DK149628C - Analogifremgangsmaade til fremstilling af 8-substitueret-4ae-amino-makrolider eller syreadditionssalte deraf - Google Patents

Analogifremgangsmaade til fremstilling af 8-substitueret-4ae-amino-makrolider eller syreadditionssalte deraf

Info

Publication number
DK149628C
DK149628C DK51778A DK51778A DK149628C DK 149628 C DK149628 C DK 149628C DK 51778 A DK51778 A DK 51778A DK 51778 A DK51778 A DK 51778A DK 149628 C DK149628 C DK 149628C
Authority
DK
Denmark
Prior art keywords
analogue
substituted
preparation
acid addition
addition salts
Prior art date
Application number
DK51778A
Other languages
Danish (da)
English (en)
Other versions
DK149628B (da
DK51778A (da
Inventor
Frank Christian Sciavolino
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of DK51778A publication Critical patent/DK51778A/da
Publication of DK149628B publication Critical patent/DK149628B/da
Application granted granted Critical
Publication of DK149628C publication Critical patent/DK149628C/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
DK51778A 1977-02-04 1978-02-03 Analogifremgangsmaade til fremstilling af 8-substitueret-4ae-amino-makrolider eller syreadditionssalte deraf DK149628C (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US05/765,486 US4125705A (en) 1977-02-04 1977-02-04 Semi-synthetic 4-amino-oleandomycin derivatives
US76548677 1977-02-04

Publications (3)

Publication Number Publication Date
DK51778A DK51778A (da) 1978-08-05
DK149628B DK149628B (da) 1986-08-18
DK149628C true DK149628C (da) 1987-02-02

Family

ID=25073683

Family Applications (1)

Application Number Title Priority Date Filing Date
DK51778A DK149628C (da) 1977-02-04 1978-02-03 Analogifremgangsmaade til fremstilling af 8-substitueret-4ae-amino-makrolider eller syreadditionssalte deraf

Country Status (34)

Country Link
US (1) US4125705A (ja)
JP (2) JPS5398981A (ja)
AR (1) AR215666A1 (ja)
AT (1) AT358169B (ja)
AU (1) AU502293B1 (ja)
BE (1) BE863618A (ja)
BG (2) BG32116A3 (ja)
CA (1) CA1106366A (ja)
CH (1) CH629821A5 (ja)
CS (3) CS200536B2 (ja)
DD (1) DD134523A5 (ja)
DE (1) DE2804509C2 (ja)
DK (1) DK149628C (ja)
ES (1) ES465322A1 (ja)
FI (1) FI65262C (ja)
FR (2) FR2383964A1 (ja)
GB (1) GB1583921A (ja)
GR (1) GR68692B (ja)
HU (2) HU181395B (ja)
IE (1) IE46395B1 (ja)
IL (2) IL53959A0 (ja)
IT (1) IT1094211B (ja)
LU (1) LU79007A1 (ja)
NL (1) NL175997C (ja)
NO (2) NO145955C (ja)
NZ (1) NZ186384A (ja)
PH (2) PH14836A (ja)
PL (3) PL113163B1 (ja)
PT (1) PT67569B (ja)
RO (3) RO79264A (ja)
SE (2) SE445222B (ja)
SU (3) SU805949A3 (ja)
YU (3) YU39504B (ja)
ZA (1) ZA78646B (ja)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4133950A (en) * 1978-01-03 1979-01-09 Pfizer Inc. 4"-Deoxy-4"-carbamate and dithiocarbamate derivatives of oleandomycin and its esters
US4124755A (en) * 1978-01-03 1978-11-07 Pfizer Inc. 11-Alkanoyl-4"-deoxy-4"-isonitrilo-oleandomycin derivatives
US4363803A (en) * 1982-03-01 1982-12-14 Pfizer Inc. 3",4"-Oxyallylene erythromycin and oleandomycin, composition and method of use
US4413119A (en) * 1982-03-01 1983-11-01 Pfizer Inc. Semi-synthetic macrolides
JPH0240447U (ja) * 1988-09-14 1990-03-19
US5141926A (en) * 1990-04-18 1992-08-25 Abbott Laboratories Erythromycin derivatives
JPH05155896A (ja) * 1991-01-18 1993-06-22 Yamanouchi Pharmaceut Co Ltd 新規マクロライド化合物及びその製造法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3022219A (en) * 1958-03-07 1962-02-20 Pfizer & Co C Acyl esters of oleandomycin
US3179652A (en) * 1961-09-05 1965-04-20 Pfizer & Co C Antibiotic recovery process and salts produced thereby
US3836519A (en) * 1973-05-04 1974-09-17 Abbott Lab Sulfonyl derivatives of erythromycin
US3842069A (en) * 1973-06-21 1974-10-15 Abbott Lab 4"-deoxy-4"-oxoerythromycin b derivatives
US4036853A (en) * 1976-08-06 1977-07-19 Pfizer Inc. Semi-synthetic oleandomycin derivatives-C8 modifications

