DK36489A - Substituerede quinolin-, quinazolin- og cinnolinderivater, fremgangsmaader til deres fremstilling samt deres anvendelse - Google Patents
Substituerede quinolin-, quinazolin- og cinnolinderivater, fremgangsmaader til deres fremstilling samt deres anvendelseInfo
- Publication number
- DK36489A DK36489A DK036489A DK36489A DK36489A DK 36489 A DK36489 A DK 36489A DK 036489 A DK036489 A DK 036489A DK 36489 A DK36489 A DK 36489A DK 36489 A DK36489 A DK 36489A
- Authority
- DK
- Denmark
- Prior art keywords
- quinazoline
- procedures
- preparation
- substituted quinoline
- cinnoline derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
- C07D239/72—Quinazolines; Hydrogenated quinazolines
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/04—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to the ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/18—Halogen atoms or nitro radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/20—Oxygen atoms
- C07D215/22—Oxygen atoms attached in position 2 or 4
- C07D215/233—Oxygen atoms attached in position 2 or 4 only one oxygen atom which is attached in position 4
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/36—Sulfur atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/38—Nitrogen atoms
- C07D215/42—Nitrogen atoms attached in position 4
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/58—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems with hetero atoms directly attached to the ring nitrogen atom
- C07D215/60—N-oxides
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
- C07D239/72—Quinazolines; Hydrogenated quinazolines
- C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
- C07D239/88—Oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
- C07D239/72—Quinazolines; Hydrogenated quinazolines
- C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
- C07D239/93—Sulfur atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
- C07D239/72—Quinazolines; Hydrogenated quinazolines
- C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
- C07D239/94—Nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Quinoline Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US15010388A | 1988-01-29 | 1988-01-29 |
Publications (2)
Publication Number | Publication Date |
---|---|
DK36489D0 DK36489D0 (da) | 1989-01-27 |
DK36489A true DK36489A (da) | 1989-07-30 |
Family
ID=22533132
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DK036489A DK36489A (da) | 1988-01-29 | 1989-01-27 | Substituerede quinolin-, quinazolin- og cinnolinderivater, fremgangsmaader til deres fremstilling samt deres anvendelse |
Country Status (14)
Country | Link |
---|---|
US (1) | US5296484A (fr) |
EP (1) | EP0326328A3 (fr) |
JP (1) | JP2695226B2 (fr) |
KR (1) | KR890011863A (fr) |
CN (1) | CN1034924A (fr) |
AU (1) | AU626280B2 (fr) |
BR (1) | BR8900355A (fr) |
DK (1) | DK36489A (fr) |
FI (1) | FI890422A (fr) |
GT (1) | GT198900008A (fr) |
HU (1) | HU206950B (fr) |
IL (1) | IL89028A0 (fr) |
NZ (1) | NZ227734A (fr) |
ZA (1) | ZA89624B (fr) |
Families Citing this family (90)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IL89026A (en) * | 1988-01-29 | 1993-02-21 | Lilly Co Eli | Substituted quinolines and cinnolines, process for their preparation and fungicidal, insecticidal and miticidal compositions containing them |
