DK148903C - Analogifremgangsmaade til fremstilling af enkephalin-analoge pentapeptidderivater eller syreadditionssalte deraf - Google Patents

Analogifremgangsmaade til fremstilling af enkephalin-analoge pentapeptidderivater eller syreadditionssalte deraf

Info

Publication number
DK148903C
DK148903C DK316981A DK316981A DK148903C DK 148903 C DK148903 C DK 148903C DK 316981 A DK316981 A DK 316981A DK 316981 A DK316981 A DK 316981A DK 148903 C DK148903 C DK 148903C
Authority
DK
Denmark
Prior art keywords
analogue
preparation
acid addition
addition salts
enkephalin
Prior art date
Application number
DK316981A
Other languages
English (en)
Other versions
DK148903B (da
DK316981A (da
Inventor
Francois Cardinaux
Rene Huguenin
Janos Pless
Original Assignee
Sandoz Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sandoz Ag filed Critical Sandoz Ag
Publication of DK316981A publication Critical patent/DK316981A/da
Publication of DK148903B publication Critical patent/DK148903B/da
Application granted granted Critical
Publication of DK148903C publication Critical patent/DK148903C/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/665—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans derived from pro-opiomelanocortin, pro-enkephalin or pro-dynorphin
    • C07K14/70—Enkephalins
    • C07K14/702—Enkephalins with at least 1 amino acid in D-form
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
DK316981A 1980-07-17 1981-07-15 Analogifremgangsmaade til fremstilling af enkephalin-analoge pentapeptidderivater eller syreadditionssalte deraf DK148903C (da)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
CH548380 1980-07-17
CH548380 1980-07-17
CH875280 1980-11-26
CH875280 1980-11-26

Publications (3)

Publication Number Publication Date
DK316981A DK316981A (da) 1982-01-18
DK148903B DK148903B (da) 1985-11-11
DK148903C true DK148903C (da) 1986-04-14

Family

ID=25697814

Family Applications (1)

Application Number Title Priority Date Filing Date
DK316981A DK148903C (da) 1980-07-17 1981-07-15 Analogifremgangsmaade til fremstilling af enkephalin-analoge pentapeptidderivater eller syreadditionssalte deraf

Country Status (16)

Country Link
US (1) US4405607A (da)
EP (1) EP0044451B1 (da)
AU (1) AU547471B2 (da)
CA (1) CA1242702A (da)
CS (1) CS228513B2 (da)
DE (1) DE3163199D1 (da)
DK (1) DK148903C (da)
ES (1) ES503993A0 (da)
FI (1) FI812190L (da)
GR (1) GR74300B (da)
IE (1) IE51967B1 (da)
IL (1) IL63323A (da)
NZ (1) NZ197736A (da)
PH (1) PH17257A (da)
PT (1) PT73374B (da)
YU (1) YU174981A (da)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4495178A (en) * 1983-10-06 1985-01-22 G. D. Searle & Co. Enkephalin analogs
US4599325A (en) * 1984-02-16 1986-07-08 G. D. Searle & Co. Substituted tyrosyl alanine dipeptide amides
JPH0680079B2 (ja) * 1984-11-09 1994-10-12 エーザイ株式会社 ポリペプチド
US4822775A (en) * 1986-02-14 1989-04-18 G. D. Searle & Co. Phenyl substituted dipeptide amides
US4880829A (en) * 1985-08-14 1989-11-14 G. D. Searle And Company Substituted dipeptide amides #3
US4758675A (en) * 1986-07-14 1988-07-19 G. D. Searle & Co. 3-thiophene-substituted tyrosyl dipeptide amides
US6297354B1 (en) 1998-08-12 2001-10-02 Abbott Laboratories Pentapeptide LHRH antagonists
WO2005007628A1 (en) 2003-07-11 2005-01-27 Bristol-Myers Squibb Company Tetrahydroquinoline derivatives as cannabinoid receptor modulators

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2338925A1 (fr) * 1976-01-26 1977-08-19 Wellcome Found Nouveaux peptides et medicament contenant ces substances
US4261888A (en) * 1976-04-12 1981-04-14 Sandoz Ltd. Organic compounds
DE2819277A1 (de) * 1977-05-16 1978-11-23 Sandoz Ag Neue polypeptidderivate, ihre herstellung und verwendung
GB1604850A (en) * 1977-11-24 1981-12-16 Wellcome Found Biologically active peptides
US4199499A (en) * 1978-08-24 1980-04-22 Eli Lilly And Company Pharmacologically active peptides
CA1175810A (en) * 1979-03-30 1984-10-09 Frank A. Momany Synthetic peptides having pituitary growth hormone releasing activity
DE2941790A1 (de) * 1979-10-16 1981-04-30 Hoechst Ag, 6000 Frankfurt Verwendung motilitaetssteigernder peptide
US4254023A (en) * 1979-10-16 1981-03-03 Pennwalt Corporation Synthesis of peptide alcohols by the solid phase method
US4251439A (en) * 1979-12-17 1981-02-17 Eli Lilly And Company Pharmacologically active peptides
US4283329A (en) * 1979-12-17 1981-08-11 Eli Lilly And Company Pharmacologically active peptides
US4322339A (en) * 1980-10-20 1982-03-30 Eli Lilly And Company Pharmacologically active peptides

Also Published As

Publication number Publication date
IE811601L (en) 1982-01-17
PH17257A (en) 1984-07-03
NZ197736A (en) 1985-04-30
CA1242702A (en) 1988-10-04
US4405607A (en) 1983-09-20
EP0044451A1 (en) 1982-01-27
IL63323A (en) 1985-08-30
PT73374A (en) 1981-08-01
PT73374B (en) 1983-01-13
DK148903B (da) 1985-11-11
ES8300685A1 (es) 1982-11-01
YU174981A (en) 1983-09-30
GR74300B (da) 1984-06-21
ES503993A0 (es) 1982-11-01
CS228513B2 (en) 1984-05-14
DE3163199D1 (en) 1984-05-24
FI812190L (fi) 1982-01-18
DK316981A (da) 1982-01-18
EP0044451B1 (en) 1984-04-18
IL63323A0 (en) 1981-10-30
AU7289381A (en) 1982-01-21
IE51967B1 (en) 1987-05-13
AU547471B2 (en) 1985-10-24

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Legal Events

Date Code Title Description
AHB Application shelved due to non-payment
PBP Patent lapsed