DK161080C - Krystallinsk hydrat af oralt anvendeligt cephalosporin og praeparat dermed - Google Patents

Krystallinsk hydrat af oralt anvendeligt cephalosporin og praeparat dermed

Info

Publication number
DK161080C
DK161080C DK336487A DK336487A DK161080C DK 161080 C DK161080 C DK 161080C DK 336487 A DK336487 A DK 336487A DK 336487 A DK336487 A DK 336487A DK 161080 C DK161080 C DK 161080C
Authority
DK
Denmark
Prior art keywords
crystallic
hydrate
preparation
oral
used cephalosporin
Prior art date
Application number
DK336487A
Other languages
Danish (da)
English (en)
Other versions
DK336487D0 (da
DK161080B (da
DK336487A (da
Inventor
Yoshio Hamashima
Kyoji Minami
Kyozo Kawata
Teruo Sakamoto
Toyohiko Takeda
Yusuke Suzuki
Masanori Tujikawa
Original Assignee
Shionogi & Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP61156954A external-priority patent/JP2544113B2/ja
Priority claimed from JP21626086A external-priority patent/JPH0717651B2/ja
Application filed by Shionogi & Co filed Critical Shionogi & Co
Publication of DK336487D0 publication Critical patent/DK336487D0/da
Publication of DK336487A publication Critical patent/DK336487A/da
Publication of DK161080B publication Critical patent/DK161080B/da
Application granted granted Critical
Publication of DK161080C publication Critical patent/DK161080C/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14—Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/542—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/545—Compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins, cefaclor, or cephalexine

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cephalosporin Compounds (AREA)
  • Medicinal Preparation (AREA)
DK336487A 1986-07-02 1987-06-30 Krystallinsk hydrat af oralt anvendeligt cephalosporin og praeparat dermed DK161080C (da)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
JP15695486 1986-07-02
JP61156954A JP2544113B2 (ja) 1986-07-02 1986-07-02 安定なカプセル製剤
JP21626086 1986-09-12
JP21626086A JPH0717651B2 (ja) 1986-09-12 1986-09-12 経口投与用セフアロスポリン水和物結晶

Publications (4)

Publication Number Publication Date
DK336487D0 DK336487D0 (da) 1987-06-30
DK336487A DK336487A (da) 1988-01-03
DK161080B DK161080B (da) 1991-05-27
DK161080C true DK161080C (da) 1991-11-11

Family

ID=26484565

Family Applications (1)

Application Number Title Priority Date Filing Date
DK336487A DK161080C (da) 1986-07-02 1987-06-30 Krystallinsk hydrat af oralt anvendeligt cephalosporin og praeparat dermed

Country Status (27)

Country Link
US (2) US4812561A (OSRAM)
KR (1) KR950005302B1 (OSRAM)
CN (1) CN1015106B (OSRAM)
AR (1) AR243893A1 (OSRAM)
AT (1) AT392472B (OSRAM)
AU (1) AU594167B2 (OSRAM)
BE (1) BE1001691A4 (OSRAM)
CA (1) CA1283405C (OSRAM)
CH (1) CH672788A5 (OSRAM)
DE (1) DE3721913A1 (OSRAM)
DK (1) DK161080C (OSRAM)
ES (2) ES2004952A6 (OSRAM)
FI (1) FI89052C (OSRAM)
FR (1) FR2601014B1 (OSRAM)
GB (1) GB2192183B (OSRAM)
GR (1) GR871014B (OSRAM)
HK (1) HK47893A (OSRAM)
HU (1) HU200777B (OSRAM)
IE (1) IE59613B1 (OSRAM)
IL (1) IL83059A (OSRAM)
IT (1) IT1211469B (OSRAM)
NL (1) NL193136C (OSRAM)
NO (1) NO170889C (OSRAM)
NZ (1) NZ220764A (OSRAM)
PL (1) PL159180B1 (OSRAM)
RU (1) RU1829932C (OSRAM)
SE (1) SE466257B (OSRAM)