IL89029A (en) * | 1988-01-29 | 1993-01-31 | Lilly Co Eli | Fungicidal quinoline and cinnoline derivatives, compositions containing them, and fungicidal methods of using them |
IL89027A (en) * | 1988-01-29 | 1993-01-31 | Lilly Co Eli | Quinazoline derivatives, process for their preparation and fungicidal, insecticidal and miticidal compositions containing them |
EP0365763A1 (fr) * | 1988-09-30 | 1990-05-02 | Agouron Pharmaceuticals, Inc. | Composés cycliques antiproléfératifs |
US5141941A (en) * | 1988-11-21 | 1992-08-25 | Ube Industries, Ltd. | Aralkylamine derivatives, and fungicides containing the same |
CA2011086A1 (fr) * | 1989-03-17 | 1990-09-17 | Karl-Heinz Geiss | 2-alkyl-4-arylmethylaminoquinolines, leur utilisation et medicaments les contenant |
DE3917233A1 (de) * | 1989-05-26 | 1990-11-29 | Basf Ag | 8-substituierte 4-(heterocyclylmethylamino)-chinoline, ihre verwendung und daraus hergestellte arzneimittel |
AT394045B (de) * | 1989-07-05 | 1992-01-27 | Chem Pharm Forsch Gmbh | Neue sulfamoyl-thiophene, verfahren zu ihrer herstellung und ihre verwendung |
JPH0791277B2 (ja) * | 1989-08-04 | 1995-10-04 | 宇部興産株式会社 | アラルキルアミン誘導体、その製法及び殺菌剤 |
NZ234854A (en) * | 1989-08-11 | 1993-02-25 | Ici Plc | Quinoline derivatives, preparation, intermediates and pharmaceutical compositions thereof |
GB2234748B (en) * | 1989-08-11 | 1993-06-30 | Ici Plc | Quinoline derivatives, process for their preparation and their use as medicaments |
EP0424125A3 (en) * | 1989-10-18 | 1991-10-09 | Ube Industries, Ltd. | Aralkylamine derivatives, preparation method thereof and fungicides containing the same |
GB9010394D0 (en) * | 1990-05-09 | 1990-06-27 | Ici Plc | Heterocyclic compounds |
JP3049093B2 (ja) * | 1990-11-19 | 2000-06-05 | ペン・ステイト・リサーチ・フアウンデーション | 殺昆虫剤性、殺ダニ剤性および殺菌・殺カビ剤性のアミノピリミジン類 |
GB9025123D0 (en) * | 1990-11-19 | 1991-01-02 | Ici Plc | Nitrogen compounds |
MX9200299A (es) * | 1991-02-07 | 1992-12-01 | Roussel Uclaf | Nuevos derivados biciclicos nitrogenados, su procedimiento de preparacion los nuevos compuestos intermedios obtenidos su aplicacion como medicamentos y las composiciones farmaceuticas que los contienen. |
GB9102804D0 (en) * | 1991-02-11 | 1991-03-27 | Ici Plc | Heterocyclic derivatives |
US5157040A (en) * | 1991-04-05 | 1992-10-20 | Merck & Co., Inc. | Substituted quinolines as angiotensin ii antagonists |
AU1625192A (en) * | 1991-05-31 | 1992-12-03 | Zeneca Limited | Heterocyclic derivatives |
GB9113626D0 (en) * | 1991-06-25 | 1991-08-14 | Ici Plc | Heterocyclic compounds |
GB9113628D0 (en) * | 1991-06-25 | 1991-08-14 | Ici Plc | Heterocyclic derivatives |
US5399564A (en) * | 1991-09-03 | 1995-03-21 | Dowelanco | N-(4-pyridyl or 4-quinolinyl) arylacetamide and 4-(aralkoxy or aralkylamino) pyridine pesticides |
DE4208254A1 (de) | 1992-03-14 | 1993-09-16 | Hoechst Ag | Substituierte pyrimidine, verfahren zu ihrer herstellung und ihre verwendung als schaedlingsbekaempfungsmittel und fungizid |
AU4790893A (en) * | 1992-08-19 | 1994-03-15 | Dowelanco | Pyridylethoxy-, pyridylethylamino-, and pyridylpropyl-derivatives of quinoline and quinazoline as insecticides and fungicides |
DE4308014A1 (de) * | 1993-03-13 | 1994-09-15 | Hoechst Schering Agrevo Gmbh | Kondensierte Stickstoffheterocyclen, Verfahren zu ihrer Herstellung und ihre Verwendung als Schädlingsbekämpfungsmittel und Fungizide |
DE4321029A1 (de) * | 1993-06-24 | 1995-01-05 | Bayer Ag | Aralkylaminochinazoline |
