-07-15
HUP0002236A2 (hu) 2003-08-28
SK181099A3 (en) 2000-07-11
OA11243A (en) 2003-07-24
PA8454301A1 (es) 2000-09-29
EA199900962A1 (ru) 2000-08-28
AR040280A2 (es) 2005-03-23
AP9801280A0 (en) 1998-06-30
CN1261794A (zh) 2000-08-02
JP2000514100A (ja) 2000-10-24
IL133076A (en) 2003-12-10
AR040279A2 (es) 2005-03-23
AU7544898A (en) 1999-01-25
DZ2548A1 (fr) 2003-02-08
UY25071A1 (es) 2000-12-29
PE97199A1 (es) 1999-10-05
CO4940495A1 (es) 2000-07-24
PL337804A1 (en) 2000-09-11
CA2290974C (en) 2004-04-27
NO996520D0 (no) 1999-12-28
AU742535B2 (en) 2002-01-03
ID23429A (id) 2000-04-20
HUP0002236A3 (en) 2003-12-29
IL133076A0 (en) 2001-03-19
CA2290974A1 (en) 1999-01-14
KR100366373B1 (ko) 2003-01-14
TNSN98124A1 (fr) 2005-03-15
TW550087B (en) 2003-09-01
EP0999829A1 (en) 2000-05-17
YU68299A (sh) 2002-06-19
KR20010013365A (ko) 2001-02-26

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