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US7842791B2 (en) * 2002-12-19 2010-11-30 Nancy Jean Britten Dispersible pharmaceutical compositions
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US8357394B2 (en) 2005-12-08 2013-01-22 Shionogi Inc. Compositions and methods for improved efficacy of penicillin-type antibiotics
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EP2197842B1 (en) * 2007-08-29 2012-05-23 Schering Corporation 2, 3-substituted indole derivatives for treating viral infections
ES2447543T3 (es) * 2007-08-29 2014-03-12 Merck Sharp & Dohme Corp. Derivados de indol sustituidos y métodos de utilización de los mismos
CA2705586A1 (en) * 2007-11-16 2009-05-22 Schering Corporation 3-heterocyclic substituted indole derivatives and methods of use thereof
EP2222672B1 (en) * 2007-11-16 2013-12-18 Merck Sharp & Dohme Corp. 3-aminosulfonyl substituted indole derivatives and methods of use thereof
WO2009152200A1 (en) * 2008-06-13 2009-12-17 Schering Corporation Tricyclic indole derivatives and methods of use thereof
TW201020245A (en) 2008-08-20 2010-06-01 Schering Corp Ethynyl-substituted pyridine and pyrimidine derivatives and their use in treating viral infections
ES2439009T3 (es) 2008-08-20 2014-01-21 Merck Sharp & Dohme Corp. Derivados de piridina y pirimidina sustituidos con etenilo y su uso en el tratamiento de infecciones virales
WO2010022126A1 (en) 2008-08-20 2010-02-25 Schering Corporation Azo-substituted pyridine and pyrimidine derivatives and their use in treating viral infections
CA2734486A1 (en) 2008-08-20 2010-02-25 Southern Research Institute Substituted pyridine and pyrimidine derivatives and their use in treating viral infections
CA2763140A1 (en) 2009-05-29 2010-12-02 Schering Corporation Antiviral compounds composed of three linked aryl moieties to treat diseases such as hepatitis c
PL2451445T3 (pl) 2009-07-06 2019-09-30 Boehringer Ingelheim International Gmbh Sposób suszenia BIBW2992, jego soli i stałych preparatów farmaceutycznych zawierających tę substancję czynną
AU2010324871A1 (en) 2009-11-25 2012-06-14 Merck Sharp & Dohme Corp. Fused tricyclic compounds and derivatives thereof useful for the treatment of viral diseases
CA2785488A1 (en) 2009-12-22 2011-07-21 Merck Sharp & Dohme Corp. Fused tricyclic compounds and methods of use thereof for the treatment of viral diseases
US9433621B2 (en) 2010-02-18 2016-09-06 Merck Sharp & Dohme Corp. Substituted pyridine and pyrimidine derivatives and their use in treating viral infections
EP2545060B1 (en) 2010-03-09 2015-11-25 Merck Sharp & Dohme Corp. Fused tricyclic silyl compounds and methods of use thereof for the treatment of viral diseases
WO2011139253A2 (en) 2010-05-04 2011-11-10 Mahmut Bilgic Pharmaceutical compositions comprising ceftibuten
WO2012018534A2 (en) 2010-07-26 2012-02-09 Schering Corporation Substituted biphenylene compounds and methods of use thereof for the treatment of viral diseases
EP2621279B1 (en) 2010-09-29 2018-04-04 Merck Sharp & Dohme Corp. Fused tetracycle derivatives and methods of use thereof for the treatment of viral diseases
US9156872B2 (en) 2011-04-13 2015-10-13 Merck Sharp & Dohme Corp. 2′-azido substituted nucleoside derivatives and methods of use thereof for the treatment of viral diseases
EP2696681B1 (en) 2011-04-13 2018-10-03 Merck Sharp & Dohme Corp. 2'-substituted nucleoside derivatives and methods of use thereof for the treatment of viral diseases
WO2013033899A1 (en) 2011-09-08 2013-03-14 Merck Sharp & Dohme Corp. Substituted benzofuran compounds and methods of use thereof for the treatment of viral diseases
WO2013033901A1 (en) 2011-09-08 2013-03-14 Merck Sharp & Dohme Corp. Heterocyclic-substituted benzofuran derivatives and methods of use thereof for the treatment of viral diseases
WO2013033900A1 (en) 2011-09-08 2013-03-14 Merck Sharp & Dohme Corp. Tetracyclic heterocycle compounds and methods of use thereof for the treatment of viral diseases
WO2013039876A1 (en) 2011-09-14 2013-03-21 Merck Sharp & Dohme Corp. Silyl-containing heterocyclic compounds and methods of use thereof for the treatment of viral diseases
WO2013151518A1 (en) * 2012-04-04 2013-10-10 Mahmut Bilgic Capsule formulations comprising ceftibuten
EP2815743A1 (en) 2013-06-21 2014-12-24 Sanovel Ilac Sanayi ve Ticaret A.S. Ceftibuten formulations
US10167298B2 (en) 2013-10-30 2019-01-01 Merck Sharp & Dohme Corp. Pseudopolymorphs of an HCV NS5A inhibitor and uses thereof
US9242965B2 (en) 2013-12-31 2016-01-26 Boehringer Ingelheim International Gmbh Process for the manufacture of (E)-4-N,N-dialkylamino crotonic acid in HX salt form and use thereof for synthesis of EGFR tyrosine kinase inhibitors
CN103948932B (zh) * 2014-04-17 2016-03-16 海南日中天制药有限公司 一种头孢克肟组合物及其制备方法
EP3031450A1 (en) 2014-12-12 2016-06-15 Sanovel Ilac Sanayi ve Ticaret A.S. Ceftibuten capsule compositions
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MY196909A (en) 2016-06-30 2023-05-09 Qpex Biopharma Inc Boronic acid derivatives and therapeutic uses thereof
CN106397454B (zh) * 2016-08-30 2018-08-24 山东罗欣药业集团股份有限公司 一种抗感染药物头孢布烯晶型化合物及其组合物
CN106432270A (zh) * 2016-09-21 2017-02-22 临沂草之美医药科技有限公司 一种制备治疗外科手术感染的药物头孢布烯晶体化合物的方法
CN106397457A (zh) * 2016-09-21 2017-02-15 临沂草之美医药科技有限公司 一种治疗外科手术感染的药物头孢布烯晶体化合物
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Also Published As