EP0669324A4 (fr) * | 1993-09-10 | 1996-04-03 | Eisai Co Ltd | Compose de quinazoline. |
DE4331178A1 (de) * | 1993-09-14 | 1995-03-16 | Hoechst Schering Agrevo Gmbh | Substituierte Pyridine und Pyrimidine, Verfahren zu ihrer Herstellung und ihre Verwendung als Schädlingsbekämpfungsmittel und Fungizide |
GB9510757D0 (en) * | 1994-09-19 | 1995-07-19 | Wellcome Found | Therapeuticaly active compounds |
DE4438807A1 (de) * | 1994-10-31 | 1996-05-02 | Hoechst Schering Agrevo Gmbh | Heterocyclyl-amino- und Heterocyclyl-oxy-cycloalkenyl-Derivate, ihre Verwendung als Schädlingsbekämpfungsmittel und Fungizide |
AU6987096A (en) * | 1995-09-12 | 1997-04-01 | Basf Aktiengesellschaft | Fungicidal quinolines |
WO1997042192A1 (fr) * | 1996-05-07 | 1997-11-13 | Basf Aktiengesellschaft | Imidazoquinazolines, agents les contenant et leur utilisation dans la lutte contre les champignons nuisibles et les parasites animaux |
GB9613021D0 (en) * | 1996-06-21 | 1996-08-28 | Pharmacia Spa | Bicyclic 4-aralkylaminopyrimidine derivatives as tyrosine kinase inhibitors |
EP0926139A4 (fr) * | 1996-07-30 | 1999-12-15 | Zenyaku Kogyo Kk | Derives de sulfure de quinoleine |
WO1998005645A1 (fr) * | 1996-08-01 | 1998-02-12 | Dow Agrosciences Llc | Derives de quinoleine 4-substituee dotes d'une activite fongicide |
WO1998005647A1 (fr) * | 1996-08-01 | 1998-02-12 | Dow Agrosciences Llc | Derives de quinolinium ayant une activite fongicide |
WO1998005646A1 (fr) * | 1996-08-01 | 1998-02-12 | Dow Agrosciences Llc | Derives de 1,2-dihydroquinoleine dotes d'une activite fongicide |
EP0927164A1 (fr) | 1996-09-10 | 1999-07-07 | PHARMACIA & UPJOHN COMPANY | 8-hydroxyquinoleines 7-substituees utilisees comme agents antiviraux |
TW521072B (en) | 1997-06-02 | 2003-02-21 | Meiji Seika Kaisha | 4-quinolinol derivatives and fungicides containing the same as an active ingredient used for agriculture and horticulture |
US6117884A (en) * | 1997-07-31 | 2000-09-12 | Daeuble; John | 4-substituted quinoline derivatives having fungicidal activity |
US6686366B1 (en) | 1998-06-02 | 2004-02-03 | Osi Pharmaceuticals, Inc. | Compounds specific to adenosine A3 receptor and uses thereof |
AR020590A1 (es) | 1998-06-02 | 2002-05-22 | Cadus Pharmaceutical Corp | 7-diazapurina-n-6 sustituida, un metodo para su preparacion, composiciones farmaceuticas que la comprenden |
US6878716B1 (en) | 1998-06-02 | 2005-04-12 | Osi Pharmaceuticals, Inc. | Compounds specific to adenosine A1 receptor and uses thereof |
US6184226B1 (en) | 1998-08-28 | 2001-02-06 | Scios Inc. | Quinazoline derivatives as inhibitors of P-38 α |
US7160890B2 (en) * | 1999-12-02 | 2007-01-09 | Osi Pharmaceuticals, Inc. | Compounds specific to adenosine A3 receptor and uses thereof |
US6576644B2 (en) * | 2000-09-06 | 2003-06-10 | Bristol-Myers Squibb Co. | Quinoline inhibitors of cGMP phosphodiesterase |
US6680324B2 (en) * | 2000-12-01 | 2004-01-20 | Osi Pharmaceuticals, Inc. | Compounds specific to adenosine A1 receptors and uses thereof |
US6602884B2 (en) * | 2001-03-13 | 2003-08-05 | Aventis Pharma S.A. | Quinolylpropylpiperidine derivatives, their preparation, and compositions containing them |
EP1381599B1 (fr) * | 2001-04-19 | 2008-09-24 | Astrazeneca AB | Derives quinazoline |
KR100834965B1 (ko) * | 2001-10-10 | 2008-06-03 | 에스케이케미칼주식회사 | 천연 살충 조성물 |
