CS228513B2 - Method for the production of pentapeptide - Google Patents

Method for the production of pentapeptide Download PDF

Info

Publication number
CS228513B2
CS228513B2 CS815449A CS544981A CS228513B2 CS 228513 B2 CS228513 B2 CS 228513B2 CS 815449 A CS815449 A CS 815449A CS 544981 A CS544981 A CS 544981A CS 228513 B2 CS228513 B2 CS 228513B2
Authority
CS
Czechoslovakia
Prior art keywords
group
formula
hydrogen
radical
ala
Prior art date
Application number
CS815449A
Other languages
Czech (cs)
English (en)
Inventor
Francois Dr Cardinaux
Rene Dr Huguenin
Janos Dr Pless
Original Assignee
Sandoz Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sandoz Ag filed Critical Sandoz Ag
Priority to CS818108A priority Critical patent/CS228546B2/cs
Priority to CS828110A priority patent/CS228548B2/cs
Priority to CS828109A priority patent/CS228547B2/cs
Publication of CS228513B2 publication Critical patent/CS228513B2/cs

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/665—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans derived from pro-opiomelanocortin, pro-enkephalin or pro-dynorphin
    • C07K14/70—Enkephalins
    • C07K14/702—Enkephalins with at least 1 amino acid in D-form
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Zoology (AREA)
  • Genetics & Genomics (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Toxicology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
CS815449A 1980-07-17 1981-07-16 Method for the production of pentapeptide CS228513B2 (en)

Priority Applications (3)

Application Number Priority Date Filing Date Title
CS818108A CS228546B2 (cs) 1980-07-17 1981-07-16 Způsob výroby pentapeptidů
CS828110A CS228548B2 (cs) 1980-07-17 1982-11-15 Způsob výroby pentapeptidů
CS828109A CS228547B2 (cs) 1980-11-26 1982-11-15 Způsob výroby pentapeptidů

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH548380 1980-07-17
CH875280 1980-11-26

Publications (1)

Publication Number Publication Date
CS228513B2 true CS228513B2 (en) 1984-05-14

Family

ID=25697814

Family Applications (1)

Application Number Title Priority Date Filing Date
CS815449A CS228513B2 (en) 1980-07-17 1981-07-16 Method for the production of pentapeptide

Country Status (16)

Country Link
US (1) US4405607A (da)
EP (1) EP0044451B1 (da)
AU (1) AU547471B2 (da)
CA (1) CA1242702A (da)
CS (1) CS228513B2 (da)
DE (1) DE3163199D1 (da)
DK (1) DK148903C (da)
ES (1) ES503993A0 (da)
FI (1) FI812190L (da)
GR (1) GR74300B (da)
IE (1) IE51967B1 (da)
IL (1) IL63323A (da)
NZ (1) NZ197736A (da)
PH (1) PH17257A (da)
PT (1) PT73374B (da)
YU (1) YU174981A (da)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4495178A (en) * 1983-10-06 1985-01-22 G. D. Searle & Co. Enkephalin analogs
US4599325A (en) * 1984-02-16 1986-07-08 G. D. Searle & Co. Substituted tyrosyl alanine dipeptide amides
JPH0680079B2 (ja) * 1984-11-09 1994-10-12 エーザイ株式会社 ポリペプチド
US4822775A (en) * 1986-02-14 1989-04-18 G. D. Searle & Co. Phenyl substituted dipeptide amides
US4880829A (en) * 1985-08-14 1989-11-14 G. D. Searle And Company Substituted dipeptide amides #3
US4758675A (en) * 1986-07-14 1988-07-19 G. D. Searle & Co. 3-thiophene-substituted tyrosyl dipeptide amides
US6297354B1 (en) 1998-08-12 2001-10-02 Abbott Laboratories Pentapeptide LHRH antagonists
US7276608B2 (en) 2003-07-11 2007-10-02 Bristol-Myers Squibb Company Tetrahydroquinoline derivatives as cannabinoid receptor modulators

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH644352A5 (en) * 1976-01-26 1984-07-31 Wellcome Found Process for the preparation of peptides
US4261888A (en) * 1976-04-12 1981-04-14 Sandoz Ltd. Organic compounds
DE2819277A1 (de) * 1977-05-16 1978-11-23 Sandoz Ag Neue polypeptidderivate, ihre herstellung und verwendung
GB1604850A (en) * 1977-11-24 1981-12-16 Wellcome Found Biologically active peptides
US4199499A (en) * 1978-08-24 1980-04-22 Eli Lilly And Company Pharmacologically active peptides
CA1175810A (en) * 1979-03-30 1984-10-09 Frank A. Momany Synthetic peptides having pituitary growth hormone releasing activity
US4254023A (en) * 1979-10-16 1981-03-03 Pennwalt Corporation Synthesis of peptide alcohols by the solid phase method
DE2941790A1 (de) * 1979-10-16 1981-04-30 Hoechst Ag, 6000 Frankfurt Verwendung motilitaetssteigernder peptide
US4283329A (en) * 1979-12-17 1981-08-11 Eli Lilly And Company Pharmacologically active peptides
US4251439A (en) * 1979-12-17 1981-02-17 Eli Lilly And Company Pharmacologically active peptides
US4322339A (en) * 1980-10-20 1982-03-30 Eli Lilly And Company Pharmacologically active peptides

Also Published As

Publication number Publication date
DK316981A (da) 1982-01-18
ES8300685A1 (es) 1982-11-01
YU174981A (en) 1983-09-30
EP0044451A1 (en) 1982-01-27
DK148903C (da) 1986-04-14
CA1242702A (en) 1988-10-04
ES503993A0 (es) 1982-11-01
IE811601L (en) 1982-01-17
PH17257A (en) 1984-07-03
DE3163199D1 (en) 1984-05-24
PT73374B (en) 1983-01-13
IL63323A (en) 1985-08-30
US4405607A (en) 1983-09-20
GR74300B (da) 1984-06-21
EP0044451B1 (en) 1984-04-18
NZ197736A (en) 1985-04-30
AU547471B2 (en) 1985-10-24
IE51967B1 (en) 1987-05-13
FI812190L (fi) 1982-01-18
DK148903B (da) 1985-11-11
IL63323A0 (en) 1981-10-30
PT73374A (en) 1981-08-01
AU7289381A (en) 1982-01-21

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