DK149106C - Analogifremgangsmaade til fremstilling af 1,2,4-oxadiazinderivater eller farmaceutisk acceptable syreadditionssalte eller kvaternaere salte deraf samt 1,2,4-oxadiazolin-5-oner til anvendelse ved fremgangsmaaden - Google Patents

Analogifremgangsmaade til fremstilling af 1,2,4-oxadiazinderivater eller farmaceutisk acceptable syreadditionssalte eller kvaternaere salte deraf samt 1,2,4-oxadiazolin-5-oner til anvendelse ved fremgangsmaaden

Info

Publication number
DK149106C
DK149106C DK429680A DK429680A DK149106C DK 149106 C DK149106 C DK 149106C DK 429680 A DK429680 A DK 429680A DK 429680 A DK429680 A DK 429680A DK 149106 C DK149106 C DK 149106C
Authority
DK
Denmark
Prior art keywords
oxadiazoline
oer
analogue
preparation
pharmaceutically acceptable
Prior art date
Application number
DK429680A
Other languages
Danish (da)
English (en)
Other versions
DK429680A (da
DK149106B (da
Inventor
Kalman Takacs
Ilona Kiss
Antal Simay
Peter Literaty Nagy
Maria Hetyey
Marian Ecsery
Jozsef Szegi
Sandor Viragh
Sandor Juhasz Nagy
Original Assignee
Chinoin Gyogyszer Es Vegyeszet
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Chinoin Gyogyszer Es Vegyeszet filed Critical Chinoin Gyogyszer Es Vegyeszet
Publication of DK429680A publication Critical patent/DK429680A/da
Publication of DK149106B publication Critical patent/DK149106B/da
Application granted granted Critical
Publication of DK149106C publication Critical patent/DK149106C/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D273/00Heterocyclic compounds containing rings having nitrogen and oxygen atoms as the only ring hetero atoms, not provided for by groups C07D261/00 - C07D271/00
    • C07D273/02Heterocyclic compounds containing rings having nitrogen and oxygen atoms as the only ring hetero atoms, not provided for by groups C07D261/00 - C07D271/00 having two nitrogen atoms and only one oxygen atom
    • C07D273/04Six-membered rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/10Antioedematous agents; Diuretics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/08Vasodilators for multiple indications
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
DK429680A 1979-10-11 1980-10-10 Analogifremgangsmaade til fremstilling af 1,2,4-oxadiazinderivater eller farmaceutisk acceptable syreadditionssalte eller kvaternaere salte deraf samt 1,2,4-oxadiazolin-5-oner til anvendelse ved fremgangsmaaden DK149106C (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
HU79CI1914A HU180708B (en) 1979-10-11 1979-10-11 Process for preparing new 1,2,4-oxadiazine derivatives
HUCI001974 1979-10-11

Publications (3)

Publication Number Publication Date
DK429680A DK429680A (da) 1981-04-12
DK149106B DK149106B (da) 1986-01-27
DK149106C true DK149106C (da) 1986-06-09

Family

ID=10994765

Family Applications (1)

Application Number Title Priority Date Filing Date
DK429680A DK149106C (da) 1979-10-11 1980-10-10 Analogifremgangsmaade til fremstilling af 1,2,4-oxadiazinderivater eller farmaceutisk acceptable syreadditionssalte eller kvaternaere salte deraf samt 1,2,4-oxadiazolin-5-oner til anvendelse ved fremgangsmaaden

Country Status (25)