CA2468673C (fr) * | 2001-11-30 | 2011-01-25 | Osi Pharmaceuticals, Inc. | Composes specifiques inhibant les recepteurs a1 et a3 de l'adenosine, et applications desdits composes |
KR20040068317A (ko) | 2001-12-20 | 2004-07-30 | 오에스아이 파마슈티컬스, 인코포레이티드 | 피리미딘 a₂b 선택성 길항 화합물, 그의 합성 방법 및용도 |
WO2004004732A1 (fr) * | 2002-07-09 | 2004-01-15 | Astrazeneca Ab | Derives de quinazoline utilises dans le traitement du cancer |
FR2844268B1 (fr) * | 2002-09-11 | 2004-10-22 | Aventis Pharma Sa | Derives de la quinolyl propyl piperidine, leurs procedes et intermediaires de preparation et les compositions qui les contiennent |
US7932272B2 (en) * | 2003-09-30 | 2011-04-26 | Eisai R&D Management Co., Ltd. | Antifungal agent containing heterocyclic compound |
ES2554330T3 (es) * | 2004-02-19 | 2015-12-18 | Rexahn Pharmaceuticals, Inc. | Derivados de quinazolina y uso terapéutico de los mismos |
US20050241110A1 (en) * | 2004-04-09 | 2005-11-03 | Bruce Baker | Ergonomic handles, especially for garden tools |
WO2006004865A1 (fr) | 2004-06-29 | 2006-01-12 | Rigel Pharmaceuticals, Inc. | Composés de quinoléine de substitution et leurs utilisations comme inhibiteurs de la cascade de signalement du récepteur d'immunoglobuline (ige) |
WO2006013896A1 (fr) * | 2004-08-04 | 2006-02-09 | Meiji Seika Kaisha, Ltd. | Dérivé de quinoline et insecticide contenant celui-ci comme constituant actif |
US20090227799A1 (en) * | 2004-08-09 | 2009-09-10 | Kazutaka Nakamoto | Novel Antimalarial Agent Containing Heterocyclic Compound |
GT200600078A (es) * | 2005-02-17 | 2007-04-12 | Derivados de indol, benzotiofeno, benzofurano e indeno cicloalquil condensados | |
EP1864980A4 (fr) | 2005-03-30 | 2010-08-18 | Eisai R&D Man Co Ltd | Agent antifongique contenant un dérivé de pyridine |
TWI385169B (zh) | 2005-10-31 | 2013-02-11 | Eisai R&D Man Co Ltd | 經雜環取代之吡啶衍生物及含有彼之抗真菌劑 |
US20070265270A1 (en) * | 2006-02-21 | 2007-11-15 | Hitchcock Stephen A | Cinnoline derivatives as phosphodiesterase 10 inhibitors |
JP2009529060A (ja) * | 2006-03-08 | 2009-08-13 | アムゲン インコーポレイティッド | ホスホジエステラーゼ10阻害剤としてのキノリン及びイソキノリン誘導体 |
EP2065377B1 (fr) | 2006-09-21 | 2011-11-23 | Eisai R&D Management Co., Ltd. | Dérivé de pyridine substitué par un cycle hétéroaryle, et agent antifongique le comprenant |
EP2143723A4 (fr) | 2007-04-27 | 2011-05-18 | Eisai R&D Man Co Ltd | Sel d'un dérivé de pyridine substitué par hétérocycle ou cristaux dudit sel |
TW200841879A (en) | 2007-04-27 | 2008-11-01 | Eisai R&D Man Co Ltd | Pyridine derivatives substituted by heterocyclic ring and phosphonoamino group, and anti-fungal agent containing same |
MX352732B (es) * | 2007-06-07 | 2017-12-06 | Bayer Animal Health Gmbh | Control de ectoparasitos. |
US8513287B2 (en) | 2007-12-27 | 2013-08-20 | Eisai R&D Management Co., Ltd. | Heterocyclic ring and phosphonoxymethyl group substituted pyridine derivatives and antifungal agent containing same |
US8268843B2 (en) | 2008-08-29 | 2012-09-18 | Dow Agrosciences, Llc. | 5,8-difluoro-4-(2-(4-(heteroaryloxy)-phenyl)ethylamino)quinazolines and their use as agrochemicals |
US8188119B2 (en) | 2008-10-24 | 2012-05-29 | Eisai R&D Management Co., Ltd | Pyridine derivatives substituted with heterocyclic ring and γ-glutamylamino group, and antifungal agents containing same |
PH12012500097A1 (en) * | 2009-07-21 | 2011-01-27 | Shanghai Inst Organic Chem | Potent small molecule inhibitors of autophagy, and methods of use thereof |