Publication number Publication date
HK47893A (en) 1993-05-27
PL159180B1 (pl) 1992-11-30
KR950005302B1 (ko) 1995-05-23
GR871014B (en) 1987-11-02
FR2601014B1 (fr) 1990-09-14
KR880001670A (ko) 1988-04-26
IT1211469B (it) 1989-11-03
CH672788A5 (OSRAM) 1989-12-29
ES2004952A6 (es) 1989-02-16
GB8715064D0 (en) 1987-08-05
PL266567A1 (en) 1988-07-21
FI872903A0 (fi) 1987-07-01
AU7504087A (en) 1988-01-07
GB2192183B (en) 1990-05-16
ES2008759A6 (es) 1989-08-01
FI89052C (fi) 1993-08-10
IL83059A0 (en) 1987-12-31
BE1001691A4 (fr) 1990-02-13
IE871738L (en) 1988-01-02
SE8702705L (sv) 1988-01-03
HU200777B (en) 1990-08-28
DE3721913A1 (de) 1988-01-07
NL8701507A (nl) 1988-02-01
IE59613B1 (en) 1994-03-09
ATA165887A (de) 1990-09-15
NZ220764A (en) 1989-09-27
AU594167B2 (en) 1990-03-01
NO872729L (no) 1988-01-04
DK336487D0 (da) 1987-06-30
RU1829932C (ru) 1993-07-23
CN1015106B (zh) 1991-12-18
CN87105009A (zh) 1988-03-23
CA1283405C (en) 1991-04-23
FI872903L (fi) 1988-01-03
HUT44257A (en) 1988-02-29
US4812561A (en) 1989-03-14
IT8767566A0 (it) 1987-07-01
FR2601014A1 (fr) 1988-01-08
IL83059A (en) 1992-03-29
NL193136C (nl) 1998-12-04
NO170889C (no) 1992-12-23
SE8702705D0 (sv) 1987-06-30
DK161080B (da) 1991-05-27
US4933443A (en) 1990-06-12
NL193136B (nl) 1998-08-03
FI89052B (fi) 1993-04-30
NO170889B (no) 1992-09-14
NO872729D0 (no) 1987-06-30
AR243893A1 (es) 1993-09-30
GB2192183A (en) 1988-01-06
DK336487A (da) 1988-01-03
AT392472B (de) 1991-04-10
SE466257B (sv) 1992-01-20

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