Country Link
US (1) US4308270A (fr)
JP (1) JPS5663970A (fr)
AT (1) AT373247B (fr)
BE (1) BE885634A (fr)
CA (1) CA1159828A (fr)
CH (1) CH649540A5 (fr)
CS (1) CS249111B2 (fr)
DD (1) DD153551A5 (fr)
DE (1) DE3037747A1 (fr)
DK (1) DK149106C (fr)
ES (1) ES495820A0 (fr)
FR (1) FR2467204B1 (fr)
GB (1) GB2062628B (fr)
GR (1) GR71205B (fr)
HU (1) HU180708B (fr)
IL (1) IL61176A (fr)
IT (1) IT1129306B (fr)
LU (1) LU82823A1 (fr)
NL (1) NL8005587A (fr)
NO (1) NO153652C (fr)
PL (2) PL129081B1 (fr)
RO (3) RO85269B (fr)
SE (1) SE448234B (fr)
SU (1) SU1087520A1 (fr)
YU (2) YU41739B (fr)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HU179951B (en) * 1979-10-11 1983-01-28 Chinoin Gyogyszer Es Vegyeszet Process for preparing 1,2,4-oxadiazolin-5-one derivatives and pharmaceutical compositions containing thereof
EP1622883A4 (fr) * 2003-04-10 2008-04-02 Cytokinetics Inc Composes, compositions, et procedes
WO2017031325A1 (fr) * 2015-08-18 2017-02-23 Forum Pharmaceuticals Inc. Composés d'oxadiazine et leurs procédés d'utilisation

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL132134C (fr) * 1963-03-22
DE1795839C3 (de) * 1964-03-02 1981-09-03 Chinoin Gyógyszer és Vegyészeti Termékek Gyára RT, 1045 Budapest Verfahren zur Herstellung von 3,5-disubstituierten 1,2,4-Oxadiazolderivaten
DE1545658C3 (de) * 1964-03-02 1981-04-23 Chinoin Gyógyszer és Vegyészeti Termékek Gyára RT, 1045 Budapest Verfahren zur Herstellung von 3,5-disubstituierten 1,2,4-Oxadiazolderivaten
IT1043838B (it) * 1971-04-22 1980-02-29 Poli Ind Chimica Spa 1 2 3 4 tetraidroisochinoline e processo per la loro preparazione
US4154598A (en) * 1975-09-11 1979-05-15 Philagro Herbicidal 1,2,4-oxadiazin-5-one compositions
US4026894A (en) * 1975-10-14 1977-05-31 Abbott Laboratories Antihypertensive agents
HU179951B (en) * 1979-10-11 1983-01-28 Chinoin Gyogyszer Es Vegyeszet Process for preparing 1,2,4-oxadiazolin-5-one derivatives and pharmaceutical compositions containing thereof

Also Published As

Publication number Publication date
RO85269A (fr) 1984-09-29
SU1087520A1 (ru) 1984-04-23
ES8106714A1 (es) 1981-09-16
LU82823A1 (de) 1981-02-02
ATA501280A (de) 1983-05-15
IT1129306B (it) 1986-06-04
US4308270A (en) 1981-12-29
GB2062628A (en) 1981-05-28
GR71205B (fr) 1983-04-11
YU42063B (en) 1988-04-30
ES495820A0 (es) 1981-09-16
SE448234B (sv) 1987-02-02
DE3037747A1 (de) 1981-06-11
YU41739B (en) 1987-12-31
PL129081B1 (en) 1984-03-31
DK429680A (da) 1981-04-12
RO81210A (fr) 1983-02-01
YU259580A (en) 1983-04-30
PL227211A1 (fr) 1981-11-27
CH649540A5 (de) 1985-05-31
IL61176A0 (en) 1980-11-30
RO85268A (fr) 1984-09-29
HU180708B (en) 1983-04-29
RO81210B (ro) 1983-01-30
PL232264A1 (fr) 1982-03-29
CA1159828A (fr) 1984-01-03
NL8005587A (nl) 1981-04-14
GB2062628B (en) 1983-08-03
DD153551A5 (de) 1982-01-13
YU291182A (en) 1983-04-30
FR2467204B1 (fr) 1986-03-28
NO803045L (no) 1981-04-13
RO85268B (ro) 1984-10-30
CS249111B2 (en) 1987-03-12
IT8068556A0 (it) 1980-10-09
AT373247B (de) 1983-12-27
PL129378B1 (en) 1984-05-31
IL61176A (en) 1984-05-31
NO153652B (no) 1986-01-20
JPH0215547B2 (fr) 1990-04-12
SE8007026L (sv) 1981-04-12
RO85269B (ro) 1984-10-30
BE885634A (fr) 1981-02-02
FR2467204A1 (fr) 1981-04-17
NO153652C (no) 1986-05-07
DK149106B (da) 1986-01-27
JPS5663970A (en) 1981-05-30

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