EA201201406A1 (ru) * | 2010-04-15 | 2013-04-30 | Басф Се | Фунгицидные смеси ii, содержащие хиназолины |
CR20120543A (es) * | 2010-04-15 | 2012-11-29 | Basf Se | Mezclas fungicidas ii que comprenden quinazolinas |
WO2013008723A1 (fr) * | 2011-07-08 | 2013-01-17 | 国立大学法人九州大学 | Matrice pour spectroscopie de masse à désorption-ionisation par impact laser assistée par matrice (maldi) |
CN103980209B (zh) * | 2014-05-21 | 2016-03-09 | 贵州大学 | 一种4-n-取代-5-氯喹唑啉类化合物及制备方法及应用 |
CN106187883B (zh) * | 2015-05-07 | 2020-07-07 | 浙江省化工研究院有限公司 | 一类含全氟烷基取代基的喹啉类化合物、其制备方法及应用 |
JP6740354B2 (ja) | 2015-10-05 | 2020-08-12 | ザ トラスティーズ オブ コロンビア ユニバーシティー イン ザ シティー オブ ニューヨーク | オートファジーの流れ及びホスホリパーゼd及びタウを含むタンパク質凝集体のクリアランスの活性化剤ならびにタンパク質症の治療方法 |
US20220235013A1 (en) | 2017-03-21 | 2022-07-28 | Bayer Pharma Aktiengesellschaft | 2-methyl-quinazolines |
JPWO2019065516A1 (ja) * | 2017-09-26 | 2020-09-10 | 日本曹達株式会社 | キノリン化合物および農園芸用殺菌剤 |
CN108299315A (zh) * | 2018-03-01 | 2018-07-20 | 杨子辉 | 一种杀螨剂喹螨醚的制备方法 |
US20220274979A1 (en) | 2018-04-18 | 2022-09-01 | Bayer Pharma Aktiengesellschaft | 2-methyl-aza-quinazolines |
JP2022514692A (ja) * | 2018-12-21 | 2022-02-14 | ユニバーシティ・オブ・ノートル・ダム・デュ・ラック | 抗酸菌症治療のためのbdオキシダーゼ阻害剤の発見 |
CN109721554A (zh) * | 2019-01-08 | 2019-05-07 | 贵州大学 | 一类4-氨基喹唑啉类化合物及其制备方法和应用 |
CN110194761B (zh) * | 2019-07-05 | 2021-08-20 | 华东理工大学 | 喹唑啉基羧酸酯类衍生物及其抗菌用途 |
CN116323623A (zh) | 2020-09-18 | 2023-06-23 | 拜耳公司 | 作为SOS1抑制剂的吡啶并[2,3-d]嘧啶-4-胺 |
EP4074317A1 (fr) | 2021-04-14 | 2022-10-19 | Bayer AG | Dérivés de phosphore en tant que nouveaux inhibiteurs de sos1 |
CN115124462B (zh) * | 2022-07-22 | 2023-08-22 | 浙江工业大学 | 2,3-二甲基-6,8-二氟喹啉-4-醚类化合物及其制备方法和应用 |
CN116003319A (zh) * | 2022-12-02 | 2023-04-25 | 浙江工业大学 | 一种含硫的喹啉类化合物及其制备方法和应用 |
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US3075981A (en) * | 1958-04-03 | 1963-01-29 | Sterling Drug Inc | 1-[aromatic-(lower-alkyl)]-4-(aromaticimino)-1, 4-dihydroquinolines and their preparation |
US3075984A (en) * | 1958-05-09 | 1963-01-29 | Sterling Drug Inc | 1-[(lower-aromatic)-(lower-alkyl)]-4-[(lower-aromatic)-(lower-alkyl) imino]-1, 4-dihydroquinolines and their preparation |
NL265777A (fr) * | 1960-06-09 | |||
US3248292A (en) * | 1963-02-06 | 1966-04-26 | Mead Johnson & Co | Pharmaceutically active dimethoxyquinazolines |
CH492395A (de) * | 1966-04-26 | 1970-06-30 | Sandoz Ag | Mittel zur Bekämpfung von Pflanzenschädlingen und Verwendung des Mittels |
US3470182A (en) * | 1967-02-09 | 1969-09-30 | Sandoz Ag | 4-amino-substituted quinazolines |
DK123301B (da) * | 1968-05-09 | 1972-06-05 | Shionogi & Co | Analogifremgangsmåde til fremstilling af substituerede 2-methyl-2,3-dihydrothieno[3,2-c]-quinoliner eller syreadditionssalte heraf. |
US3800039A (en) * | 1970-10-21 | 1974-03-26 | Mead Johnson & Co | Antithrombogenic process employing substituted 6,7-dialkoxyquinazolines |
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JPS5576803A (en) * | 1978-12-06 | 1980-06-10 | Sankyo Co Ltd | Agent for controlling noxious life |
US4236912A (en) * | 1979-03-05 | 1980-12-02 | The Dow Chemical Company | Quinolinyloxyphenoxy and quinolyinylthiophenoxy alkanoic acids and derivatives thereof and methods of herbicidal use |
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US4522945A (en) * | 1979-10-12 | 1985-06-11 | Janssen Pharmaceutica N.V. | (Piperidinylalkyl) quinazoline derivatives |
AU541697B2 (en) * | 1979-11-19 | 1985-01-17 | Ici Australia Limited | Quinoline derivatives |