Also Published As

Publication number Publication date
JPS56135497A (en) 1981-10-22
SE445222B (sv) 1986-06-09
PL204041A1 (pl) 1979-06-04
NO780390L (no) 1978-08-07
CS200538B2 (en) 1980-09-15
CH629821A5 (fr) 1982-05-14
IT1094211B (it) 1985-07-26
FI65262B (fi) 1983-12-30
FI780355A (fi) 1978-08-05
BG32117A4 (en) 1982-05-14
RO79258A (ro) 1982-06-25
YU39518B (en) 1984-12-31
YU300377A (en) 1982-10-31
JPS5398981A (en) 1978-08-29
DE2804509A1 (de) 1978-08-10
SE8300869D0 (sv) 1983-02-16
JPS5652036B2 (ja) 1981-12-09
NL175997C (nl) 1985-02-01
AT358169B (de) 1980-08-25
FR2396022B1 (ja) 1980-06-13
YU151782A (en) 1982-10-31
SE457085B (sv) 1988-11-28
CA1106366A (en) 1981-08-04
YU151882A (en) 1982-10-31
BE863618A (fr) 1978-08-03
ZA78646B (en) 1978-12-27
NL175997B (nl) 1984-09-03
CS200537B2 (en) 1980-09-15
FR2396022A1 (fr) 1979-01-26
GR68692B (ja) 1982-02-01
DD134523A5 (de) 1979-03-07
LU79007A1 (fr) 1979-09-06
BG32116A3 (en) 1982-05-14
US4125705A (en) 1978-11-14
HU181395B (en) 1983-07-28
DK149628B (da) 1986-08-18
PL110793B1 (en) 1980-07-31
AR215666A1 (es) 1979-10-31
PH16491A (en) 1983-10-28
RO79264A (ro) 1982-06-25
IT7820006A0 (it) 1978-02-03
PL113163B1 (en) 1980-11-29
FI65262C (fi) 1984-04-10
AU502293B1 (en) 1979-07-19
NO150439B (no) 1984-07-09
FR2383964B1 (ja) 1981-11-27
IE780240L (en) 1978-08-04
ES465322A1 (es) 1978-09-16
ATA72078A (de) 1980-01-15
JPS5827799B2 (ja) 1983-06-11
NZ186384A (en) 1980-08-26
PL111160B1 (en) 1980-08-30
SU888824A3 (ru) 1981-12-07
FR2383964A1 (fr) 1978-10-13
YU39517B (en) 1984-12-31
RO75387A (ro) 1980-11-30
NO811914L (no) 1978-08-07
SU1020004A3 (ru) 1983-05-23
SU805949A3 (ru) 1981-02-15
YU39504B (en) 1984-12-31
IL53959A0 (en) 1978-04-30
IL61606A0 (en) 1981-01-30
DE2804509C2 (de) 1982-12-02
NO150439C (no) 1984-10-17
SE7800269L (sv) 1978-08-05
IE46395B1 (en) 1983-06-01
DK51778A (da) 1978-08-05
GB1583921A (en) 1981-02-04
NO145955B (no) 1982-03-22
PT67569B (en) 1979-06-18
PH14836A (en) 1981-12-16
PT67569A (en) 1978-02-01
NO145955C (no) 1982-06-30
NL7801259A (nl) 1978-08-08
CS200536B2 (en) 1980-09-15
HU179744B (en) 1982-12-28

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