DE3028387A1 (de) * | 1980-07-26 | 1982-02-25 | Hoechst Ag, 6000 Frankfurt | Derivate des 1,2,4-triazols und imidazols, verfahren zu ihrer herstellung und ihre verwendung als schaedlingsbekaempfungsmittel |
US4551474A (en) * | 1981-02-19 | 1985-11-05 | Hoechst-Roussel Pharmaceuticals Incorporated | Methods of alleviating convulsions and pain employing 4-aryloxy-1,2,3,4 tetrahydroisoquinolines |
GB2135887A (en) * | 1983-03-08 | 1984-09-12 | Sandoz Ltd | 4-Alkylamino-quinazolines used as insecticides |
JPS6165869A (ja) * | 1984-09-07 | 1986-04-04 | Kyowa Hakko Kogyo Co Ltd | キノリン−n−オキシド誘導体 |
HU211997B (en) * | 1986-01-29 | 1996-01-29 | Sandoz Ag | Process to prepare n-methyl-n-(1-naphtyl-methyl)-4-(2-phenyl-propyl)-benzylamine and pharmaceutical compns. contg. it |
JPS646261A (en) * | 1987-03-31 | 1989-01-10 | Nisshin Flour Milling Co | 4-thioquinazoline derivative, its production and antiulcer agent containing said derivative as active component |
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IL89029A (en) * | 1988-01-29 | 1993-01-31 | Lilly Co Eli | Fungicidal quinoline and cinnoline derivatives, compositions containing them, and fungicidal methods of using them |
IL89026A (en) * | 1988-01-29 | 1993-02-21 | Lilly Co Eli | Substituted quinolines and cinnolines, process for their preparation and fungicidal, insecticidal and miticidal compositions containing them |
IL89027A (en) * | 1988-01-29 | 1993-01-31 | Lilly Co Eli | Quinazoline derivatives, process for their preparation and fungicidal, insecticidal and miticidal compositions containing them |
CA2011086A1 (fr) * | 1989-03-17 | 1990-09-17 | Karl-Heinz Geiss | 2-alkyl-4-arylmethylaminoquinolines, leur utilisation et medicaments les contenant |
-
1989
- 1989-01-23 IL IL89028A patent/IL89028A0/xx unknown
- 1989-01-23 GT GT198900008A patent/GT198900008A/es unknown
- 1989-01-24 AU AU28748/89A patent/AU626280B2/en not_active Ceased
- 1989-01-25 NZ NZ227734A patent/NZ227734A/en unknown
- 1989-01-25 EP EP89300656A patent/EP0326328A3/fr not_active Withdrawn
- 1989-01-26 ZA ZA89624A patent/ZA89624B/xx unknown
- 1989-01-27 KR KR1019890000871A patent/KR890011863A/ko not_active Application Discontinuation
- 1989-01-27 DK DK036489A patent/DK36489A/da unknown
- 1989-01-27 BR BR898900355A patent/BR8900355A/pt not_active IP Right Cessation
- 1989-01-27 CN CN89100470A patent/CN1034924A/zh active Pending
- 1989-01-27 HU HU89424A patent/HU206950B/hu unknown
- 1989-01-27 JP JP1019401A patent/JP2695226B2/ja not_active Expired - Fee Related
- 1989-01-27 FI FI890422A patent/FI890422A/fi not_active Application Discontinuation
- 1989-03-20 US US07/325,734 patent/US5296484A/en not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
GT198900008A (es) | 1990-07-17 |
US5296484A (en) | 1994-03-22 |
AU2874889A (en) | 1989-08-03 |
FI890422A (fi) | 1989-07-30 |
DK36489D0 (da) | 1989-01-27 |
HU206950B (en) | 1993-03-01 |
JPH01246264A (ja) | 1989-10-02 |
EP0326328A3 (fr) | 1990-08-22 |
JP2695226B2 (ja) | 1997-12-24 |
NZ227734A (en) | 1991-11-26 |
IL89028A0 (en) | 1989-08-15 |
FI890422A0 (fi) | 1989-01-27 |
KR890011863A (ko) | 1989-08-23 |
ZA89624B (en) | 1989-12-27 |
HUT49789A (en) | 1989-11-28 |
CN1034924A (zh) | 1989-08-23 |
BR8900355A (pt) | 1989-09-19 |
EP0326328A2 (fr) | 1989-08-02 |
AU626280B2 (en) | 1992-07-30 |
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